
Dostinex (Cabergoline) Lub Cev Lub Cev Lub Cev Muaj Zog CAS: 81409-90-7
Cabergoline yog thawj zaug siv rau kev kho mob hauv xyoo 1993. Nws yog feem ntau siv los kho cov qib prolactin siab. Nws kuj yog siv rau hauv kev kho mob ntawm Prolactinomas thiab Parkinson tus kab mob. Txij thaum ntawd los, nws kuj tau siv dav hauv bodybuilding rau ntxiv qhov hnyav rau lub cev hnyav. Thaum xyoo 1990s lig, qee qhov kev mob tshwm sim tau pib tawm ntawm qhov kev siv no thiab qhov no ua rau nws raug txwv los ntawm ntau lub tebchaws rau lub hom phiaj tsim lub cev. Cabergoline tau pom tias nce qib prolactin hauv cov neeg mob. Nws kuj tseem tuaj yeem ua rau lub sijhawm ntev ntawm galactorrhea thiab gynecomastia. Qhov no yog vim li cas rau ntau lub teb chaws txwv tsis pub siv Cabergoline hauv kev tsim lub cev thaum xyoo 1990s.
Cabergoline yog thawj zaug siv rau kev kho mob hauv xyoo 1993. Nws yog feem ntau siv los kho cov qib prolactin siab. Nws kuj yog siv rau hauv kev kho mob ntawm Prolactinomas thiab Parkinson tus kab mob. Txij thaum ntawd los, nws kuj tau siv dav hauv bodybuilding rau ntxiv qhov hnyav rau lub cev hnyav. Thaum xyoo 1990s lig, qee qhov kev mob tshwm sim tau pib tawm ntawm qhov kev siv no thiab qhov no ua rau nws raug txwv los ntawm ntau lub tebchaws rau lub hom phiaj tsim lub cev. Cabergoline tau pom tias nce qib prolactin hauv cov neeg mob. Nws kuj tseem tuaj yeem ua rau lub sijhawm ntev ntawm galactorrhea thiab gynecomastia. Qhov no yog vim li cas rau ntau lub teb chaws txwv tsis pub siv Cabergoline hauv kev tsim lub cev thaum xyoo 1990s.
Nws yog feem ntau siv los tiv thaiv cov kev mob tshwm sim tsis zoo ntawm progesterone tshwm sim los ntawm kev siv AAS vim tias nws qhov cuam tshuam ncaj qha rau 5 -reductase. Tsis tas li ntawd, finasteride feem ntau yog siv ua ke nrog AAS kom txo tau qhov muaj feem cuam tshuam los ntawm kev siv AAS los ntawm kev txo qis DHT. Nws kuj tau pom tias muaj qee yam tshuaj tua kab mob thiab tshuaj tua kab mob, uas tej zaum yuav cuam tshuam rau nws lub peev xwm los inhibit ntau yam enzymes ntsig txog steroidogenesis. Finasteride yog cadaverine-type inhibitor ntawm 5 -reductase thiab yog ib qho kev sib tw inhibitor ntawm 5 -reductase. Nws tiv thaiv kev hloov pauv ntawm androgen, dihydrotestosterone (DHT), rau hauv daim ntawv muaj zog ntau ntawm testosterone, los ntawm kev tiv thaiv cov enzyme no los ntawm kev khi rau qhov chaw nquag. Lub tshuab molecular ntawm finasteride tsis nkag siab tag nrho, tab sis nws xav tias yuav ua haujlwm raws li hauv qab no: Nws khi rau thiab inhibits enzyme 5 -reductase, uas hloov testosterone rau hauv DHT. Qhov no tiv thaiv kev hloov pauv ntawm testosterone rau hauv DHT, uas txo nws cov qib hauv lub cev thaum tib lub sijhawm txo cov prostate ntim.


Cov ntaub ntawv sib xyaw
Caber yog ib qho tshuaj ntawm qhov ncauj uas feem ntau tuaj hauv {{0}}.25, 0.5, thiab 1mg koob. Qhov no txhais tau tias Cabergoline muaj qhov nqus tsawg heev. Ib nrab-lub neej ntawm Cabergoline yog nyob ib ncig ntawm 5 teev. Qhov no txhais tau hais tias nws muaj lub sijhawm ntev heev ntawm kev nqis tes ua thiab tsis tas yuav tsum tau ua txhua hnub.
