STROMUSC Primobolan (Methenolone Enanthate) 200mg / ml Rau Bodybuilding CAS: 303-42-4
Methenolone enanthate occupies ib tug peculiar txoj hauj lwm nyob rau hauv lub anabolic toj roob hauv pes. Nws tsis yog qhov muaj zog tshaj plaws lossis qhov nrawm tshaj plaws - ua yeeb yam muaj nyob rau hauv, tsis tau nws tau ua raws li kev mob siab rau ntawm cov neeg ncaws pob lub cev rau ntau tshaj li ib nrab xyoo pua. Cov tshuaj txhaj tshuaj, feem ntau lees paub nyob rau hauv lub npe lag luam Primobolan Depot, tau txais lub koob npe nrov li "tus txiv neej lub steroid" - qhov sib xyaw ua ke nrog kev huv, qhuav, muaj txiaj ntsig zoo dua li cov khoom tawg lossis cov dej khaws cia. Qhov 200 mg/ml concentration sawv cev rau cov qauv siv tau ntau dua rau cov neeg siv niaj hnub no, txo cov ntim ntim thaum khaws cia cov khoom sib xyaw ua ke cov yam ntxwv qeeb - tso tshuaj pharmacokinetics. Qhov profile no tshuaj xyuas methenolone enanthate los ntawm kev tsim lub cev, npog nws cov tshuaj lom neeg, cov yam ntxwv ntawm cov tshuaj, kev siv tswv yim, kev xav txog ntau npaum li cas, kev tsim lub voj voog, ib nrab - lub neej, thiab tom qab - cov kev cai kho mob.
Methenolone Enanthate yog dab tsi
Methenolone enanthate yog ib qho hluavtaws anabolic -androgenic steroid muab los ntawm dihydrotestosterone (DHT). Chemically, nws yog tus 17 -enanthate ester ntawm methenolone, tsim los ntawm esterifying niam txiv hormone nrog enanthic acid (heptanoic acid). Qhov sib ntxiv ntawm cov ester no tsis yog qhov nthuav dav me me - nws hloov pauv cov kev coj ua hauv lub cev. Thaum unesterified methenolone yuav raug tshem tawm sai heev, cov enanthate ester ua rau nws muaj lipophilic heev, ua rau nws nqus tau maj mam los ntawm qhov chaw txhaj tshuaj intramuscular mus rau hauv cov hlab ntsha. Thaum circulating, ntshav esterases maj mam cleave ester daim ntawv cog lus, liberating lub active tshuaj hormone methenolone.
Methenolone nws tus kheej yog 1-methyl derivative ntawm DHT. Qhov kev hloov kho ntawm cov qauv no yog qhov tseem ceeb: pawg methyl ntawm C1 txoj hauj lwm confers tsis kam mus rau hepatic metabolism thaum khaws cia cov dej num anabolic. Qhov tseem ceeb, methenolone twb 5 - txo qis, txhais tau tias nws tsis tuaj yeem hloov pauv ntxiv los ntawm 5 -reductase enzyme rau hauv lub zog androgen ntau dua. Qhov no piav qhia ntau ntawm nws tus cwj pwm androgenic me me.
Cov anabolic-rau-androgenic piv ntawm methenolone enanthate feem ntau raug suav hais tias yog 88:44 txog 88:57 thaum piv rau testosterone raws li tus qauv siv 100:100. Hauv cov ntsiab lus siv tau, qhov no txhais tau hais tias qhov sib xyaw ua rau kwv yees li 88% ntawm testosterone's anabolic (cov leeg-tsim) kev ua si thaum pom tsuas yog 44-57% ntawm nws cov haujlwm androgenic (masculinizing). Nws yog ib qho tsim nyog sau cia tias qhov piv txwv no, thaum muaj txiaj ntsig zoo rau kev sib piv cov tebchaw, tsis tuaj yeem ntes tag nrho cov complexity ntawm steroid tus cwj pwm hauv cov kab mob muaj sia. Methenolone enanthate tsis yog aromatizable-nws tsis hloov mus rau estrogen- uas tshem tawm tag nrho cov kev mob tshwm sim estrogenic.


Pharmacological nta thiab qhov zoo
Lub ntsiab pharmacological feature ntawm methenolone enanthate yog nws tsis yog - aromatizing xwm. Vim nws tsis tuaj yeem hloov mus rau estradiol, cov neeg siv tsis paub txog cov dej tuav, gynecomastia txaus ntshai, lossis ntshav - siab siab uas nrog cov tshuaj aromatizing xws li testosterone lossis Dianabol. Cov txiaj ntsig uas tsim tawm yog li "qhuav"- uas yog, lawv muaj feem ntau ntawm cov leeg nqaij contractile es tsis yog cov kua dej subcutaneous. Qhov kev ua tau zoo no ib leeg piav qhia tias vim li cas methenolone tau dhau los ua ib qho tseem ceeb ntawm kev ua ntej - kev sib tw kev sib tw thaum lub sij hawm tsim lub cev kub thiab tseem nrov ntawm cov neeg ncaws pob lub cev niaj hnub no.
