
Dianabol (MethandRostenolone) steroids hmoov rau CAS bodybeilding CAS: 72-63-9
Dianabol, lub npe cim npe rau cov hluavtaws Anabian}}}}} methhantenolone (}}}} Hydrotadostenolone (}}}} Hydrotadostenolone (}} Thaum muaj keeb kwm ntawm qhov ncauj, "dianabol hmoov" yog hais txog lub ntsej muag nyoos, crystalline sau nyob rau hauv nws cov lus tseem ceeb tshaj plaws hauv kev tshawb fawb, chaw tsim tshuaj lag luam, lossis kev kuaj mob tsis zoo. Qhov kev ntsuas no ua kom muaj txiaj ntsig tob rau hauv cov yam ntxwv kev tsim txuj ci, theoretical cov ntawv thov, thiab hmoov tseem ceeb, nthuav tawm nruj me ntsis rau kev nkag siab thiab kev tshawb fawb.
Kev Txhais Lus Methandostenolone Hmoov: Qaum Cawv
● Cov qauv tshuaj lom neeg:MethandRostenolone belongs rau cov thawj coj ntawm lub neej no (DHT) derivative tsev neeg tab sis yog hloov kho qauv. Cov yam ntxwv tseem ceeb suav nrog:
○ 1,2-dehydrogenation:Taw qhia ntawm ob daim ntawv cog lus ntawm cov pa roj carbon atoms 1 thiab 2 (zoo ib yam li tus poj niam hormone estradiol) tau nce ntxiv piv rau Testosterone.
{17 - methylation:Ib qho ntxiv ntawm methyl pawg (-}} Txoj Haujlwm ntawm lub siab los ntawm kev mob siab rau lub siab thaum xub thawj-}}}}}}}}}}}}}}} kev sib tw ntawm qhov ncauj. Qhov kev hloov kho no tseem muaj lub luag haujlwm rau nws qhov kev pab hepatotoxic tseem ceeb.
Lub cev daim ntawv lub cev:Raws li hmoov, methandrostenolone feem ntau zoo nkaus li zoo li tsis zoo rau -} Crystalline khoom. Nws cov particle loj xa tuaj yeem sib txawv raws li synthesis thiab txoj kev ua kom huv, cuam tshuam nrog solubility thiab ntws cov yam ntxwv.
Solubility:Cov khoom ua pov thawj tsis tshua muaj solubility hauv dej. Nws ua rau pom kev sib txawv zoo dua rau cov kuab tshuaj yeeb yaj kiab zoo li ethanol, chloroform, lossis dimethyl dulfoxide (DMSO), yog ib qho tseem ceeb ntawm kev tshawb fawb lossis kev tshawb fawb.


Cov yam ntxwv txawv ntawm cov hmoov daim
Purity & Potency:Kws Tshuaj Kho Mob - Cov hmoov qib raws li cov tshuaj dawb (API), pub dawb los ntawm cov kws ua tshuaj ua haujlwm, fryes, los yog pleev xim rau hauv cov ntsiav tshuaj tiav. Theoretical potency yog maximized ib chav tsev loj. Txawm li cas los xij, immicitly noj cov hmoov huv huv yog heev sib txawv thiab tsis sib haum yam tsis muaj kev sim siab tshaj tawm (HPLC, MS).
● Kev tuav tes & ruaj khov:Yuav tsum tau nruj nruj tuav cov cai hauv kev tshawb fawb:
Yes Stability: Degrades upon prolonged exposure to light, heat (>25 degree), oxygen, thiab ya raws. Yuav tsum tau ntim rau hauv airtight, lub teeb agertight, lub teeb - Cov khaub ncaws tiv taus qis dua (1}} 8 degree) rau kev ruaj khov ntev.
○ Hygroscopicity:Tej zaum yuav nqus noo noo los ntawm huab cua, ua rau clumping, muaj peev xwm, thiab dosing.
Kev Nyab Xeeb:Cov kev ua haujlwm ruaj ntseg kev nyab xeeb (hnab looj tes, ntsej muag hoods) yog qhov tseem ceeb rau kev nqus tau kev nqus tau los yog dermal nqus vim nws cov kev phom sij thiab muaj peev xwm noj qab haus huv.
Producation versatulation versatility (theoretical):Hauv kev tswj cov tshuaj tsim kho, cov hmoov ua haujlwm raws li cov khoom pib rau kev tsim ntau yam ntawm cov kua txiv (cov duab hloov pauv ntawm qhov ncauj Kev siv tsis haum feem ntau cuam tshuam nrog kev piam sij thiab tsis muaj tseeb "kev ua haujlwm" mus rau hauv cov ntsiav tshuaj lossis kua.
