
Minoxidil kho Androogenic alopecia CAS: 38304-91-5
Minoxidil, pib tsim nyob rau hauv xyoo 1950 los ua cov tshuaj tiv thaiv kab mob siab, ua rau cov plaub hau kev txhim kho ntawm cov ntshav rau And30Sing alopecia (aga) xyoo 1980} {}
Taw qhia rau Minoxidil
Minoxidil, pib tsim nyob rau hauv xyoo 1950 los ua cov tshuaj tiv thaiv kab mob siab, ua rau cov plaub hau kev txhim kho ntawm cov ntshav rau And30Sing alopecia (aga) xyoo 1980} {} Kev kho cov dej numicicic, invic minoxidil cov plaub hau tau ncaj qha, kev ua haujlwm ntawm cov kev ua haujlwm ntawm tes uas rejuvertate plaub hau kev ua si {}}

Mechanism ntawm Kev Ua: Tshaj dhau Vasodation
Minoxidil txoj kev ua tau zoo hauv aga stems los ntawm kev sib txuas ntau ntawm kev sib txuam muaj ntau yam roj ntsha:
● Cov Potassium Channel Ua Kom Taus:Minoxidil sulfate, nws cov metabolite (qhib calcium calcium
● Kev caij nyoog ntawm Anagen theem:Los ntawm upregulating wnt / -catenin signings, Minoxidil txuas ntxiv ntawm cov hauv paus plaub hau, ncua kev nkag mus rau hauv Catagen (regression) theem.
● Los tiv thaiv cov teebmeem:Nws inhibits kev hloov pauv kev loj hlob-beta (tgf-), txo cov fibosulation fibrosis uas txuam nrog aga kev vam meej.
● Sulfotteras:Kev ua tau zoo nrog sulfottransferase enzyme kev sib tw hauv cov yeeb yaj kiab plaub hau hauv no enzymidil rau cov neeg siv plaub hau (30-40% ntawm cov neeg siv).
Cov qauv thiab cov yam ntxwv
Minoxidil muaj nyob rau hauv ob FDA-pom zoo cov qauv tsim:
Cov kua ua kua (2% thiab 5%):Siv nyob rau ntawm tus tsuj, feem ntau muaj propylene glycol, uas yuav ua rau tawv taub hau .
Foam ua npuas dej cawv (5%):Nyiam rau cov tawv nqaij rhiab, nrog lub sijhawm kom qhuav sai dua .
Cov yam ntxwv tseem ceeb suav nrog:
● Cov kev siv rov qab rau-kev sib kis tau:Tsis muaj daim ntawv yuav tshuaj yuav tsum muaj, txhim kho cov neeg siv khoom siv .
● Kev siv hom kev siv:5% kev pom zoo yog FDA pom zoo rau tus txiv neej, thaum 2% yog pom zoo rau cov poj niam vim muaj kev tiv thaiv hypertrichosis txaus ntshai ntawm 5,6% nyob rau hauv kev saib xyuas kev kho mob.
Cov ntawv thov kev kho mob thiab kev ua tau zoo
Txiv neej txawv (MpB):Kev tshawb fawb qhia tau 5% minoxidil nce cov plaub hau los ntawm 10-15% tom qab 24% ntawm cov neeg siv .
● Poj niam ua qauv plaub hau (FPHL):2% kev daws teeb meem cov plaub hau ntom ntom hauv 40-60% ntawm cov poj niam, txawm tias cov txiaj ntsig tsis tshua muaj zog piv rau cov txiv neej.
● Adjectant Kev Kho Mob:Ua ke nrog kev kho cov ncauj ntawm qhov ncauj lossis cov qib qis laser, Minoxidil tau txais txiaj ntsig los ntawm kev tsom cov kev sib txawv vs {{1 {{.
Cov txiaj ntsig thiab cov txiaj ntsig zoo
● Tsis muaj qhov:Daim ntawv thov cov ncauj lus txiav kom tsis txhob muaj cov xwm txheej tshwm sim txuas rau hauv kev mob siab .
● Cov pov thawj kev nyab xeeb kev nyab xeeb:Kaum xyoo ntawm kev siv cov kev pheej hmoo ntev ntev thaum siv raws li qhia .
Them Nqi-Ua Haujlwm:Cov qauv dav dav muaj peev xwm pheej yig rau kev xaiv cov kev xaiv zoo li cov plaub hau hloov cua daj cua dub {}}}
Muab thiab Cov Lus Qhia Txog Kev Tswj Xyuas
Txiv neej:Thov 1 ml ntawm 5% daws ob zaug ib zaug ib hnub twg rau lub taub hau qhuav to taub.
Cov poj niam:1 ml ntawm 2% daws ob zaug ib hnub ob zaug, txawm tias 5% yuav siv tawm-daim ntawv lo nrog soj ntsuam.
