
Nolvadex (tamoxify citrate) rau CAS ntawm lub cev CAS: 54965-24-1
Tsis pub dhau lub inricate tshuaj ntawm kev ua tiav, nolvadeex (tamoxifalex (tam sim no muaj kev sib txawv thiab tseem ceeb, txawm yog daim ntawv lo, niche. Tsis zoo li cov tshuaj scabolic uas tsav cov leeg txoj kev loj hlob ncaj qha, cov lus estrogen muaj zog, kev xaiv tshuaj estrogen uas muaj qhov xav tau tshuaj estrogen rau hauv anabolic steroid siv. Nkag siab txog cov khoom siv, kev siv, thiab cov kev txwv, thiab cov kev txwv tsis muaj kev sib tw ntawm cov neeg ua haujlwm hormonal.
Dab tsi yog nolvadex (tamoxify citrate) hmoov?
Tus Kheej Tus Kheej:Tamoxifen citrate yog cov kua zaub ntsev npuaj ntawm tamoxifen, tsis yog - stergoidal compound ua tus xaiv tshuaj estrogen (cov tub ki). Nws yogtsisSCOIDCOOLIC, AROMATIVE ARIBITOR (AI), lossis ib qho prohormone.
Lees Daim Ntawv:Qhov "hmoov tsim yog hais txog qhov nyoos, bulk tshuaj ua ntej encapsulation lossis kev npaj daws teeb meem. Daim foos no feem ntau yog tsuj rau tus nqi {{1} dosing yoog raws li cov kev pheej hmoo siab thiab ncaj ncees piv rau cov tshuaj- cov ntsiav tshuaj qib.
Txuas kev siv tshuaj kho mob:Tamoxifen yog cov tshuaj kho mob cancer rau kev kho mob cancer mis (kev txo qis thaum ntxov rau estrogen receptor {{0}) cancer. Nws ua raws li anti - estrogen nyob rau hauv cov kua mis.
● Cov ntsiab lus ntawm lub cev:Nws daim ntawv thov nyob rau hauv kev ua kom lub cev tsis tau ua tiav - daim ntawv lo rau cov nqaij mos (zoo li cov tshuaj anabolic (cov kev hloov mus rau estrogen).


Cov Nta Tshwj Xeeb: Cov Serm Mechanism
Tamoxifen lub zog nyob hauv nwsrabELLIALS, sib txawv nws hauv phau ntawv los ntawm aromatase inhibitors (AIS) zoo li Anastrozle:
● Cov nqaij - kev ua tshwj xeeb (agonist / agonistist):
Ugselsection hauv cov nqaij mos:Qhov no yog nws cov khoom muaj txiaj ntsig tshaj plaws hauv kev ua kom lub cev. Tamoxifen kev sib tw khi rau tshuaj ntsuab rau estrogen receptors (ers) nyob rau hauv cov kua mis, thaiv cov tshuaj steroids uas muaj ntxhiab los ntawm cov tshuaj steromatized los ntawm kev sib tw thiab siv nyiaj ntau. Qhov no qhia ncaj qha los ntawm kev txhim kho ntawm Gynecomastia ("Gyno").
○ agonist nyob rau lwm cov ntaub so ntswg:Qhov muag, hauv cov nqaij xws li pob txha, nplooj siab, thiab qhov endometrium (uterine phlu), tamoxifen taume nyuamQee qhov teebmeem ntawm estrogen (ua yeeb yam raws li ib nrab agonist). Qhov no muaj qhov cuam tshuam tseem ceeb:
Cov pob txha ceev:Tej zaum yuav pab tswj cov pob txha ntxhia pob hluav taws xob, uas tuaj yeem cuam tshuam tsis zoo los ntawm cov tshuaj estrogen tsawg (ib txwm muaj ecct).
◇Lipid Profile:Muaj peev xwm muaj peev xwm ntau dua (lossis tsawg dua qhov tsis zoo) cuam tshuam rau cov roj (HDL / LDL) piv rau cov tshuaj HDL ("zoo" cholesterol).
◇Endometrial teebmeem:Cov tshuaj estrogen ua rau lub tsev menyuam yog ib qho kev paub txaus ntshai rau qhov hloov pauv thiab cov kabmob khees xaws rau cov poj niam; Qhov no feem ntau tsis muaj kev txhawj xeeb rau tus txiv neej bodybuilders tab sis tseem ceeb cov nqaij mos.