Tshawb nrhiav cov ntawv thov & theoretical cov txiaj ntsig (tshuab ntawm kev ua)
Kev tshawb fawb mus rau MethandRostenolone lub tshuab ua qhia cov kab feem cuam tshuam rau cov leeg cev nqaij daim tawv:
1.anabolic stimulation:Binds ruaj khov rau androgen receptors (AR) nyob rau hauv cov leeg nqaij leeg. Qhov kev ua txhaum no ua kom muaj cov khoom siv proteination (Actin) thiab lwm yam qauv txheej txheem, tsav hypertrophy.
2.Ua protein synthesis:Tseem ceeb Upregulates lub cellular tshuab lub luag hauj lwm rau txhais lus genetic code rau cov protecle cov leeg tshiab. Qhov no tshwm sim ntawm kev hloov kho ntawm kev teeb tsa txoj hauv kev zoo li mtor.
3.nitrogen cia:Txhawb nqa cov nitrogen zoo heev nyob rau hauv cov nqaij hlwb. Nitrogen yog qhov tseem ceeb ntawm cov amino acids (protein tsev cov khoom thaiv). Khaws ntau cov nitrogen tsim cov kev ua kom zoo sab hauv cov chaw rau kev txhawb nqa cov leeg loj thiab kho.
4.GLYCOGENOLYsisy & Substrate Siv:Tej zaum yuav nce glycogen tsoo hauv cov leeg thiab nplooj siab, muaj peev xwm ua cov piam thaj ntau ntau rau lub zog thaum lub zog ua haujlwm. Nws kuj tseem yuav cuam tshuam rau kev siv cov fatty acids thiab cov amino acids rau roj, tab sis cuam tshuam yog qhov nyuaj.
5.Yhroproiessis Stimulation:Tuaj yeem nce cov qe ntshav liab (RBC) ntau lawm (Erchthropoiesis) los ntawm kev ua kom muaj lub raum me me) los ntawm kev txhawb nqa lub raum loj (EPO) tso tawm thiab muaj peev xwm ua ncaj qha rau cov pob txha ua ntej. Kev nce RBC Suav txhim kho txhim kho cov ntshav oxygen - nqa muaj peev xwm, muaj peev xwm ncua kev qaug zog.
6.Central hlab ntsha (CNS) teebmeem:Cov kev nthuav qhia me me glucocorticoid artagionicoid artagionoid kev tawm tsam cuam tshuam nrog cov tshuaj hormones ntxhov siab zoo li cortisol. Tej zaum kuj tseem tuaj yeem ua rau muaj kev zoo siab me me thiab nce kev ua kom loj hlob ("Roid npau taws"), tsis ncaj ncees cuam tshuam kev cob qhia kev kawm.
Kev txiav txim siab ntau npaum: precision thiab peril
Dosing cov hmoov nplej raw yog qhov tshwj xeeb muaj kev phom sij vim yog cov teeb meem hnyav hauv kev ua tiav yam tsis muaj cov khoom siv tshwj xeeb.Microgram nplai yog cov npliag txaus ntshai thiab nquag muaj qhov tseem ceeb ua yuam kev.Theoretical dosages tau kawm txog hauv kev tshawb fawb cov ntaub ntawv rau qhov ncauj methhandrostenolone feem ntau ntau:
● Kev Tshawb Fawb Txog qib:Kev tshawb fawb tshawb xyuas cov teebmeem ntau zaus pib txhaj tshuaj tsawg (piv txwv li, 2-5 mg / hnub) los tsim cov hauv paus kev teb.
● Ntau yam ntau:Ntau cov kev tshawb fawb tau kuaj xyuas kev ua tau zoo lossis kev cuam tshuam ntawm kev siv nyiaj tau 15 {}}}}}}}}}}} kev sib cais rau 2-3 koob tshuaj vim nws lub neej luv luv.
Wigh - Kev Tshawb Fawb Dose:Qee qhov kev tshawb nrhiav tau tshawb txog cov koob tshuaj xyuas txog li 50 m lossis ntau dua, tsis pom tseeb txog kev ua kom muaj kev cuam tshuam tsis zoo uas tsis muaj txiaj ntsig zoo.
Ceeb Toom Ceeb Toom Tseem Ceeb:Sim ua kom haum "ntsuas" hmoov yeeb tshuaj siv cov cuab yeej hauv tsev lossis cov qauv milligram teev yog muaj kev phom sij heev. Kev noj tshuaj tsis muaj tseeb tuaj yeem ua rau muaj kuab lom lossis mob ntev, muaj kev noj qab haus huv. Kws tsim khoom lag luam siv cov khoom lag luam zoo heev rau cov qauv.
