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Sildenafil citrate yog cov tshuaj noj uas paub zoo tshaj plaws nyob rau hauv lub npe Viagra, tsim los ntawm Pfizer thiab thawj zaug pom zoo los ntawm FDA hauv 1998. Interestingly, nws tsis tau tsim rau erectile kawg (ED) txhua. Cov kws tshawb fawb tau pib sim nws li kev kho mob rau angina - mob hauv siab los ntawm kev txwv cov ntshav mus rau lub plawv. Hauv kev sim tshuaj, cov txiv neej cov neeg koom tau qhia txog qhov tshwm sim tsis zoo thiab tsis xav txog: txhim kho erections. Cov tshuaj tau rov ua dua, thiab nws tau los ua thawj qhov kev kho qhov ncauj ntawm nws hom.

Xa kev nug
Hauj lwm lawm

    Sildenafil Tiag tiag yog dab tsi

Sildenafil citrate yog cov tshuaj noj uas paub zoo tshaj plaws nyob rau hauv lub npe Viagra, tsim los ntawm Pfizer thiab thawj zaug pom zoo los ntawm FDA hauv 1998. Interestingly, nws tsis tau tsim rau erectile kawg (ED) txhua. Cov kws tshawb fawb tau pib sim nws li kev kho mob angina - mob hauv siab los ntawm kev txwv cov ntshav mus rau lub plawv. Hauv kev sim tshuaj, cov txiv neej cov neeg koom tau qhia txog qhov tshwm sim tsis zoo thiab tsis xav txog: txhim kho erections. Cov tshuaj tau rov ua dua, thiab nws tau los ua thawj qhov kev kho qhov ncauj ntawm nws hom.

Chemically, sildenafil belongs rau chav kawm hu uaphosphodiesterase type 5 (PDE5) inhibitors. Txhawm rau kom nkag siab qhov ntawd txhais tau li cas, nws yuav pab kom paub tias erection ua haujlwm li cas. Kev sib deev stimulation ua rau kev tso tawm ntawm nitric oxide nyob rau hauv cov ntaub so ntswg penile, uas nce qib ntawm ib tug messenger molecule hu ua cGMP. cGMP relaxes cov nqaij ntshiv hauv cov hlab ntsha, tso cai rau cov ntshav kom puv lub erectile chamber. Lub enzyme PDE5 rhuav tshem cGMP, xaus cov nyhuv. Sildenafil blocks PDE5, yog li cGMP nyob ntev dua thiab cov ntshav - ntws cov lus teb muaj zog thiab ruaj khov dua.

Ob lub ntsiab lus ua raws li cov txheej txheem no uas ntau tus neeg to taub yuam kev:

1.Sildenafil tsis tsim ib qho erection ntawm nws tus kheej.Kev sib deev arousal yuav tsum tau pib lub nitric oxide cascade. Nws ua kom cov txheej txheem ntuj tsim; nws tsis hloov nws.

2.Nws tsis yog aphrodisiac.Nws tsis cuam tshuam rau libido, muaj siab, lossis testosterone.

Tshaj li ED, sildenafil (nyob rau hauv ib hom tshuaj sib txawv, Revatio, ntawm koob tshuaj qis) kuj tau pom zoo los kho.pulmonary arterial hypertension, vim tib cov ntshav-cov hlab ntsha- so kom txaus ua kom lub siab nyob hauv cov hlab ntsha ntawm lub ntsws.

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Cov yam ntxwv tseem ceeb thiab cov yam ntxwv

● Pib:feem ntau 30-60 feeb tom qab nqos ib ntsiav tshuaj ntawm lub plab khoob. Ib qho hnyav, siab - pluas mov rog tuaj yeem ncua kev nqus thiab ua rau cov nyhuv.

● Lub sijhawm muaj txiaj ntsig zoo:kwv yees li 4 teev, nrog maj mam taper. Qhov no yog qhov rais ntawmkev teb, tsis yog plaub - teev erection.