In Central Hoom Ceg Kev Pom Zoo Loop cuam tshuam:Tsis zoo li AIS, uas muaj kev txo qiskev ncig ua siCov qib tshuaj estrogen ua haujlwm, tamoxifen feem ua haujlwm ntawm qib receptor nyob rau hauv cov ntaub so ntswg tshwj xeeb. Tseem ceeb, los ntawm thaiv cov recetors estrogen hauv hypothalamus, nwsua kom yuam kevlub cev ua rau pom cov qib tshuaj estrogen tsawg. Qhov no txhawb cov hypothalamic - pituitary - gonadal (hpg) axis:
○Lub hypothalamus tso ntau cov gonadotropin - tso cov hormone (GNRH).
○Gnrh teeb liab lub caj pas pituitary kom nce kev tso tawm ntawm Luteinizing Hormone (LH) thiab cov hauv paus {}} stim) stim}.
○Ua kom LH / FSH BISTULATES cov kev sim los ua cov testosterone ntau dua thiab rov pib phevitogenesis. Qhov no ua rau tamoxifen invaluable rauNcej Post (PCT).
Cov ntawv thov nyob rau hauv lub cev hauv lub cev: dhau Gyno kev tiv thaiv
Thaum kev tiv thaiv thiab kho Gynecomastia yog nws cov kev lees paub tshaj plaws, Tamoxifen cov ntawv thov yog dav dav:
● Gynecomastia (Gyno) Kev Tiv Thaiv & Reversal:Thawj tus tsav tsheb rau ntawm - kev voj voog lossis tshaj tawm {1} {1} {kev siv. Los ntawm kev thaiv ntawm ers hauv cov ntaub so ntswg noj mov, nws tau tso qhov loj heev ntawm cov tawv nqaij glandular tshwm sim los ntawm kev nce qib tshuaj estrogen. Kev cuam tshuam thaum ntxov (ntawm thawj cov cim ntawm khaus, muaj kev sib tw, lossis cov qog) yog qhov ua tau zoo tshaj; tsim, fibrous gyno feem ntau yuav tsum phais.
Roory Post Kev voj voog (PCT):Qhov no yog kev sib cav nwstseem ceeb tshaj plawsNtawv thov. Tom qab lub voj voog ntawm suppressive compounds (tshwj xeeb yog cov tshuaj steromyizing lossis prochormones, sarms, thiab lwm yam khoom siv tau kaw. Tamoxifen pab rov ua dua HPTA:
○ Blocks Estrogen Tswv yim ntawm hypothalamus / pituitary.
○ Ua kom muaj LH thiab FSH zais cia.
○ Ua lwm cov neeg ua haujlwm hauv cov kev sim los ua cov testosterone.
Aids Aids hauv kev rov qab kho kom zoo endogenous hormone sib npaug ntau dua ais ib leeg thaum PCT.
● Cov estrogen - Cov Dej Muaj Feem Kom Zoo Nkauj:Thaum tsis muaj zog tshaj ais rau tag nrho cov dej hauv dej, los ntawm kev thaiv cov ntaub so ntswg, nws tuaj yeem pab txo cov ntaub so ntswg, txhawb kev nyuaj, txhais tau tias lub cev tawv dua. Cov nyhuv no feem ntau yog qhov hloov maj mam hloov pauv dua li ais.
"Ntawm kev voj voog" Tshuaj Ntsuam Xyuas Kev Tswj Xyuas (Feem Pua):Qee lub sij hawm siv nrog aromatizing steroidsfab ntxeevNtawm AI, tshwj xeeb yog los ntawm cov tib neeg uas ua siab loj dua li ais lossis muaj kev txhawj xeeb txog lipid supression lossis mob sib koom tes los ntawm cov tshuaj estrogen tsawg dhau. Txawm li cas los xij, AIS nyob twj ywm thawj ntawm - lub voj voog xaiv rau kev tswj hwmkev ncig ua siCov qib tshuaj estrogen. Tamoxifen yog siv rau ntawm -} pa feem ntau thaum gyno cov tsos mob tshwm sim txawm tias ai siv lossis raws li kev tiv thaiv yog tias muaj kev tiv thaiv Gyno.
Pom cov txiaj ntsig (vs. AIS & hauv cov ntsiab lus)
●onupy HTA txhawb nqa rau PCT:Ntau dua li AIS ntawm LH / Fsh tso tawm tseem ceeb rau kev rov qab.
Lipid Profile sparing:Feem ntau ua rau muaj tsawg dua kev puas tsuaj cuam tshuam rau HDL cov cholesterol piv rau lub zog AIS zoo li Letrozole lossis txawm Aastrozole.