Qhov thib ob feature yog nws qhov cuam tshuam androgenic tsawg. Txawm hais tias tsis muaj cov tshuaj anabolic steroid tag nrho tsis muaj cov teebmeem androgenic, methenolone twb tau -5 -txo cov qauv txhais tau tias nws tsis tau ua kom muaj zog ntxiv hauv androgen- cov ntaub so ntswg rhiab heev. Pob txuv, oily ntawm daim tawv nqaij, thiab ceev cov txiv neej- qauv plaub hau poob yog ua tau tab sis feem ntau koob- nyob ntawm thiab tsis muaj suab ntau dua li muaj zog androgens. Qhov no ua rau methenolone enanthate ib qho kev sib piv txaus nyiam rau cov poj niam uas xav siv cov tshuaj anabolic nrog kev txo qis ntawm virilization, txawm tias ceev faj tseem ceeb.
Thib peb, tus enanthate ester muab qhov kev tso tawm ntev ntev. Ib qho kev txhaj tshuaj intramuscular nkaus xwb tswj cov ntshav siab rau kwv yees li ob lub lis piam, txhais tau tias kev txhaj tshuaj tsuas yog siv ib zaug lossis ob zaug hauv ib lub lis piam. Qhov 200 mg / ml concentration txo qhov ntim ntawm cov roj uas yuav tsum tau txhaj rau ib koob, uas yog qhov kev txiav txim siab zoo rau cov neeg siv khiav ntau dua txhua lub lim tiam.
Thaum kawg, methenolone enanthate tsis yog 17 -alkylated. Tsis zoo li qhov ncauj methenolone acetate, uas tau hloov kho kom muaj sia nyob ua ntej- dhau lub siab metabolism thiab yog li ntawd muaj qee qhov muaj peev xwm hepatotoxic, cov tshuaj enanthate hla lub siab ntawm nws thawj zaug thiab suav tias yog qhov tseem ceeb tsis yog -hepatotoxic ntawm cov koob tshuaj tsim nyog.
Kev siv lub cev tsim
Methenolone enanthate feem ntau yog ua hauj lwm thaum lub sij hawm txiav los yog recomposition theem. Nws cov kev sib xyaw ua ke ntawm tsis yog - aromatization, kev ua haujlwm androgenic me me, thiab qab los noj mov- cov teebmeem stimulating ua rau nws zoo- haum rau cov khoom noj uas tsis muaj calorie ntau ntau. Cov neeg siv tau tshaj tawm tias qhov sib xyaw ua ke pab khaws cov nqaij ntshiv nqaij thaum lub sijhawm tsis txaus thaum ua rau muaj qhov hnyav, ntom ntom thaum lub cev muaj roj tsawg. Nws tsis yog ib qho loj- tsim tshuaj nyob rau hauv cov lus pom zoo; cov neeg nrhiav kev loj hlob sai feem ntau saib rau testosterone, nandrolone, lossis oxymetholone. Methenolone qhov kev koom tes yog ib qho zoo dua li qhov ntau.
Vim tias nws tsis aromatize, methenolone enanthate feem ntau stacked nrog cov tshuaj testosterone tsawg los tswj libido, mus ob peb vas, thiab tag nrho cov hormonal tshuav. Kev khiav methenolone ib leeg yuav txwv tsis pub endogenous testosterone ntau lawm, thiab txij li nws tsis muaj kev txhawb nqa estrogenic, cov neeg siv uas txwv lawv cov testosterone yam tsis muaj kev hloov pauv hauv exogenous tuaj yeem ntsib qis - cov tsos mob estrogen xws li kev sib koom ua ke tsis xis nyob, lethargy, thiab txo libido. Cov txheej txheem txoj hauv kev yog li no kom suav nrog tsawg kawg ib qho tshuaj hloov pauv ntawm testosterone hauv ib qho methenolone- muaj lub voj voog.
Methenolone enanthate kuj tseem siv tau los ua "choj" sib xyaw ntawm cov voj voog hnyav dua, txawm tias qhov kev coj ua no yog qhov tsis sib haum xeeb. Nws qhov xwm txheej me me ua rau nws tsis muaj zog ntau dua li ntau lwm txoj hauv kev siv tshuaj tsawg, tab sis ib qho exogenous androgen yuav tawm tswv yim tsis zoo rau ntawm hypothalamic{1}}pituitary-gonadal axis.