● Daim ntawv:Cov ntsiav tshuaj ntawm qhov ncauj, feem ntau 25mg, 50mg, thiab 100mg muaj zog.

●Generics:txij li thaum Pfizer's patent tas sij hawm, generic sildenafil yog dav muaj thiab bioequivalent, uas tau txo tus nqi ntau heev.

● Kev tshuaj xyuas raws li txoj cai:nyob rau hauv feem ntau lub teb chaws nws yuav tsum tau ib daim ntawv tshuaj, vim hais tias nws cuam tshuam txaus ntshai nrog tej yam tshuaj mob plawv - ntxiv rau qhov hauv qab no.

Daim ntawv thov thiab leej twg Nws pab

Thawj daim ntawv thov yogerectile kawg- qhov tsis muaj peev xwm ua tiav lossis tswj kom muaj zog txaus rau kev sib deev txaus siab. ED tsis yog ib yam kab mob nkaus xwb tab sis yog cov tsos mob uas muaj ntau cov hauv paus hniav:

● Cov hlab ntsha ua rau(feem ntau): atherosclerosis, ntshav siab, roj cholesterol siab, ntshav qab zib, thiab kev haus luam yeeb tag nrho cov hlab ntshav ntawm tes. Qhov tseeb, ED feem ntau yog ib qhoceeb toom ntxovntawm cov kab mob plawv, vim cov hlab ntsha penile yog nqaim dua li coronary sawv daws yuav thiab clog sai dua.

● Psychological ua rau:kev ua haujlwm ntxhov siab, kev ntxhov siab, kev nyuaj siab, thiab kev sib raug zoo nyuaj. Ntawm no sildenafil feem ntau ua haujlwm rau "txoj kev ntseeg siab" - rov ua haujlwm txhim khu kev qha thaum qhov teeb meem tshwm sim.

●Mixed ua rau:Feem ntau hauv cov txiv neej tshaj 40 xyoo, qhov teeb meem ntawm lub cev ua rau muaj kev ntxhov siab uas ua rau nws.

● Kev siv qhov xwm txheej:qee tus txiv neej uas muaj kev ua haujlwm ib txwm raug sau tseg nws tawm - daim ntawv lo rau cov xwm txheej tshwj xeeb, xws li kev ua haujlwm tsis zoo los ntawm SSRI tshuaj tiv thaiv kev ntxhov siab.

Nws tsim nyog sau cia tias sildenafil yog dab tsitsis yogpom zoo los yog pab tau rau: tsis muaj libido, ejaculation ntxov ntxov (uas yog lub sij hawm qhov teeb meem, tsis yog ib tug ntshav-flow teeb meem), infertility, los yog noov o. Cov kev thov hauv cov cheeb tsam no yog kev lag luam cov ntawv tseeb.

Cov txiaj ntsig, Hais Honestly

Cov ntaub ntawv kho mob muaj zog. Hauv kev sim thiab ntau xyoo ntawm kev siv tiag tiag - ntiaj teb no, feem ntau ntawm cov txiv neej nrog ED qhia txog kev txhim kho tseem ceeb ntawm PDE5 inhibitors, nrog sildenafil muaj cov ntaub ntawv ceev tshaj plaws ntawm cov chav kawm. Cov txiaj ntsig txuas ntxiv dhau ntawm kev siv tshuab:

●Restored spontaneity thiab kev ntseeg siab:lub nra ntawm lub hlwb ntawm ED - kev cia siab rau kev ntxhov siab, kev zam ntawm kev sib raug zoo - feem ntau nqa ib zaug ua haujlwm tau zoo dua.

● Kev sib raug zoo:Cov neeg koom tes tsis tu ncua qhia txog kev txaus siab thiab kev sib txuas lus hauv kev tshawb fawb txog kev kho ED.

● Kev kuaj mob plawv:nrhiav kev kho mob feem ntau ua rau kev tshawb pom ntawm qhov tsis pom kev mob ntshav siab, ntshav qab zib, lossis teeb meem cholesterol. Hauv qhov kev nkag siab ntawd, "cov txiaj ntsig" tuaj yeem yog lub neej- txuas mus rau txoj kev sib txawv kiag li.

