
BNP Cialis (Tadanafil) Rau Kev Sib Deev CAS: 171596-29-5
Cialis, lub npe lag luam rau Tadalafil, yog cov tshuaj feem ntau paub txog kev kho erectile kawg (ED). Tau ntau xyoo, nws tau txais kev saib xyuas rau nws cov ntawv thov sib txawv, cov khoom siv tshuaj, thiab cov txiaj ntsig kho mob. Hauv phau ntawv qhia ntxaws ntxaws no, peb yuav tshawb txog Cialis los ntawm ntau lub ces kaum, suav nrog nws cov tshuaj profile, cov txheej txheem ntawm kev txiav txim, kev siv tshuaj kho mob thiab cov ntawv sau tawm, cov txiaj ntsig, ntau npaum li cas, ib nrab-lub neej, kev ncig, thiab lub luag haujlwm uas nws tuaj yeem ua hauv cov kev kho mob tshwj xeeb. .
Cialis yog dab tsi?
Cialis yog phosphodiesterase type 5 (PDE5) inhibitor tsim los txhim kho cov ntshav khiav thiab so cov leeg nqaij. Pom zoo los ntawm FDA hauv 2003 rau kev kho mob ntawm erectile kawg, nws tau txij li thaum tau siv rau lwm yam mob, xws li benign prostatic hyperplasia (BPH) thiab pulmonary arterial hypertension.
Tadalafil txawv nws tus kheej los ntawm lwm yam PDE5 inhibitors zoo li Viagra (Sildenafil) vim nws lub neej ntev dua, tau txais nws lub npe menyuam yaus "Lub lis piam Pill." Nws txoj kev ua tau zoo, kev ua siab ntev, thiab ncua sij hawm ntawm kev txiav txim ua rau nws yog qhov kev xaiv zoo rau ntau tus.


Cov khoom ntawm Cialis
Tshuaj muaj pes tsawg leeg
● Cov Qauv Tshuaj: C22H19N3O4
● Molecular LujYog ': 389.4 g/mol
● Mechanism of Action: Xaiv inhibition ntawm PDE5 enzyme, nce cyclic guanosine monophosphate (cGMP) ntau ntau.
Pharmacokinetics
● Absorption: sai sai absorbed nyob rau hauv lub plab zom mov nrog ib tug bioavailability ntawm 80%.
● Peak Plasma Concentration: Ua tiav hauv 2 teev tom qab noj qhov ncauj.
● Ib nrab Lub Neej: Kwv yees li 17.5 teev, ntev dua li lwm cov PDE5 inhibitors.
Cov qauv tsim
Cialis muaj nyob rau hauv ntau npaum li cas, suav nrog:
●2.5 mg ib
●5mg ib
●10 mg
●20 mg
Nws versatility pub rau ob leegsiv txhua hnubntawm cov koob tshuaj qis dua thiabsiv raws li xav tauthaum noj ntau dua.
Mechanism ntawm Action
Cialis aims lubPDE5 enzyme, uas yog lub luag haujlwm rau kev rhuav tshem cGMP hauv cov leeg nqaij. Los ntawm inhibiting PDE5, Cialis txhim kho cov teebmeem ntawm nitric oxide, txhawb kev so ntawm cov leeg nqaij hauv cov hlab ntsha. Qhov no ua rau muaj ntshav ntau ntxiv hauv cov cheeb tsam tshwj xeeb, tshwj xeeb yog corpus cavernosum ntawm noov.
Rau cov xwm txheej zoo li BPH thiab pulmonary hypertension, tib lub tswv yim txhawb kev txhim kho kev ncig thiab txo cov leeg nqaij nruj hauv cov hlab ntsha prostate thiab pulmonary arteries.
Kev siv ntawm Cialis
A. Cov ntawv thov kho mob
1.Erectile Dysfunction (ED):
●Qhov taw qhia tseem ceeb rau Cialis, nws pab cov txiv neej ua tiav thiab tswj cov erections los ntawm kev txhim kho cov ntshav ntawm tes.
2.Benign Prostatic Hyperplasia (BPH):
●Cialis txo cov tsos mob tso zis los ntawm kev ua kom cov leeg du hauv lub zais zis thiab prostate.
3. Pulmonary Arterial Hypertension (PAH):
●Nws yog qee zaum siv los txo qis cov hlab ntshav siab thiab txhim kho kev tawm dag zog.