Technique:Ntu plaub hau kom ntov tawv taub hau, zaws maj mam muab, thiab tsis txhob ntxuav rau 4 teev tom qab ntawv thov.
Kev Kho Mob Kev Kho thiab Sijhawm
● Khais Thaum Kawg Shedding (Ziam Yes 2-8):Ib qho kev nce siab hauv cov plaub hau poob tshwm li dormant cov hauv paus nkag rau theem kev loj hlob .
● Cov ntsiab lus thaum ntxov (hli 3-6):Vellus plaub hau hloov mus rau lub davhlau ya nyob twg plaub hau, txhim kho kev pab them nqi .
● Kev ua tau zoo (hli 12):Qhov siab tshaj plaws plaub hau ua tiav; Kev siv txuas ntxiv yog qhov tsim nyog los txhawb nqa cov txiaj ntsig .
Pharmaconinetics: Ib nrab-lub neej thiab metabolism
● Kev nqus nqus:~ 1 {. 3% kev nqus cov txheej txheem 3%, nrog ntshav ib nrab-lub neej ntawm 4,2 teev.
● Metabolism:Hepcatic gluidation tsim cov metabolites ua tsis muaj zog tshaj tawm renally .
Kev txiav txim siab tom qab kho mob (PTC) txiav txim siab
Discontinuation thim rov qab cov txiaj ntsig tsis pub dhau 3-4 lub hlis, raws li cov neeg hauv paus ua rau lawv cov miniate teb, hais txog qhov xav tau rau lub neej ua neej zoo {}}
Chaw Hais Cov Lus Tsis Yog thiab Txhim Kho Kev Noj Txiaj Ntsig
● Microneedling:Txhua lub limtiam Dermarler siv (0 .}}}}} 5-1.5 mm) txhim kho Minoxidil kev nqus thiab Upregulates kev loj hlob ntawm cov yam ntxwv.
● Cov khoom siv hluav taws xob rov qab:Tretinoin nce sulfottransferase kev ua si, muaj peev xwm hloov pauv tsis yog-teb .
● Qhov ncauj minoxidil (tawm-daim ntawv lo):Tsawg cov tshuaj (0 {. 25-2.5 mg / hnub) qhia cov lus cog tseg hauv kev tsis txaus siab thiab kev saib xyuas kev xav yog qhov tseem ceeb.
Kev Nyab Xeeb thiab Kev Mob tshwm sim
● Ntau:Tawv taub hau khaus (7% ntawm cov neeg siv), hypertrichosis (5% ntawm cov poj niam).
Tsis tshua muaj:Tachycardia, tsis haum rau tus mob dermatitis .
● Cov lus qhia:Cev xeeb tub (qeb c), tawv tawv tawv tawv nqaij, lossis kev sib zog ntawm cov lej .
Nrhav thiab cov lus qhia yav tom ntej
● Nanotechnology:Liposomal encapsulation txhim kho cov follicular .
● Gene Edapy:Hom phiaj Sulfotransferase polymorphisms rau tus kheej kev kho .
Lem Siv Lub Tsev Ua Kom Teg Dag:Kev Tshawb Fawb Tshawb Nrhiav Minoxidil lub luag haujlwm hauv kev ua kom cov plaub hau follices qia ntawm prostaglandin evkways {}}
Cov lus qhia tswv yim rau cov neeg siv
Sib xws li:Cov plaub hau ploj mus nrawm dua cov plaub hau hle dua .
Lub neej Syningergy:Kev ntxhov siab kom tsawg dua thiab kev noj zaub mov sib npaug (hlau, biotin) ua tiav kev kho .
● Zam kev tso tseg:Tsis txhob tshaj tawm; tshaj kev daws tsis txhim kho cov txiaj ntsig tab sis nce sab kev mob tshwm sim .
Cov ntaub ntawv kho mob
|
Kev Lag Luam Npe |
Loolfee, Rogaine, 2, 4- diamero_}} piperidinoprimididble {}} xide |
|
Cas |
38304-91-5 |
|
Tus hniav loj |
209.253 |
|
Mf |
C9H15N5O |
|
Kev coj dawb huv |
Saum toj no 98% |
|
Kev tsim nyog |
Dawb crystalline hmoov |
Kev xav tau, thov hu rau peb
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Tag
Cov neeg siv tshuaj loog AGA vim nws qhov kev cia siab uas muaj kev cia siab rau nws txoj kev xav tau zoo li kev cia siab rau kev sib tw thiab kev sib tw uas muaj kev sib tw ntawm cov kev daws teeb meem ib puag ncig kev cuam tshuam .
Cim npe nrov: Minoxidil kho Androtrasenic alopecia CAS: {{}}}} Mine}} {{} Cov chaw tsim khoom, cov chaw tsim khoom, chaw tsim khoom
