
Oxymetholone
Oxymetholone, muag raws li cov npe lag luam Anadrol thiab Anapolon ntawm lwm tus, yog cov tshuaj androgen thiab anabolic steroid (AAS) uas yog siv feem ntau hauv kev kho mob ntshav qab zib. Nws kuj yog siv los kho pob txha, HIV / AIDS wasting syndrome, thiab txhawb kev hnyav nce thiab cov leeg nqaij loj hlob hauv qee lub sijhawm. Nws yog noj los ntawm qhov ncauj.
Oxymetholone, muag raws li cov npe lag luam Anadrol thiab Anapolon ntawm lwm tus, yog cov tshuaj androgen thiab anabolic steroid (AAS) uas yog siv feem ntau hauv kev kho mob ntshav qab zib. Nws kuj yog siv los kho pob txha, HIV / AIDS wasting syndrome, thiab txhawb kev hnyav nce thiab cov leeg nqaij loj hlob hauv qee lub sijhawm. Nws yog noj los ntawm qhov ncauj.
Oxymetholone, tseem paub los ntawm nws lub npe npe Anadrol, yog ib qho anabolic steroid uas tau muab los ntawm dihydrotestosterone (DHT). Nws yog feem ntau siv nyob rau hauv kev kho mob teb rau kev kho mob xws li anemia thiab nqaij nkos kab mob. Txawm li cas los xij, nws kuj tau muaj koob meej ntawm cov kws tsim lub cev thiab cov neeg ncaws pob rau nws lub peev xwm los txhim kho cov leeg nqaij thiab lub zog.
Cov kev mob tshwm sim ntawm oxymetholone suav nrog kev muaj siab sib deev ntxiv nrog rau cov tsos mob ntawm masculinization xws li pob txuv, plaub hau loj hlob, thiab lub suab hloov. Nws kuj tuaj yeem ua rau lub siab puas tsuaj. Cov tshuaj yog ib qho hluavtaws androgen thiab anabolic steroid thiab li no yog ib qho agonist ntawm androgen receptor (AR), lub hom phiaj lom neeg ntawm androgens xws li testosterone thiab dihydrotestosterone (DHT). Nws muaj zog anabolic teebmeem thiab tsis muaj zog androgenic teebmeem.
Oxymetholone tau tsim thawj zaug hauv xyoo 1959 thiab tau qhia txog kev siv tshuaj kho mob tab sis tsis ntev tom qab raug txiav tawm vim nws cov lipid toxicity siab hauv xyoo 1961. Nws yog siv feem ntau hauv Tebchaws Meskas. [3][10] Ntxiv rau nws txoj kev kho mob, oxymetholone yog siv los txhim kho lub cev thiab kev ua haujlwm.

Kev siv tshuaj kho mob
Cov kev kho mob tseem ceeb ntawm oxymetholone suav nrog kev kho mob ntshav qab zib thiab pob txha pob txha, nrog rau kev txhawb nqa cov leeg nqaij hauv cov neeg mob uas tsis muaj zaub mov tsis zoo lossis tsis muaj kev tsim kho. Txawm li cas los xij, hauv Tebchaws Meskas, tsuas yog qhov tseem ceeb ntawm FDA pom zoo yog kev kho mob ntshav qab zib.
Tom qab kev qhia txog oxymetholone, cov tshuaj nonsteroidal xws li epoetin alfa tau tsim thiab pom tias muaj txiaj ntsig zoo dua li kev kho mob ntshav qab zib thiab pob txha tsis muaj kev phiv ntawm oxymetholone. Cov tshuaj tseem muaj txawm tias qhov no thiab nws thiaj li pom muaj kev siv tshiab hauv kev kho mob HIV / AIDS nkuaj.
Tshaj tawm feem ntau raws li 50 mg ntsiav tshuaj, oxymetholone tau hais tias yog ib qho "muaj zog tshaj" thiab "muaj zog tshaj" AAS muaj rau kev siv kho mob. Ib yam li ntawd, muaj kev pheej hmoo ntawm kev mob tshwm sim. Oxymetholone muaj txiaj ntsig zoo hauv kev txhawb nqa kev nce hauv lub cev loj, feem ntau los ntawm kev txhim kho cov protein synthesis. Vim li no, nws feem ntau siv los ntawm bodybuilders thiab ncaws pob.
Oxymetholone yog siv rau lub cev- thiab kev ua tau zoo-txhim kho lub hom phiaj los ntawm kev sib tw ncaws pob, bodybuilders, thiab powerlifters.
Cov leeg nqaij thiab lub zog: Oxymetholone yog cov anabolic heev, txhais tau tias nws txhawb cov leeg nqaij thiab nce protein synthesis. Nws yog lub npe hu rau nws lub peev xwm los ua kom cov leeg nqaij thiab lub zog sai, ua rau nws nrov hauv zej zog bodybuilding.