● Tsis yog -invasiveness:piv rau kev txhaj tshuaj, tshuaj suppositories, lub tshuab nqus tsev nqus tsev vacuum, los yog implants, ib ntsiav tshuaj yog nyob deb ntawm qhov tsawg tshaj plaws intrusive thawj - kab xaiv.

Dosage: Yuav ua li cas lub zog 100mg Fits In

Tus qauv pib koob tshuaj rau cov txiv neej feem ntau yog50mg ib, noj li ntawm ib teev ua ntej xav txog kev sib deev. Raws li kev ua tau zoo thiab kev ua siab ntev, tus kws kho mob tuaj yeem hloov kho mus rau 25mg lossis ntau dua100mg - qhov siab tshaj plaws pom zoo koob tshuaj. Cov cai tseem ceeb:

● Tsis txhob ntau tshaj ib koob tshuaj rau 24 teev.

●100mg yog lub qab nthab, tsis yog lub hom phiaj.Tsis zoo dua: koob tshuaj ntau dua ua rau muaj qhov tshwm sim ntawm cov kev mob tshwm sim (mob taub hau, lub ntsej muag yaug, qhov ntswg congestion, plab zom mov, ib ntus xiav - tinged tsis pom kev) yam tsis tau lees paub qhov txiaj ntsig zoo dua.

● qis pib koob tshuajyog cov qauv rau cov txiv neej tshaj 65 xyoo, cov neeg uas muaj lub siab lossis lub raum tsis zoo, thiab cov tshuaj tiv thaiv kab mob (qee cov tshuaj tiv thaiv kab mob, HIV protease inhibitors, qee cov tshuaj tua kab mob).

● Noj ntawm lub plab khoob lossis lub plabrau qhov ua tau zoo tshaj plaws, thiab mus yooj yim ntawm cawv - nws ob qho tib si blunts cov tshuaj ua thiab nws tus kheej impairs erections.

Kev ceeb toom kev nyab xeeb tseem ceeb

Sildenafil yuav tsumyeej tsisua ke nrog nitrates (nitroglycerin, isosorbide - siv rau mob hauv siab) lossis ua si "poppers" (amyl nitrite). Kev sib xyaw ua ke tuaj yeem ua rau muaj kev puas tsuaj loj hauv ntshav siab. Kev ceev faj thiab kev saib xyuas kev kho mob kuj tseem yuav tsum tau nrog alpha-blockers thiab hauv cov txiv neej uas tsis muaj kab mob plawv. Ib qho erection ntev tshaj li plaub teev (priapism) yog kev kho mob xwm txheej ceev.

"Lub voj voog" thiab "PCT": Kho Cov Lus Tsis Txaus Siab

Cov ntsiab lus no suav nrog kev siv tshuaj anabolic steroid, qhov twg "lub voj voog" txhais tau hais tias lub sijhawm npaj rau thiab tawm cov tshuaj hormones, thiab "PCT" (post- kev kho lub voj voog) txhais tau hais tias cov tshuaj noj tom qab ntawd rov pib lub cev ntawm tus kheej testosterone ntau lawm, uas steroids suppress.

●Sildenafil tsis muaj lub voj voog thiab tsis muaj PCT, vim nws tsis kov cov tshuaj hormones lossis cov kab mob endocrine.Nov yog qhov kev sib cais:

● Tsis muaj kev txwv:Sildenafil tsis cuam tshuam rau testosterone, estrogen, LH, FSH, lossis lwm yam tshuaj hormones. Tsis muaj dab tsi los "rov pib dua."

● Tsis muaj kev vam khom hauv lub cev lub cev:Nws tsis ua rau muaj kev zam txim rau cov neeg siv feem ntau, thiab txwv tsis pub nws yuav tsis thim tawm. (Kev cia siab ntawm kev puas siab puas ntsws yog ua tau - qee tus txiv neej tuaj yeem xav tias lawv ua tsis tau yam tsis muaj nws - tab sis qhov ntawd yog qhov teeb meem kev ntseeg siab, tsis yog kws tshuaj.)