Cabergoline yog dopamine D2 receptor agonist. Qhov no txhais tau hais tias nws ua haujlwm los ntawm kev khi rau dopamine receptors los tiv thaiv kev tso tawm ntawm prolactin. Cov kws tsim lub cev uas siv cabergoline txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau nws, cov kws kho mob lub cev yuav tsum tau ceev faj saib xyuas lawv cov qib thiab xyuas kom meej tias lawv tsis siab dhau. Rimonabant yog cannabinoid receptor antagonist. Qhov no txhais tau hais tias nws tiv thaiv kev ua haujlwm ntawm CB1 receptors, uas yog lub luag haujlwm rau ntau lub cev ua haujlwm, suav nrog kev noj zaub mov. Hauv ntau lub tebchaws xws li Brazil thiab Tuam Tshoj, rimonabant tsuas yog cov tshuaj uas tau pom zoo rau kev kho mob ntawm kev nyuaj siab.
Olanzapine yog atypical antipsychotic. Nws ua haujlwm los ntawm kev nce dopamine txhawm rau txhawm rau txhim kho kev xav zoo thiab txo cov kev xav tsis zoo, xws li kev ntxhov siab thiab kev nyuaj siab. Olanzapine kuj tseem muaj txiaj ntsig zoo rau qee cov neeg uas muaj tus mob schizophrenia, uas tej zaum yuav muaj lub zog manic.
Cabergoline yog dopamine D2 receptor agonist. Qhov no txhais tau hais tias nws ua haujlwm los ntawm kev khi rau dopamine receptors los tiv thaiv kev tso tawm ntawm prolactin. Cov kws tsim lub cev uas siv cabergoline txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau txhawm rau nws, cov kws kho mob lub cev yuav tsum tau ceev faj saib xyuas lawv cov qib thiab xyuas kom meej tias lawv tsis siab dhau.
Nws kuj yog ib qho chaw nrov ua haujlwm nrog Nandrolone raws li steroids. Cov tshuaj steroids nce progesterone thiab prolactin hauv lub cev uas tuaj yeem ua rau muaj kev phiv tsis zoo xws li txo qis libido, dej tuav, lossis gynecomastia. Qhov no yog vim li cas qee tus neeg tsim lub cev xaiv siv cov tshuaj anabolic steroid Primobolan yam tsis muaj qhov sib xyaw no, ua lwm txoj hauv kev nyab xeeb. Primobolan kuj tau pom tias ua rau lub siab puas tsuaj hauv qee qhov kev tshawb fawb.
Cabergoline bodybuilding voj voog cov ntaub ntawv
Thaum lub sij hawm Cabergoline bodybuilding lub voj voog nrog rau nandrolone raws li cov tebchaw xws li trenbolone, NPP, lossis Deca, nws raug nquahu kom muaj qee lub caber ntawm tes yog tias muaj kev phiv progestogenic. Yog hais tias ib qho ntawm cov teeb meem no yuav tsum tshwm sim ces ib lub lim tiam koob tshuaj ntawm 0.25mg ib lub lis piam. Qhov no tej zaum yuav muaj tsawg dua rau cov poj niam uas tsis hnov mob rau progestogens vim tias lawv cov tshuaj estrogen qis, lossis nws yuav muaj ntau dua yog tias lawv muaj cov qib endogenous progestogenic siab. Caber yog lub npe hu ua tshuaj tiv thaiv kab mob hauv qhov ncauj, thiab tuaj yeem siv los kho ib qho ntawm cov kev mob tshwm sim saum toj no. Nws kuj yog ib qho kev kho mob zoo heev rau kev los ntshav ntau dhau thaum cev xeeb tub thiab tuaj yeem ua ke nrog norethindrone txhawm rau txhawm rau los ntshav tib lub sijhawm.
Nandrolone yog ib qho 19-tsis yog steroid derivative ntawm testosterone thiab muaj cov qauv zoo sib xws ntawm cov tshuaj hormonal. Nws kuj yog ib qho ntawm cov muaj zog tshaj plaws anabolic steroids nyob rau hauv kev ua lag luam, tab sis hmoov tsis, nws qhia qhov zoo ntawm no nrog ob peb lwm yam tshuaj uas muaj ntau yam tshuaj lom los yog raug txwv tsis pub siv tag nrho los ntawm WADA. Vim qhov tseeb tias nws muaj zog, qee qhov anabolic-androgenic steroids (AAS) uas muaj nandrolone yog siv los ua kev ua tau zoo ntawm cov tshuaj hauv kev ua si. Anabolic androgenic steroids (AAS) uas muaj nandrolone muaj xws li oxandrolone, methandienone, thiab stenbolone.
