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AC-262536 Sarms Bodybuilding CAS:870888-46-3

AC-262536 Sarms Bodybuilding CAS:870888-46-3

AC -262 356, tseem hu ua AC 262, yog ib qho kev tsis zoo tshaj plaws uas tsis yog steroidal xaiv androgen receptor modulator (SARM) nrog kev cuam tshuam zoo. Hauv kev tshawb fawb tsis ntev los no tau ua los ntawm cov txiv neej nas castrated tshaj li ntawm 2-lub lim tiam, AC-262 356 tau nthuav tawm qhov muaj peev xwm zoo tshaj plaws hauv kev txhim kho cov kab mob anabolic. Tshwj xeeb, nws pom tau tias muaj txiaj ntsig zoo hauv kev txhawb nqa kev loj hlob ntawm levator ani cov leeg thiab ua kom muaj txiaj ntsig zoo ntawm qib siab ntawm cov tshuaj hormones luteinizing. Cov kev tshawb pom no qhia txog qhov cuam tshuam tseem ceeb ntawm AC-262 356 raws li cov khoom siv txhim kho kev ua haujlwm hauv cov qauv tsiaj.

Xa kev nug
Hauj lwm lawm

    AC 262 356 Powder yog dab tsi?

   AC 262 356 hmoov yog ib qho kev xaiv androgen receptor modulator (SARM) uas tau txais kev saib xyuas hauv thaj tsam ntawm cov leeg nqaij thiab kev loj hlob. Selective androgen receptor modulators yog cov tebchaw uas xaiv khi rau thiab qhib lub androgen receptor hauv cov ntaub so ntswg tshwj xeeb, xws li cov leeg pob txha, thaum txo qis kev ua kom cov receptor hauv lwm cov ntaub so ntswg, xws li cov qog prostate.

AC 262 356 tau pom cov lus cog tseg hauv kev txhawb nqa cov leeg nqaij thiab ua kom cov leeg nqaij. Nws exerts nws cov teebmeem los ntawm tshwj xeeb lub hom phiaj thiab activating androgen receptors nyob rau hauv lub cev nqaij daim tawv nqaij hlwb, ua rau txhim kho protein synthesis thiab nqaij hypertrophy. Qhov kev xaiv no yog qhov tseem ceeb hauv kev zam cov kev mob tshwm sim uas feem ntau cuam tshuam nrog androgens, xws li tib neeg cov qog nqaij hlav cancer.

Los ntawm kev ua kom cov androgen receptor nyob rau hauv cov leeg pob txha, AC 262 356 pab txhawb kev loj hlob ntawm cov nqaij ntshiv. Nws txhawb cov synthesis ntawm cov proteins tshiab, pab kho cov leeg nqaij thiab kev loj hlob. Tsis zoo li cov tshuaj androgenic ib txwm muaj, AC 262 356 yog tsim los txo qis cov teebmeem androgenic uas tsis xav tau, ua rau nws yog ib qho kev xaiv zoo rau cov neeg tshawb fawb nrhiav kev txhim kho lawv lub cev.

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Nws Ua Haujlwm Li Cas?

AC-262 ua haujlwm los ntawm kev ua raws li kev ua ntawm testosterone, txawm tias muaj kev xaiv ntau dua. Hloov chaw ntawm kev khi rau androgen receptors thoob plaws hauv lub cev, AC-262 feem ntau tsom rau cov androgen receptors pom hauv cov pob txha thiab cov leeg nqaij. Qhov tseem ceeb, nws nthuav tawm qhov kev sib txuas tsawg kawg rau lub caj pas prostate, teeb tsa nws sib nrug ntawm testosterone qhov cuam tshuam thoob plaws.

Kev txhawb nqa pov thawj los ntawm 2-lub lim tiam kev tshawb fawb nyob rau hauv castrated txiv neej nas lees paub qhov txawv ntawm qhov no. Feem ntau, kev tswj hwm androgen hauv cov nas castrated ua rau cov prostate tseem ceeb thiab cov hlab ntsha loj zuj zus. Txawm li cas los xij, txoj kev tshawb fawb tau qhia tias thaum testosterone ua rau muaj qhov zoo tshaj plaws 10-fold nce hauv prostate loj, AC -262 tau pom tias tsis muaj zog ntawm prostate o.

Ib yam li ntawd, kev kho testosterone ua rau muaj ntau yam 14-fold nce hauv qhov loj me me piv rau cov tsheb kho cov nas tsuag. Hauv qhov sib piv, kev tswj hwm ntawm AC -262 ntawm ib koob ntawm 3mg / kg tsuas yog ua kom muaj txiaj ntsig zoo ntawm qhov loj me ntawm cov vesicle. Txawm tias nyob rau ntawm nws cov koob tshuaj ntau tshaj, qhov nce hauv cov hlab ntsha hauv lub cev yog 29.9 ± 2.2% txheeb ze rau kev kho testosterone.