Kev tsim cov qe ntshav liab: Oxymetholone txhawb kev tsim cov qe ntshav liab, uas tuaj yeem txhim kho cov pa oxygen hauv lub cev. Qhov no tuaj yeem txhim kho kev ua siab ntev thiab kev ua tau zoo thaum lub sijhawm ua haujlwm lub cev hnyav.
Pharmacodynamics
Zoo li lwm yam AAS, oxymetholone yog ib qho agonist ntawm androgen receptor (AR). Nws tsis yog substrate rau 5 -reductase (raws li nws twb 5 - txo) thiab yog ib tug tsis zoo substrate rau 3 -hydroxysteroid dehydrogenase (3 -HSD), thiab yog li ntawd qhia tau hais tias siab piv ntawm anabolic rau androgenic kev ua.
Raws li ib tug DHT derivative, oxymetholone tsis yog ib tug substrate rau aromatase thiab li no yuav tsis tau aromatized rau estrogenic metabolites. Txawm li cas los xij, tshwj xeeb ntawm DHT derivatives, oxymetholone tseem cuam tshuam nrog cov tshuaj estrogenicity siab, thiab paub tias muaj peev xwm tsim cov tshuaj estrogenic xws li gynecomastia (tsis tshua muaj) thiab dej tuav. Nws tau raug qhia tias qhov no yuav yog vim kev khi ncaj qha rau thiab ua kom cov tshuaj estrogen receptor los ntawm oxymetholone. Oxymetholone tsis muaj cov haujlwm tseem ceeb ntawm progestogenic.
Pharmacokinetics
Muaj qee cov ntaub ntawv muaj nyob rau ntawm cov tshuaj pharmacokinetics ntawm oxymetholone. Nws zoo nkaus li yog nqus tau zoo nrog kev tswj qhov ncauj. Oxymetholone muaj affinity tsawg heev rau tib neeg cov tshuaj hormone-binding globulin (SHBG), tsawg dua 5 feem pua ntawm cov testosterone thiab tsawg dua 1 feem pua ntawm DHT. [1] Cov tshuaj yog metabolized hauv daim siab los ntawm oxidation ntawm C2 txoj hauj lwm, txo ntawm C3 txoj hauj lwm, hydroxylation ntawm C17 txoj hauj lwm, thiab conjugation. C2 hydroxymethylene pab pawg neeg ntawm oxymetholone tuaj yeem tsim cov mestanolone (17 -methyl-DHT), uas tuaj yeem ua rau muaj kev cuam tshuam ntawm oxymetholone. Kev tshem tawm ib nrab-lub neej ntawm oxymetholone tsis paub. Oxymetholone thiab nws cov metabolites raug tshem tawm hauv cov zis.
Cov ntaub ntawv kho mob
1) CAS:
2) Lub npe lag luam: Anadrol, Anapolon
3) PubChem CID: 5281034
4) Molecular Formula: C21H32O3
5) Molecular Luj: 332.484g / mol
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Vim li cas thiaj xaiv peb cov khoom?
1. Zoo siab nrog tus nqi sib tw:
1) Txuj: BP / USP / EP / Enterprise txuj
2) Tag nrho Purity Ntau dua lossis sib npaug li 99 feem pua
3) Peb yog cov chaw tsim khoom thiab tuaj yeem muab cov khoom lag luam zoo nrog lub Hoobkas nqi.
2. Kev xa khoom sai thiab nyab xeeb
1) Parcel tuaj yeem xa tawm hauv 24 teev tom qab them nyiaj. Tus lej taug qab muaj
2) Kev ruaj ntseg thiab kev xa khoom xa tuaj. Ntau yam kev thauj mus los rau koj xaiv.
3) Kev lis kev cai hla tus nqi Ntau dua lossis sib npaug li 99 feem pua
4) Peb muaj peb tus kheej tus neeg sawv cev / xa rov qab / tus xa khoom tuaj yeem pab peb xa peb cov khoom sai thiab nyab xeeb, thiab peb muaj cov khoom xa tuaj rau hauv.
3. Peb muaj cov neeg siv khoom thoob plaws ntiaj teb.
1) Kev pabcuam tshaj lij thiab kev nplua nuj ua rau cov neeg siv khoom xav tau yooj yim, cov khoom tsim nyog thiab xa khoom sai raws li lawv lub siab nyiam.
2) Kev lag luam tawm tswv yim thiab cov khoom tawm tswv yim yuav raug qhuas, ua tau raws li cov neeg siv khoom xav tau yog peb lub luag haujlwm.
3) Zoo siab, tus nqi sib tw, xa khoom sai, kev pabcuam thawj zaug tau txais kev ntseeg siab thiab qhuas los ntawm cov neeg siv khoom
Cim npe nrov: Tuam Tshoj oxymetholone manufacturers, lwm tus neeg, Hoobkas