Yog tias cov Nandrolone raws li cov khoom sib xyaw no tau siv ces nws kuj tseem pom zoo kom ntxiv caber rau hauv koj li PCT raws tu qauv nrog Nolva, Clomid thiab HCG. Rau lub hom phiaj no, koob tshuaj yuav nyob ib ncig ntawm {{0}}.5mg ib lub lis piam thiab qhov no yuav muab faib ua ob koob tshuaj 0.25mg ib lub lis piam.
Cov txiaj ntsig xav tau
Caber yog ib qho muaj zog sib xyaw ua ke yog li cov teebmeem yuav pom tau sai sai, cov kev tshawb fawb pom tias qhov txo qis hauv cov qib prolactin sai li sai tau 3 teev hauv qee cov neeg siv vim muaj ntau txoj hauv kev dopamine thiab txo txoj hauv kev serotonin hauv lub hlwb. Cov kev tshawb fawb tseem qhia tau tias nce qib dopamine thiab noradrenaline ntxiv nrog rau kev txo qis hauv acetylcholine, uas qhia tau tias lwm cov neurotransmitters raug tso tawm los teb rau cov teebmeem ntawm caber.
Cov neeg siv kuj tuaj yeem ntsib kev pw tsaug zog zoo dua thiab ua kom pom tseeb vim muaj kev txhim kho REM pw tsaug zog thiab cov teebmeem ntawm dopamine. Caber kuj tau pom tias muaj kev nkag siab zoo ntawm kev noj qab haus huv, kev cia siab thiab kev nkag siab ntawm kev ntxhov siab. Qhov no yog vim citicoline ua rau cov neurotransmitters xws li serotonin, dopamine thiab norepinephrine. Caber kuj tseem yuav pab tau rau kev kho mob me me ntawm kev paub tsis meej uas cuam tshuam nrog kev laus. Qhov no yog vim nws tau pom tias muaj cov txiaj ntsig tseem ceeb hauv kev txhim kho kev hais lus zoo, nco thiab mloog.
Kuj tseem yuav muaj qhov nce hauv libido txij li Caber zoo li ua rau kev tso tawm ntawm testosterone thiab estrogen. Nws tsis paub tias qhov no cuam tshuam li cas rau fertility vim tsis muaj kev tshawb fawb hauv cheeb tsam no. Caber kuj tau pom tias muaj cov khoom tiv thaiv kabmob kheesxaws uas tuaj yeem siv los kho mob qog noj ntshav, vim nws cov teebmeem ntawm cell proliferation, autoimmunity thiab apoptosis.
Bodybuilders uas siv Caber hauv lawv cov kev tswj hwm kuj tseem tuaj yeem muaj kev nce hauv cov leeg nqaij vim nws txo lub cev rog thiab pab txhawb kev nqus ntawm lwm cov leeg nqaij. Cov nyhuv inhibitory ntawm Caber ntawm aromatase yuav txo qis cov tshuaj estrogen tsim los ntawm lub cev, uas tuaj yeem cuam tshuam libido vim nws inhibits kev sib deev hormone-binding globulin (SHBG) qib, nrog rau nce qib testosterone. Txawm li cas los xij, qhov kev cuam tshuam no yog thim rov qab thiab txawm tias nws yuav muaj txiaj ntsig, tsis muaj pov thawj los qhia tias nws tsim nyog rau cov leeg nqaij. Tsis muaj kev tshawb fawb tau tshawb xyuas qhov ua tau zoo ntawm Caber hauv kev nce lean pawg, txawm li cas los xij, muaj cov kev tshawb fawb uas qhia tias nws tuaj yeem pab txhawb cov leeg nqaij thaum lub sij hawm anabolic steroid cycles vim nws cov nyhuv stimulatory ntawm 5-alpha reductase thiab inhibition ntawm aromatase.
Yuav ua li cas ua haujlwm Cabergoline hauv bodybuilding
Cov ntsiab cai zoo sib xws tswj hwm cabergoline lub peev xwm los txhawb cov leeg nqaij. Cov khoom no txhawb cov leeg nqaij loj hlob los ntawm kev txuas mus rau dopamine receptors hauv cov leeg. Qhov tseeb tias cabergoline tuaj yeem pab koj tsim cov leeg loj dua, cov leeg muaj zog yog vim li cas nws thiaj li nrov ntawm bodybuilders. Tsis tas li ntawd, cabergoline tau pom tias yuav ua kom cov nqaij ntshiv rov qab los ntawm kev tawm dag zog, tso cai rau koj rov pib koj lub sijhawm kawm sai dua.