Nws yog ib qho tsim nyog sau cia tias txawm hais tias nws muaj kev cuam tshuam me me rau ntawm prostate thiab seminal vesicle loj, AC -262 tseem pom muaj txiaj ntsig zoo rau cov kab mob endocrine thiab anabolic. Qhov tseeb, nws tau mus txog 117% thiab 66% ntawm qhov siab tshaj plaws tshwm sim nrog testosterone rau cov kev txwv no, feem. Yog li ntawd, AC-262 qhia tau zoo kawg nkaus cov ntaub so ntswg-xaiv cov khoom uas muaj tsawg kawg nkaus androgenic liabilities thiab phiv.

Cov txiaj ntsig muaj peev xwm ntawm AC 262 356

AC -262 thiab Luteinizing Hormone

Luteinizing hormone, secreted los ntawm pituitary caj pas, plays lub luag haujlwm tseem ceeb hauv kev loj hlob ntawm kev sib deev hauv cov txiv neej thiab poj niam. Kev nce qib ntawm LH tshaj li qhov qub tuaj yeem ua rau muaj ntau yam teeb meem xws li kev xeeb tub hauv cov poj niam, txo libido hauv cov txiv neej, thiab ntxov ntxov lossis ncua kev puberty rau cov menyuam yaus.

Hauv cov lus hais saum toj no 2- txoj kev tshawb fawb lub lim tiam, AC-262 tau ua rau muaj txiaj ntsig zoo rau kev nce qib ntawm cov ntshav plasma LH. Ntawm qhov koob tshuaj ntawm 3mg / kg, AC-262 txo qis LH qib los ntawm 40%. Ntxiv mus, ntawm cov koob tshuaj ntau dua ntawm 10 thiab 30mg / kg, AC-262 tau pom tias muaj kev cuam tshuam ntau dua hauv kev tawm tsam LH piv rau testosterone.

AC-262 thiab cov leeg nqaij

Ib qho tseem ceeb ntawm 2-lub lim tiam txoj kev tshawb fawb ntawm castrated txiv neej nas tau pom qhov muaj zog anabolic cuam tshuam ntawm AC-262 ntawm cov leeg nqaij. Kev tswj hwm ntawm AC -262 tau coj mus rau kev kho kom zoo ntawm qhov hnyav ntawm levator ani cov leeg, ncav cuag li 70% ntawm qhov siab tshaj plaws tshwm sim nrog testosterone (T). Nws yog ib qho tseem ceeb uas yuav tsum nco ntsoov tias qhov siab tshaj plaws cuam tshuam los ntawm AC-262 hauv cov ntaub so ntswg tau qis dua piv rau cov uas raug ntxias los ntawm T.

Cov kev tshawb pom no qhia txog lub peev xwm ntawm AC-262 raws li qhov tshiab xaiv androgen receptor modulator (SARM) nrog cov txiaj ntsig zoo anabolic rau cov leeg nqaij.

AC -262 thiab Alzheimer's Disease

Hauv kev tshawb fawb nas, AC-262 tau nthuav tawm qhov kev cog lus kho mob rau hnub nyoog txog kev paub txog kev poob qis thiab Alzheimer's disease. Qhov no SARM nce- tswj androgen receptor qib hauv lub hlwb tom qab castration, qhia nws lub peev xwm los hloov kho androgen signaling. Tsis tas li ntawd, AC-262 antagonized impairments nyob rau hauv siab spatial nco retention tshwj xeeb nyob rau hauv poj niam nas. Cov kev tshawb pom no qhia tias SARMs, suav nrog AC-262, muaj peev xwm tiv thaiv kev paub tsis meej hauv tus qauv nas ntawm Alzheimer's disease.

Hauv cov ntsiab lus, kev tshawb fawb tsiaj tau muab kev nkag siab zoo rau qhov cuam tshuam ntawm AC-262. Cov khoom sib xyaw ua ke tau qhia txog cov teebmeem anabolic tseem ceeb ntawm cov leeg nqaij loj hlob, ua haujlwm zoo txo ​​qis LH qib, thiab nthuav tawm cov peev txheej kho mob rau hnub nyoog txog kev paub txog kev poob qis thiab Alzheimer's kab mob hauv cov qauv tsiaj.

Kev tshawb fawb ntxiv yog tsim nyog kom nkag siab txog qhov cuam tshuam thiab muaj peev xwm siv AC -262 hauv tib neeg.