● Cov pob txha ceev txhawb:Tej zaum yuav muaj cov laus laus cov nyhuv rau cov pob txha yuav muaj kev tiv thaiv pob txha uas tuaj yeem tshwm sim nrog lub sijhawm ntev {{0} ▪ Hormone CCT theem.
Sib koom nrog lubrication tiv thaiv:Los ntawm tsis sib tsoo lub cev tshuaj estrogen raws li profoundly li AIS, nws yuav pab tswj cov tshuaj ntsuam estrogen tiv thaiv qee zaum cuam tshuam nrog kev txhoj puab rau kev txhoj puab.
Byno Kev Tiv Thaiv Ncaj Nraim:Cov Tub Txib txoj cai ntawm lub xaib ntawm kev txhawj xeeb (lub mis ers).
● Qhov ncauj cov khoom siv:Zoo thaum noj cov ncauj lus.
DOSAGE & CAWM QHIA: Precision yog Ntsiab
Dosing tamoxifen citrate hmoov yuav tsum tau ceev faj vim tias tsis muaj qauv thiab muaj kev txhawj xeeb nyob rau hauv cov hmoov nplej.Kws Tshuaj ntsiav yog vastly nyiam rau kev nyab xeeb thiab raug.Cov koob tshuaj uas hais txog tamoxifen citrate ntsev (uas muaj kwv yees li 65-70% tiag tiag tamoxifen paus).
● Gyno kev tiv thaiv / kev tswj hwm (ntawm - lub voj voog):
Tiv thaiv tiv thaiv:10Mg txhua hnub (ED) lossis txhua lwm hnub (EOD) feem ntau txaus thaum siv cov nyom sib xyaw. Cov koob tshuaj ntau dua tuaj yeem xav tau rau cov tshuaj steromatizy ntau lossis cov tib neeg nquag nquag rau Gyno.
○Kev kho mob (cov cim thaum ntxov):20-40mg ib hnub kom txog thaum cov tsos mob ntawm cov tsos mob (1-3 lub lis piam), tom qab ntawd muaj feem txo mus rau 10mg / hnub rau qhov tseem tshuav ntawm lub voj voog raws li kev saib xyuas.
Roory Post Kev voj voog (PCT):(Feem ntau ua ke nrog clomiphene citrate - cllomid)
○Cov PCT raws txoj kev cai (tamoxifen tsom):
◇Lub lis piam 1-2: 40mg ib hnub
◇Lub lis piam 3-4: 20mg ib hnub
◇Lub lis piam 5-6 (yeem yog xav tau / rov qab qeeb): 10mg ib hnub
○Ntev:Feem ntau 4 {{- 6 lub lis piam, pib 1-3 lub lis piam tom qab txhaj tshuaj ib nrab-lub neej) lossis tam sim ntawd tom qab lub sijhawm kawg ntawm qhov ncauj / SEARM DOSS.
● hmoov tshwj xeeb:Yog qhov tseeb koob tshuaj raw hmoov yog fraught nrog kev pheej hmoo. Micro - scoops yog cov lus tsis muaj tseeb. Demise Milligram nplai (0.001 daws teeb meem) yog qhov yuav tsum tau ua, tab sis txawm tias, homogeneity) Volumetric Dosing (yaj tus nqi paub nyob rau hauv ib lub zog zoo li kev ncua cov hmoov lossis dej cawv) yog tseem nqa cov kev pheej hmoo ntau dua rau cov ntsiav tshuaj.
Kev sib xyaw ua ke thiab pcct raws tu
● On - lub voj voog:Siv kev siv dag zog (ntawm thawj cov cim ntawm gyno) lossis proactively (yog keeb kwm muaj keeb kwm) nrog cov tshuaj propomatizing. Nws yogtsisHloov chaw rau AI yog tias muaj kev sib tw estrogen ua rau qhov tseem ceeb bloat lossis cov teeb meem ntshav siab yog qhov kev txhawj xeeb tseem ceeb. Dose: 10-20mg / hnub feem ntau.
● PCT:Lub pob zeb ntawm nws txoj kev ua kom siv lub cev. Pib tom qab exogenous anabolics / sarms muaj txaus tshem tawm cov kab ke (dictated byer ib nrab {{1} lub neej). Qauv PCT feem ntau ua ke:
○ Tam sim no:40mg / hnub (wk1 {{{{4 4}} 2), 20mg / hnub (wk3-4) - thawj qhov kev tiv thaiv kab mob, Gyno tiv thaiv.