Cabergoline kuj tuaj yeem txhim kho lub cev lub peev xwm los hlawv rog. Qhov no yog vim li cas cabergoline nce lub cev qhov siab ntawm lipolytic enzymes uas ua rau cov rog kom tawg thiab hloov mus rau lub zog. Cabergoline kuj tseem pab txhawb kev qab los noj mov, uas ua rau nws yooj yim dua los tswj kev noj zaub mov kom zoo. Qhov txiaj ntsig no yog ib feem ntawm cov tshuaj muaj peev xwm nce qib serotonin hauv lub cev, uas cuam tshuam rau lub siab zoo siab thiab noj tsawg dua.
Vim li cas Cabergoline hauv Bodybuilding thiaj li nrov?
Qhov nrov ntawm cabergoline hauv kev tsim lub cev ntawm cov neeg siv tuaj yeem raug ntaus nqi rau ntau yam. Ua ntej ntawm tag nrho cov, nws tau raug pom tias yog ib tug muaj zog cov leeg tsim. Cabergoline kuj tseem txhawb nqa lub zog thiab lub zog, ua rau nws yog qhov kev xaiv zoo heev rau cov neeg uas xav thawb lawv tus kheej mus rau qhov siab tshaj plaws. Qhov thib ob, cabergoline paub zoo rau kev pab hauv kev rog rog thiab txhawb nqa qhov hnyav. Qhov no ua rau nws zoo meej rau txhua tus neeg uas xav kom poob phaus thiab ua kom zoo. Thaum kawg, thaum siv raws li kws kho mob tau sau tseg, cabergoline feem ntau muaj kev nyab xeeb thiab muaj kev cuam tshuam tsawg heev. Koj tuaj yeem ua tiav koj lub hom phiaj nrog kev pab ntawm cabergoline, lub cuab yeej tshiab thiab ntxim nyiam rau cov kws tsim lub cev.
Cabergoline Qhov hnyav poob cuam tshuam rau kev loj hlob Hormones
Kev loj hlob hormone ntau lawm yog ib qho ntawm Cabergoline qhov zoo tshaj plaws intriguing. Kev loj hlob cov tshuaj hormones yog qhov tseem ceeb rau kev noj qab haus huv qhov hnyav nrog rau kev loj hlob thiab kev loj hlob ntawm cov leeg. Ib qho ntawm ob peb cov tshuaj uas tau ua pov thawj kom nce qib ntawm kev loj hlob hormone yog cabergoline. Yog li ntawd nws yog qhov kev xaiv zoo tshaj plaws rau bodybuilders uas xav txhim kho lawv txoj kev loj hlob.
Cov kws tshawb fawb tau saib seb cabergoline cuam tshuam li cas rau qib ntawm kev loj hlob hormone hauv cov neeg noj qab haus huv. Raws li kev tshawb fawb, cabergoline tuaj yeem txhawb kev loj hlob cov tshuaj hormones nce mus txog ob zaug. Cov kws tshawb fawb kuj tau tshawb pom tias cabergoline nce qib ntawm IGF-1, qhov tseem ceeb ntawm kev loj hlob hormone. Qhov no qhia tau hais tias cabergoline tuaj yeem pab txhim kho kom muaj zog thiab cov leeg loj.
Cabergoline, paub txog nws cov ntawv kho mob, tau pom muaj peev xwm poob phaus. Cov kev tshawb fawb qhia tias nws tuaj yeem tswj kev qab los noj mov, txo kev ntshaw, thiab txhawb kev rog. Txawm li cas los xij, kev saib xyuas kev kho mob kom raug thiab kev taw qhia yog tsim nyog ua ntej txiav txim siab Cabergoline rau kev poob phaus. Kev sab laj nrog tus kws kho mob yog qhov tseem ceeb los txiav txim siab txog qhov tsim nyog npaum li cas thiab ntsuas txhua qhov kev pheej hmoo.