●Siv yog qhov xwm txheej-raws li, tsis yog voj voog-raws li:Nws tau noj raws li qhov xav tau, thaum xav txog kev sib deev, nrog tsawg kawg 24 teev ntawm koob tshuaj. Tsis muaj kev nce qib - nce, taper, lossis lub sijhawm rov qab los.

Qhov tsis meej pem tuaj qhov twg? Cov zej zog tsim lub cev qee zaum siv sildenafilthaumlub voj voog steroid - ib nrab rau cov nyhuv "tswj" hauv lub gym, ib feem los tiv thaiv steroid- ntxias kev sib deev tsis ua haujlwm - thiab qee qhov kev sib tham hauv online piav qhia qhov no yog ib feem ntawm "lub voj voog" lossis txawm tias PCT raws tu qauv. Qhov ntawd yog kev tawm ntawm -label, zej zog- tsim kev xyaum, tsis yog kev kho mob. Yog tias cov tshuaj anabolic steroids tau ua rau muaj kev sib deev tsis ua haujlwm, cov lus teb yog kev ntsuam xyuas endocrine thiab kev rov zoo ntawm cov tshuaj hormone axis, tsis yog PDE5 inhibitor npog cov tsos mob.

Ib nrab-Lub Neej thiab Pharmacokinetics

Sildenafil muaj ibib nrab-lub neej ntawm kwv yees li 3-5 teevnyob rau hauv cov neeg laus noj qab nyob zoo - txhais tau tias ntshav concentration poob los ntawm ib nrab ntawm lub qhov rais. Qhov no yog vim li cas lub qhov rais ua haujlwm zoo nyob ib puag ncig 4 teev. Tom qab tsib ib nrab -nyob (kwv yees ib hnub), cov tshuaj yog qhov tseem ceeb tshem tawm ntawm lub cev. Nws cov metabolite tseem ceeb, N-desmethylsildenafil, kuj tseem ua haujlwm thiab muaj ib nrab zoo sib xws -lub neej. Kev tshem tawm feem ntau yog los ntawm daim siab thiab quav. Rau kev sib piv, nws cov kwv tij kwv tij tadalafil (Cialis) muaj ~ 17.5-teev ib nrab- lub neej, uas yog vim li cas tadalafil tau ua lag luam txog li 36-teev kev pab them nqi - ib qho tshuaj pharmacokinetic tiag tiag uas tsim nyog paub thaum tham txog kev xaiv nrog kws kho mob.

Cov ntaub ntawv kho mob

Hom

STROMUSC

Cov npe lag luam

Viagra, Sildenafil, Revatio

CAS

139755-83-2

Molar loj

474.6

Formula

C22H30N6O4S

Purity

Tshaj 98%

Yam khoom

100 mg x 100

 

 

Txhua yam kev xav tau, thov hu rau peb

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Kab hauv qab

Sildenafil 100mg yog qhov siab tshaj plaws - koob tshuaj lub zog ntawm lub qhov dej- tau kawm, feem ntau muaj kev nyab xeeb cov tshuaj uas kho erectile kawg los ntawm kev txhim kho lub cev cov ntshav - ntws teb rau arousal. Siv kom raug - raws li qhov xav tau, tsis pub ntau tshaj ib zaug ib hnub, tsis muaj nitrates, raws li kev qhia kho mob - nws tau rov qab ua haujlwm ntawm kev sib deev thiab kev ntseeg siab rau ntau pua lab tus txiv neej. Nws tsis muaj lub voj voog, tsis tas yuav tsum muaj PCT, tsim tsis muaj hormonal dependence, thiab ua haujlwm zoo tshaj plaws raws li ib feem ntawm daim duab loj: kev noj qab haus huv ntawm lub plawv, kev sib txuas lus ncaj ncees nrog tus khub, thiab kev ntsuam xyuas kev kho mob kom paub seb vim li cas ED tshwm sim thawj zaug.

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