Clomiphene (Clomid):50Mg / hnub (WK1 {- 2), 25mm / hnub (wk3-4) - tseem txhawb HPTA, syneroistic nrog Nolvadee nrog Nolvadex.
○Yeem txhawb nqa:HCG (siv ua ntej PCT rau KickStart Test), qis - Dose AI (tsuas yog cov tshuaj i (tsuas yog muaj cov tshuaj tiv thaiv loj
● Kev tseem ceeb:Pib pct dhau ntxov (nrog suppressive tebchaw tseem nquag) renders nws tsis muaj txiaj ntsig. Pib lig dhau sijhawm ntev ntev lub xeev suppressed. Kev Tshawb Fawb ASTEETER ASTEEN {2 2}} neeg lub neej meticulously.
Ib nrab - lub neej & phartectics: qhov ntev log
Ib nrab - lub neej:Tamoxifen nws tus kheej muaj ib qho teeb meem metabolic. Nws thawj cov metabolite,Endoxifen, yog lub luag haujlwm loj rau lub anti - estrogenic cuam tshuam hauv cov nqaij mos. Cov ntawv tshaj tawmTerminal ib nrab - lub neej ntawm tamoxifen yog kwv yees li ntawm 5-7 hnubCov. Txawm li cas los xij, vim cov metabolites thiab tsub zuj zuj, nws cov teebmeem yog lub sijhawm ntev.
● Mob khov kho:Vim hais tias ntawm no ib nrab ib nrab - lub neej, kwv yees li 4 lub lis piam) kom ncav cuag ruaj khov- lub xeev ntau zaus.
Ult Siv qhov cuam tshuam:Lub sijhawm ntev ib nrab - lub neej txhais tau tias ib zaug- kev noj mov txhua hnub yog txaus. Nws kuj tseem piav qhia yog vim li cas teebmeem (ob leeg kho thiab cov kev mob tshwm sim) tuaj yeem ua haujlwm rau lub lis piam tom qab ua kom tsis tu ncua. Thaum lub sijhawm PCT, cov qauv ua tiav cov kev sib tw muaj kev txhawb nqa cov kev txhawb nqa no thaum maj txo cov stimulus.
PCT (PT COPLE CARRAPY): Tamoxifen's Adining Lub Luag Haujlwm
PCT tsis yog kev xaiv tau; Nws yog qhov tseem ceeb rau kev txo cov leeg leeg cov leeg, rov kho kom zoo -}-}}} kev noj qab haus huv tom qab lub voj voog supressive. Tamoxifen yog ib qho cuab yeej siv ua lag luam:
● Cov mechanism recap: Blocks estrogen negative feedback -> Increases GnRH -> Increases LH/FSH -> Stimulates Testes ->Restores Ntuj Testendone Ntau Lawm.
● Cov hom phiaj:
○ Rov kho endogenous Testosterone ntau lawm sai thiab ua tau zoo li sai tau.
○ Tsawg txoj kev sib tsoo "tsoo" lub sijhawm (cov tshuaj hormones tsis tshua muaj zog
○ Tiv thaiv cov tshuaj estrogen (uas tuaj yeem ua rau gyno) raws li cov tshuaj hormones exabenous meej thiab cov hpta restarts.
○ tswj tau ntau npaum li tau txais cov leeg nqaij loj li sai tau.
Vim li cas tamoxifen yog nyiam tshaj Ai rau PCT:AIS tsuas yog txo cov kab sib ncig ntawm cov tshuaj estrogen; Lawv tsis ncaj qha txhawb lub HPTA. Tsawg estrogen thaum PCT tuaj yeem ua rau muaj kev puas tsuaj (pob txha pob txha, lipids, pob qij txha, zaum siab). Tamoxifen muab qhov tsim nyog hypotalamic / pituitary stimulationthaumKev thaiv cov tshuaj ntsuam estrogen lub tswv yim tsis zoo thiab tiv thaiv cov nqaij mos, tsis tas yuav tsoo cov qib tshuaj estrogen. Clomid ua tiav qhov kev txiav txim no.
Cov kev xav tseem ceeb & lus ceeb toom
1.Qhov fda -} Pom zoo rau kev ua haujlwm ntawm lub cev:Txhua qhov kev siv tau piav qhia ntawm no yog tawm ntawm - daim ntawv lo thiab tsis pom zoo rau kev ua tau zoo.
2. Tsis yog:Raw Tamring hmoov citrate hmoov cov hmoov av tseem ceeb: kev ua kom dawb huv / tsis muaj teeb meem, tsis muaj teeb meem (nyob rau hauv), clumping), tsis muaj menyuam.Kws Khoos phib tawj - Cov ntsiav tshuaj qib yog muaj kev nyab xeeb dua.