Kev voj voog muaj thiab ib nrab - lub neej
Ib nrab - lub neej:Methandrostenolone muaj ib tug kujluv ib nrab - lub neej, kwv yees tau kwv yees3.5 txog 6 teevCov. Qhov no yuav tsum ntau cov koob tshuaj txhua hnub (piv txwv li, txhua 8- 12 teev) kom tswj cov ntshav nyob ruaj khov thaum tshawb nrhiav, ua rau muaj kev sib txawv ntawm kev ua haujlwm ntev. Cov metabolites nquag tuaj yeem ua rau ntev dua.
● Lub voj voog Duration (Tshawb Xyuas Cov Ntsiab Lus):Kev tshawb fawb tshawb txog qhov cuam tshuam ntawm {{methylated Athhandrostenolone yog feem ntau muaj kev pheej hmoo ntawm Hepatotoxicity nrog lub sijhawm ntev. Siv sij hawm ntev dua li lub siab ntev thiab lwm yam kev sib raug zoo.
Er "Kickstarting":Nyob rau hauv keeb kwm kev tshawb fawb kev tshawb fawb cov ntsiab lus, nws tau txais kev cuam tshuam sai ntawm cov hnub) ua rau nws muaj kev sib tw nyob rau hauv hnub) ua rau tus neeg tes hauj lwm ntev (zoo li testosterone los yog nandrolone) tau siv tib lub sijhawm. Lub methandostenolone yuav muab cov kev mob anabolic tam sim ntawd thaum tos kom muaj estrable ester kom ncav cuag cov kev ruaj khov ntau lub lim tiam.
Post - Nrhiav Kev Tshawb Fawb (PCT) -} Tseem Ceeb Ua Physiology
MethandRostenolone, zoo li txhua yam exogenous androgently suppresses lub cev tsim ntawm hypothalamic {} particular axis (HTA):
1.supressionchism:Txhawb cov cim Androgenen teeb liab ntawm cov kev hypothalamus kom txo gonadotropin {}} tso cov khoom siv (GNRH) tso pa. Qhov no txo cov zis pituitary ntawm Luteinizing hormone (lh) thiab follicle- stimulating hormone (fsh). Yog tias tsis muaj lh dag, cov kev sim ua kom tsawg lossis tsis txhob ua testosterone ntau lawm thiab cov noob phevitogenesis.
2.PCT imptative:Raws li kev txiav methandrostenolone, tus mob HPTA tseem suppressed. Yog tias tsis muaj kev cuam tshuam, kev rov qab yuav yog cov tsos mob qeeb heev (lub hlis) lossis qee zaum tsis tiav, ua rau tsis tiav, kev poob siab, mob plab, rog tau txais).PCT yog tsis xaiv; Nws yog ib txheej txheem kev cawm ntawm lub cev tseem ceeb.
3.PCT cov neeg sawv cev (kev tshawb fawb tsom):
Cov Lus Qhia (Xaiv cov tshuaj ntsiav tshuaj estrogen receptor modulators):
Tamoxifen citrate:Blocks Etrogenors hauv hypothalamus / pituitary, txo cov lus tsis zoo los ntawm cov qib qis qis. Qhov no txhawb zog nce GNRH, LH, thiab FSH tso tawm ua kom rov muaj nuj nqi. Ib qho kev tshawb fawb dav dav muaj 20-40 mg / hnub rau 4-6 lub lis piam.
Terromiphene citrate (clomid):Zoo sib xws mechanism rau tamoxifen tab sis feem ntau suav tias yog me ntsis ntau zog rau lh kev txhawb zog. Siv ntawm 25-50 mg / hnub rau 4-6 lub lis piam.
○ Noob aromase intibitors ({- adjuncts, tsis yog Core Pct):Cov tshuaj zoo li Aastrozole lossis letraszole thaiv hluav taws xob estrogen synthesis. Thaum qee zaum sivthaumLub voj voog muaj aromatizable tebchaw los tswj cov tshuaj estrogen, lawv feem ntautsis tshua muaj txiaj ntsig zoo dua li cov sermsTxog kev txhawb nqa HPTA rov qab tshaj tawm - kev voj voog. Lawv lub luag haujlwm hauv PCT feem ntau lossis rau kev tswj hwm cov tshuaj ntsuam estrogen rebound yog tias cov kab lus ua rau nws.