4.Kev kho mob sib xyaw:
●Cialis tuaj yeem ua ke nrog alpha-blockers lossis lwm yam tshuaj rau kev tswj hwm cov zis lossis vascular.
B. Off-Label Applications
1. Kev ua kis las:
●Vim nws cov vasodilatory zog, Cialis tuaj yeem txhim kho cov leeg nqaij thiab kev ua siab ntev.
2. Mob plawv:
● Kev tshawb fawb tam sim no qhia tias PDE5 inhibitors zoo li Cialis tuaj yeem pab cov neeg mob plawv tsis ua haujlwm lossis endothelial tsis ua haujlwm.
3. Raynaud's Phenomenon:
●Cialis tau siv los kho tus mob no, uas txo cov ntshav ntws mus rau sab kawg vim vasospasm.
4. Cov txiaj ntsig ntawm kev puas siab puas ntsws:
●Los ntawm kev hais txog ED, Cialis tuaj yeem txhim kho kev hwm tus kheej, txo kev ntxhov siab, thiab txhim kho tag nrho lub neej zoo.
Cov txiaj ntsig ntawm Cialis
1.Nyob ntev:
● Nrog rau ib nrab ntawm lub neej ntawm 17.5 teev, Cialis tseem siv tau ntev txog 36 teev, tso cai rau tus kheej ntau dua piv rau lwm cov tshuaj ED.
2. Yooj yim:
● Tsis tshua muaj koob tshuaj txhua hnub Cialis tshem tawm qhov xav tau ntawm kev npaj raws li qhov xav tau, muab cov txiaj ntsig kho mob zoo ib yam.
3.Kev sib cuam tshuam khoom noj tsawg tsawg:
● Tsis zoo li Viagra, Cialis tsis cuam tshuam los ntawm cov zaub mov muaj roj ntau, muab kev yooj yim dua hauv kev siv.
4.Dual Efficiency:
● Ib txhij kho ED thiab BPH, ua rau nws xaiv ntau yam rau cov txiv neej uas muaj kev sib tshooj.
5. Txhim kho kev ua haujlwm muaj peev xwm:
● Hauv cov neeg mob PAH, Cialis txhim kho cov pa oxygen thiab txo qis ntawm cov hlab ntsha pulmonary.
6. Kev Mob Siab:
● Los ntawm kev hais txog ED kom zoo, Cialis pab txo qis kev ntxhov siab thiab kev sib raug zoo.
Dosage thiab Administration
A. Erectile Dysfunction
1.On-Demand Dosing:
● Hom pib koob tshuaj:10 mg, noj 30-60 feeb ua ntej kev sib deev.
● Kho rau20 mglos yog5mg ibraws li kev ua tau zoo thiab kam rau ua.
2. Noj txhua hnub:
●2.5 mg los yog 5 mgtxhua hnub, zoo tagnrho rau cov txiv neej uas xav tias yuav muaj kev sib deev ntau zaus.
B. Benign Prostatic Hyperplasia
● Pom zoo koob tshuaj:5 mg ib hnub twg, noj tib lub sijhawm txhua hnub.
C. Pulmonary Arterial Hypertension
● Cov koob tshuaj ntau dua (piv txwv li, 40 mg txhua hnub) yuav raug siv raws li kev saib xyuas nruj.
Cov Lus Qhia dav dav:
● Tsis txhob noj ntau tshaj ib koob tshuaj ib hnub.
● Tej zaum yuav muaj kev hloov kho rau cov neeg uas muaj lub raum lossis lub siab tsis zoo.
Pharmacokinetics: Ib nrab-Lub Neej thiab Kev Tshaj Tawm
Cialis qhov ntev ib nrab-lub neej ua kom muaj qhov muaj nyob hauv cov hlab ntsha, tso cai rau:
●Yooj yim rau lub sijhawm ntawm kev sib deev.
●Cov teebmeem kev kho mob ruaj khovrau cov mob ntev xws li BPH.
Metabolism
● Feem ntau metabolized hauv daim siab los ntawm cytochrome P450 enzyme system (CYP3A4).
●Metabolites raug tso tawm los ntawm quav (61%) thiab zis (36%).
Kev tso tawm
●Thaum Cialis tshem tawm cov txheej txheem qeeb dua li qhov ua haujlwm luv luv PDE5 inhibitors, qhov no ua rau nws ua haujlwm ntev dua.