3. Cov teebmeem cuam tshuam (Cov txiv neej):Thaum feem ntau zoo -}}}}}}}}}}}}}}}}}}}}}}} a in in hauv qee qhov, muaj peev xwm nyob nrog:
Ofkes Cov Kub Kub
○ Hloov pauv, kev nyuaj siab
Hunkaches
○ Kev daws teeb meem (tsawg kawg, qhia tam sim ntawd)
○ Gastrointestinal chim (xeev siab)
○Nce thrombosis pheej hmoo:Tamoxifen yog txuam nrog kev pheej hmoo ntawm cov ntshav txhaws (DVT, pulmonary embolism) thiab mob stroke. Kev pheej hmoo yog siab dua nrog kev haus luam yeeb, immobility, caj ces, lossis lwm yam tawgicenic tebchaw.
○Tej zaum Mauv Feem Lipid cuam tshuam:Thaum feem ntau zoo dua li AIS, nws tseem tuaj yeem cuam tshuam li Lipids hauv qee tus neeg.
4.Qhov kev daws teeb meem:PCT yuav tsum muaj cov hau kev (Nolvadeex + Clomid + lub sijhawm ua neej + sijhawm). Tamoxifen tsis kho tam sim ntawd.
5.gynecomastia txwv:Zoo rauntxov, estrogen -}} tsav gyno. Paub tab, fibrous glandular nqaij feem ntau yuav tsum tau tshem tawm kev phais mob.
6. Kev Saib Xyuas Kev Saib Xyuas 6.:Qhia tawm. Ntshav ua haujlwm (ua ntej, nruab nrab, ncej {{1} {{2} {{2} {{2}, mob siab, thiab muaj kev noj qab haus huv tag nrho.
7.Legal xwm txheej:Muaj yam uas tsis muaj tshuaj yuav tsis raug cai nyob rau hauv feem ntau cov teb chaws.
Cov ntaub ntawv kho mob
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Kev Lag Luam Npe |
Nolcalx, Genox, Tamifen, TMX; ICI-46474 |
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Cas |
10540-29-1 |
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Tus hniav loj |
371.524 |
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Cov lus ntawm ib txoj kab ke |
C26H29Tsis muaj |
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Kev coj dawb huv |
Saum toj no 98% |
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Kev tsim nyog |
Dawb crystalline hmoov |
Kev xav tau, thov hu rau peb
Email: Jasonraws106@gmail.com
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Xaus: Ib qho cuab yeej tshwj xeeb, tsis yog lub mos txwv khawv koob
NolvadEX (Tamoxify citrate) hmoov, nyob rau hauv realm ntawm kev ua kom lub cev, yog lub zog thiab tshwj xeeb pharmacological ntsuas. Nws tus nqi tshwj xeeb stems los ntawm nws dual xwm raws li xaiv tau recordor airs thiab ib nrab agis thaum lub sij hawm tseem ceeb sib zog ntawm PCT. Nws tau txais kev tiv thaiv thiab tiv thaiv Gynecomastia thiab yog qhov tseem ceeb los ua kom tiav lub testosterone ntau lawm tom qab lub voj voog anabolic. Txawm li cas los xij, nws tawm - daim ntawv lo rau cov muaj kev pheej hmoo, ua kom muaj kev pheej hmoo txaus ntshai. Lub sijhawm ntev ib nrab- lub neej tsim nyog tsim tawm tswv yim koob tshuaj thiab tapering. Kev quaj ntsuag, tamoxifen tsis yog tus sawv cev Anabolic; Nws tsis tsim cov leeg. Nws yog daim ntaub thaiv tiv thaiv kev phiv tshuaj estrogen thiab catalyst rau kev rov qab los hauv hormonal. Nws txoj kev xav tau txais kev hwm, kev ua kom zoo nkauj, thiab kev ua kom muaj kev phom sij rau cov qauv kev kho mob thiab kev kho mob-} qib cov khoom lag luam. To taub nws cov tshuab, cov ntawv thov, cov txiaj ntsig, thiab muaj kev pheej hmoo ntau yog tsis yog xav txog nws siv.
Cim npe nrov: nolvadex (tamoxify citrate) rau lub cev lub cev: 54965-24-1, Tuam Tshoj Citrate) rau CAS BodyBuilding CAS: 54-1 manritorder: 54-1 manufacturers, chaw tsim khoom, Hoobkas