Cabergoline Bodybuilding Stacks
Cabergoline tuaj yeem siv ib leeg lossis ua ke nrog lwm cov tshuaj los tsim ntau yam txiaj ntsig. Qee qhov zoo-nyiam cabergoline stacks rau bodybuilding yog teev hauv qab no:
Kev loj hlob hormone nrog cabergoline: Cabergoline yog qhov kev xaiv zoo heev rau cov neeg tsim lub cev uas xav ua kom zoo dua lawv cov txiaj ntsig vim nws tuaj yeem nce qib cov tshuaj hormones.
IGF-1, lwm qhov tseem ceeb ntawm kev loj hlob hormone, thiab cabergoline tuaj yeem nce qib ntawm IGF-1.
Testosterone thiab cabergoline: Cabergoline tuaj yeem pab koj nce qib ntawm testosterone, uas tuaj yeem txhim kho koj lub zog, kev ua siab ntev, thiab cov leeg nqaij.
SARMs, ib hom tshuaj uas tuaj yeem pab koj nce cov leeg nqaij thiab txo cov rog, ua haujlwm zoo nrog cabergoline. Koj tuaj yeem ua kom tiav qhov cuam tshuam ntawm koj lub voj voog SARMs nrog kev pab ntawm cabergoline.
HCG nrog cabergoline: HCG yog ib yam tshuaj uas tuaj yeem pab koj txo qhov hnyav thaum tswj koj cov leeg nqaij. Koj tuaj yeem ua kom cov txiaj ntsig zoo ntawm koj lub voj voog HCG los ntawm kev siv cabergoline.
Cov ntaub ntawv kho mob
|
Cov npe lag luam |
Dostinex, Cabergoline |
|
CAS |
81409-90-7 |
|
Molar loj |
451.615 |
|
Formula |
C26H37N5O2 |
|
Purity |
Tshaj 98% |
|
Yam khoom |
0.25mg*100 |
Txhua yam kev xav tau, thov hu rau peb
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tswv yim
Cabergoline rau poob phaus
Cabergoline txhawb nqa qhov hnyav los ntawm kev txo qis qab los noj mov thiab, yog li, calorie noj. Cabergoline kuj nce basal metabolic tus nqi, uas ua rau muaj calorie ntau ntau hlawv. Tsis tas li ntawd, nws pab tswj thiab khaws cov leeg nqaij thaum noj zaub mov. Yog li ntawd, cabergoline tsis tsuas yog pab kom poob phaus tab sis kuj tswj cov leeg nqaij.
Cov neeg uas xav kom poob yim nrog kev pab ntawm Caber yuav tsum siv cov khoom noj uas txo qhov hnyav nrog kev noj zaub mov qis thiab kev tawm dag zog. Cabergoline yog siv los kho mob hnyav ntawm premenstrual dysphoric teeb meem, uas cuam tshuam txog li 12% ntawm cov poj niam thoob ntiaj teb. Tus mob no yog tus cwj pwm los ntawm kev hloov siab lees txim, kev nyuaj siab thiab kev chim siab thaum coj khaub ncaws. Nws kuj yog siv los kho tus kab mob Parkinson .Cabergoline kuj tseem siv los ua cov tshuaj tiv thaiv kab mob los kho qee yam mob qog noj ntshav.
Caber tseem tuaj yeem pab tib neeg kom poob phaus los ntawm kev txo qis kev tso tawm ntawm qee cov tshuaj hormones hauv plab hnyuv uas tuaj yeem ua rau overeating. Qhov no yog xov xwm zoo rau cov neeg uas xav kom poob phaus, tab sis nws kuj tuaj yeem ua rau muaj kev phiv. Qee qhov kev mob tshwm sim ntawm cilantro yog mob thiab ntuav.
Cabergoline rau cov leeg loj hlob
Cabergoline yog qhov zoo rau cov leeg nqaij vim nws nce qib ntawm IGF-1 thiab kev loj hlob hormone, ob qho tib si tsim nyog rau cov leeg nqaij. Tsis tas li ntawd, cabergoline ua kom koj rov qab los tom qab kev tawm dag zog kom koj tuaj yeem tawm dag zog thiab tau txais txiaj ntsig ntau dua. Cabergoline yog cov tshuaj zoo tshaj plaws rau cov neeg tsim lub cev uas xav txo cov rog thaum ua kom lawv cov leeg nqaij vim nws kuj pab tiv thaiv cov leeg nqaij thaum lub sij hawm txo qhov hnyav. Cov tshuaj no yog ib qho kev xaiv nrov ntawm cov zej zog tsim lub cev, thiab nws kuj tau siv los kho tus kab mob Parkinson.
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