○ HCG (tib neeg chorionic gonadotropin - priming):Mimics LH, qha rau cov kev sim los ua cov testosterone los tsim cov testosterone thaum lub voj voog lossis tam sim ntawd ua ntej PCT pib. Qhov no tiv thaiv cov lus dag kev ua pov thawj thiab muaj peev xwm "Prime" cov kev kuaj kom teb tau zoo dua rau LH sawv kev los ntawm cov lus qhuab qhia thaum PCT. Siv luv - sij hawm (piv txwv li, 500-1000 iu od rau 10 hnub) ntawm lub voj voog kawg,ua ntejPib cov lus qhuab qhia. Tsis siv thoob plaws thoob plaws PCT.
4.Qhov sijhawm sijhawm:Kev pib yog nyob ntawm cov compound ib nrab - lub neej thiab metabolites. Rau methandrostenolone ib leeg, PCT feem ntau pib 1 {- 2 hnub tom qab koob kawg vim nws lub neej luv. Yog tias ua ke nrog cov kav ntev, PCT pib lub lis piam tom qab.
5.PleXity:PVct raws li cov leeg muaj zog thiab vam khom cov khoom sib xyaw tshwj xeeb uas siv, kev siv tshuaj, nce siab ntev, thiab cov lus teb ntev li cas. Tsis muaj universal "ib - loj-
Cov Hluav Taws Xob Cov Txiaj Ntsig Zoo & Kev Nyab Xeeb Kev Noj Qab Haus Huv
Kev tshawb fawb cuam tshuam cov ntaub ntawv ntau dhau ntawm kev pheej hmoo ntau nrog Methantrostenolone siv:
● Hepatotoxicity:Qhov 17 - methyl pab pawg ua rau muaj kev chim siab. Qhov teebmeem suav nrog:
○RESULATING DAIM NTAWV TXIAV (AST, ALT)
○Hepatocyte kev puas tsuaj, cholestasis (tsis zoo kua txiv ntws)
○Hepatic peliosis (ntshav {- pu} puv cyst)
○Nce kev pheej hmoo ntawm Hepatocellular Adenoma / Carcinoma nrog siv lub sijhawm ntev.
● Cardiovascular:Kev cuam tshuam tsis zoo ntawm cov cholesterol profiles (lowers HDL "cov roj (cholesterol), nce siab" cholerosclerosis, thiab thrombosis (txhaws ntshav).
● Cov 10 itocrine:HPTA loj (raws li tau sib tham txog), muaj txuj ci keeb kwm, gynecomastia (mob pob txuv rau estrogen), ntxau txiv neej ua qauv ua paug (Androgenic).
● Kev siv hlwb:Mob viav vias, txob taus, kev ua phem ("Roid npau taws"), kev nyuaj siab (tshwj xeeb yog tshaj tawm {{
Lwm yam:Edema (dej khaws cia), muaj kev phom sij rau cov poj niam (lub suab tob tob, clitibergaly, plaub hau poob), insulin tsis kam, prostate ow.
Cov ntaub ntawv kho mob
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Kev Lag Luam Npe |
Methandienone; Methandrostenolone; Methadrolone; Perabol; Dehydromethyltestosterone; Methylboldenone; |
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Cas |
72-63-9 |
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Tus hniav loj |
300.442 |
|
Mf |
C20H28O2 |
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Kev coj dawb huv |
Saum toj no 98% |
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Kev tsim nyog |
Dawb crystalline hmoov |
Kev xav tau, thov hu rau peb
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Xaus: Qhov sib txuas ntawm lub zog tseem ceeb thiab muaj kev pheej hmoo txaus ntshai
Dianabol (methandrostenolone) hmoov sawv cev rau lub zog, tsis muaj tshuaj lom neeg cov txuj ci ntawm keeb kwm anabolic steroid. Nws cov nta - siab bioavailability vim {{{}} methylation, nitrogen cia, thiab kev txiav txim sai - piav qhia nws cov keeb kwm sau ntawv. Txawm li cas los xij, cov no tuaj inextricably txuas rau kev cuam tshuam loj thiab muaj peev xwm ua rau muaj kev puas tsuaj ntawm Hepatotoxicity, thiab Incounline cuam tshuam kev cuam tshuam, thiab kev cuam tshuam muaj kev puas tsuaj uas yuav tsum muaj kev cuam tshuam nrog kev ua kom rov zoo.
Cim npe nrov: Dianabol (MethandRostenolone) steroids hmoov rau CAS bodybeilding CAS: 72-63-9, Tuam Tshoj Dianabolone rau BodybeDing Cas: 72-63-9 Cov Chaw Tsim Tshuaj, Chaw Tsim Tshuaj