Kev txiav txim siab tom qab kev kho mob (PTC)
Cialis tsis feem ntau cuam tshuam nrog cov tshuaj tiv thaiv hormonal pom nrog anabolic steroids, yog li kev caiKev kho mob tom qab lub voj voog (PCT)yog tsis tsim nyog. Txawm li cas los xij, nyob rau hauv rooj plaub uas Cialis siv nrog rau kev ua tau zoo-txhim kho cov tshuaj, hais txog cov tshuaj hormonal rov qab los ntawm SERMs (Selective Estrogen Receptor Modulators) lossis lwm tus neeg ua haujlwm yuav xav tau.
Cov Kev Phem Phem thiab Kev Phem
Thaum Cialis feem ntau zam tau zoo, cov kev mob tshwm sim muaj xws li:
Cov teebmeem tshwm sim:
● Mob taub hau
● Dej ntws tawm
● Qhov ntswg congestion
● Dyspepsia (mob plab)
● Mob nraub qaum lossis mob nqaij
Kev txiav txim siab thiab kev ncaj ncees
Cialis yog cov tshuaj noj hauv ntau lub tebchaws, thiab nws txoj kev siv yuav tsum yog nyob rau hauv kev taw qhia ntawm tus kws kho mob. Kev yuav cov ntawv cuav lossis tsis raug cai hauv online ua rau muaj kev pheej hmoo loj rau kev noj qab haus huv.
Kev sib piv nrog Lwm PDE5 Inhibitors
Vs. Viagra (Sildenafil):
Ntev ib nrab-lub neej thiab lub sijhawm ua haujlwm.
Tsawg rhiab heev rau kev noj zaub mov.
Vs. Levitra (Vardenafil):
Cov kev ua tau zoo sib xws tab sis zoo dua yooj yim vim yog ncua sij hawm ntev.
Vs. Stendra (Avanafil):
Kev pib sai dua tab sis lub sijhawm luv dua piv rau Cialis.
Innovation thiab Kev Tshawb Fawb Yav Tom Ntej
Muaj peev xwm siv tshiab:
1. Kev Tshawb Fawb Txog Kab Mob:
● Tshawb xyuas lub luag haujlwm ntawm PDE5 inhibitors hauv kev txhim kho cov tshuaj khomob zoo.
2.Neuroprotection:
● Cov kev tshawb fawb tshiab tshawb nrhiav Cialis qhov muaj peev xwm hauv cov kab mob neurodegenerative.
3. Novel Delivery Systems:
● Kev txhim kho ntawm cov txheej txheem transdermal lossis sublingual rau kev txhim kho bioavailability thiab txo cov kev mob tshwm sim.
Cov ntaub ntawv kho mob
| Hom |
BNP |
|
Cov npe lag luam |
Tadalafil, Cialis, Cidala, Adcirca |
|
CAS |
171596-29-5 |
|
Molar loj |
389.41 |
|
Formula |
C22H19N3O4 |
|
Purity |
Tshaj 98% |
|
Yam khoom |
20 mg x 100 |
Txhua yam kev xav tau, thov hu rau peb
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Xaus
Cialis (Tadalafil) yog cov tshuaj ntau yam uas muaj pov thawj muaj txiaj ntsig rau erectile kawg, benign prostatic hyperplasia, thiab pulmonary arterial hypertension. Nws txuas ntxiv ib nrab-lub neej, kev ua tau zoo dua qub, thiab cov ntaub ntawv muaj kev nyab xeeb zoo ua rau nws muaj txiaj ntsig zoo ntawm PDE5 inhibitors. Txawm li cas los xij, zoo li txhua yam tshuaj, kev siv lub luag haujlwm hauv kev saib xyuas kev kho mob yog qhov tseem ceeb los ua kom nws cov txiaj ntsig zoo tshaj plaws thiab txo qis kev pheej hmoo.
Raws li kev tshawb fawb tsis tu ncua txuas ntxiv nthuav tawm cov peev txheej kho tshiab rau Cialis, nws tseem yog lub hauv paus kev kho mob rau vascular thiab kev sib deev. Txawm hais tias siv rau nws cov lus qhia thawj lossis cov ntawv thov tawm ntawm daim ntawv lo, Cialis muaj kev sib xyaw ua ke ntawm kev ua tau zoo, yooj yim, thiab kev tsim kho tshiab.
Cim npe nrov: bnp cialis(tadanafil) rau kev sib deev cas:171596-29-5, Tuam Tshoj bnp cialis(tadanafil) rau kev sib deev cas:171596-29-5 manufacturers, lwm tus neeg, Hoobkas