Kev ceev faj xav txog

AC-262, ua ib qho tsis-steroidal compound nrog anabolic kev ua, tau pom cov txiaj ntsig tau zoo hauv cov kev tshawb fawb ntawm cov qauv tsiaj, tshwj xeeb tshaj yog nyob rau hauv cov ntsiab lus tseem ceeb ntawm luteinizing cov tshuaj hormones thiab nce cov leeg nqaij. Txawm li cas los xij, nws yog ib qho tseem ceeb uas yuav tsum nco ntsoov tias AC -262 poob rau hauv qeb ntawm cov tshuaj tshawb fawb thiab tsis tau kawm ntau yam hauv tib neeg.

Vim qhov kev tshawb fawb tsis tshua muaj nyob ntawm AC-262 thiab nws cov kev cuam tshuam rau cov ntaub so ntswg, yuav tsum tau ceev faj. Cov tib neeg uas muaj kev txhawj xeeb txog lawv cov kev noj qab haus huv ntawm cov menyuam yaus lossis cov uas tab tom nrhiav kev tiv thaiv kev xeeb tub yuav tsum tsis txhob siv AC -262 kom txog thaum muaj kev tshawb fawb ntxiv los ntsuas nws qhov cuam tshuam rau cov ntaub so ntswg.

Tej yam tshwm sim

Raws li AC-262 yog cov tshuaj tshawb fawb nrog tib neeg kev tshawb fawb, nws qhov kev nyab xeeb thiab cov kev mob tshwm sim tsis tau nkag siab tag nrho. Txawm li cas los xij, raws li cov ntaub ntawv muaj, nws yog ib qho tseem ceeb uas yuav tau txiav txim siab txog kev pheej hmoo thiab siv ceev faj thaum siv AC -262. Qee tus neeg yuav muaj kev cuam tshuam tsis zoo xws li hormonal imbalances, hloov mus ob peb vas, lossis hloov pauv hauv lipid profile. Tsis tas li ntawd, txij li AC -262 yog ib qho tsis-steroidal compound nrog cov khoom siv anabolic, muaj peev xwm tsis paub txog qhov cuam tshuam ntev rau ntau lub cev.

Cov ntaub ntawv kho mob

Cov npe lag luam

AC -262,536

CAS

870888-46-3

Molar loj

278.355

MF

C18H18N2O

Purity

Tshaj 98%

Yam khoom

Dawb Cyrstalline hmoov

 

 

Txhua yam kev xav tau, thov hu rau peb

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Xaus

Hauv kev xaus, kev siv AC-262, uas tsis yog-steroidal androgen receptor modulator, muaj ntau yam txiaj ntsig. AC-262 xaiv lub hom phiaj ntawm lub cev androgen receptors, tsom feem ntau ntawm cov leeg pob txha thaum sparing cov ntaub so ntswg. Qhov tshwj xeeb no txo ​​qhov kev pheej hmoo ntawm kev mob qog noj ntshav prostate, kev txhawj xeeb cuam tshuam nrog qee cov tshuaj anabolic steroids. AC-262 tau pom tias muaj peev xwm ua kom cov leeg nqaij, txhawb kev nco ntau dua, thiab muaj peev xwm pab txo cov rog.

Tsis tas li ntawd, AC-262 tau qhia txog kev nyab xeeb zoo nrog kev txwv tsis pub muaj kev cuam tshuam rau daim siab enzymes thiab natural testosterone ntau lawm.

Txawm hais tias AC-262 cov txiaj ntsig tau txais kev txhawb nqa los ntawm kev tshawb fawb tsiaj thiab cov ntaub ntawv pov thawj, nws txoj kev ua tau zoo thiab kev nyab xeeb hauv tib neeg kev sim siab tseem yuav tsim kom tiav. Txawm li cas los xij, raws li kev tshawb fawb tshuaj nrog siab purity thiab tsis-steroidal xwm, AC -262 sawv cev rau kev cog lus muaj peev xwm kho mob rau cov tib neeg nrhiav kev txhim kho lawv cov kev ua tau zoo thiab kev ua siab ntev thaum txo qis cov kev pheej hmoo cuam tshuam nrog cov tshuaj anabolic steroids.

Kev tshawb fawb ntxiv yog xav tau los piav qhia txog cov kev hloov pauv ntawm cov molecular thiab cov teebmeem mus sij hawm ntev ntawm AC-262, nrog rau kev tshawb nrhiav nws lub peev xwm los ua qhov kev nyab xeeb dua rau lwm cov SARMs thiab cov tswj hwm anabolic.

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