Kev txiav txim siab noj tshuaj
Kev noj tshuaj rau methenolone enanthate yog ib qho kev sib cav loj heev. Qhov sib xyaw ua ke yog koob tshuaj -rhiab heev: ntau tus neeg siv qhia tias qis dua qhov pib, cov txiaj ntsig tsis tsim nyog. Rau cov txiv neej, feem ntau hais txog ntau yam pib ntawm kwv yees li 300-400 mg ib lub lis piam rau cov pib tshiab thiab txuas mus rau 600-800 mg ib lub lis piam rau cov neeg siv paub txog. Qee qhov chaw qhia tias 500-700 mg ib lub lis piam sawv cev rau "qhov chaw qab zib" rau cov txiv neej feem ntau cev nqaij daim tawv. Qhov 200 mg / ml concentration yog qhov yooj yim hauv cov ntsiab lus no: 600 mg txhua lub lim tiam yuav tsum tsuas yog 3 ml ntawm cov roj, uas tuaj yeem muab faib ua ob txoj kev txhaj tshuaj ntawm 1.5 ml txhua.
Cov poj niam raug qhia kom siv cov koob tshuaj qis dua. Cov kws kho mob thiab cov tswv yim qhia pom zoo 50-100 mg ib lub lis piam, muab rau hauv ib qho kev txhaj tshuaj lossis faib ua ob koob me me. Qee cov ntaub ntawv soj ntsuam pom zoo kom tsis pub ntau tshaj 50 mg txhua ob mus rau peb lub lis piam rau cov poj niam ntshiv heev. Virilization kev pheej hmoo, thaum txo qis piv rau ntau cov tshuaj androgenic, tsis yog xoom, thiab cov poj niam yuav tsum saib xyuas lub suab hloov, clitoral o, thiab cov plaub hau loj hlob txawv txawv.
Kev txhaj tshuaj ntau zaus rau enanthate ester feem ntau yog ib zaug lossis ob zaug hauv ib lub lis piam. Ob zaug- kev tswj hwm txhua lub lim tiam ua rau cov ntshav ruaj khov dua, uas tuaj yeem txo qhov kev hloov pauv ntawm lub siab thiab lub zog. Cov chaw txhaj tshuaj yuav tsum tau tig los tiv thaiv kev tsim cov caws pliav.
Cycle Design
Ib lub voj voog methenolone enanthate rau cov txiv neej kav ntev li 10-16 lub lis piam. Lub voj voog luv luv ntawm 8-10 lub lis piam qee zaum siv, tab sis vim tias cov enanthate ester siv sijhawm ntau lub lis piam kom mus txog qhov tsis tu ncua - cov ntshav hauv xeev, lub voj voog luv luv yuav tsis tso cai rau tus neeg siv kom paub txog qhov sib xyaw ua ke. Ib qho kev sib koom ua ke yog raws li hauv qab no: lub lis piam 1-12 ntawm 400-600 mg ib lub lim tiam ntawm methenolone enanthate, ua ke nrog kev saib xyuas koob tshuaj testosterone (feem ntau 150-200 mg ib lub lis piam) los khaws cov tshuaj hormonal. Lub voj voog yog ua raws li lub sijhawm tos kom tso cai rau ester kom tshem tawm ua ntej pib tshaj tawm - kev kho lub voj voog.
Thaum lub sij hawm lub voj voog, kev txhawb nqa ntxiv feem ntau yog ncaj nraim. Vim tias methenolone tsis aromatize, aromatase inhibitors feem ntau tsis tsim nyog. Lipid kev txhawb nqa-xws li omega-3 fatty acids thiab citrus bergamot-yog qhov pom zoo, vim tias anabolic steroids tuaj yeem cuam tshuam rau cov roj cholesterol profile. Kev tawm dag zog lub plawv thiab kev saib xyuas ntshav siab tsis tu ncua yog cov kev coj ua zoo rau txhua lub voj voog.
Ib nrab-Lub Neej thiab Pharmacokinetics
Kev tshem tawm ib nrab - lub neej ntawm methenolone enanthate tom qab txhaj tshuaj intramuscular yog kwv yees li 10.5 hnub. Qhov ntev ib nrab - lub neej no yog qhov tshwm sim ncaj qha ntawm cov enanthate ester, uas ua rau qeeb qhov tso tawm ntawm cov tshuaj hormones los ntawm kev txhaj tshuaj depot. Peak plasma concentrations feem ntau mus txog ob peb hnub tom qab kev tswj hwm, tom qab ntawd maj mam poob. Lub neej nquag ntawm ib qho kev txhaj tshuaj feem ntau raug suav hais tias yog 10-14 hnub.
Qhov ntev ib nrab-lub neej muaj ob qhov cuam tshuam. Ua ntej, kev txhaj tshuaj tsuas yog siv ib zaug lossis ob zaug hauv ib lub lis piam. Qhov thib ob, tom qab kev txhaj tshuaj zaum kawg, qhov sib xyaw tseem nyob hauv qhov system rau lub sijhawm tseem ceeb. Qhov no yog vim li cas lub sijhawm tos ntawm kwv yees li 14-18 hnub tau pom zoo ua ntej pib tom qab- kev kho lub voj voog. Pib PCT ntxov dhau lawm, thaum methenolone tseem ua rau cov hypothalamic-pituitary-gonadal axis, yuav yog qhov tsis zoo.
Methenolone feem ntau metabolized hauv daim siab, nrog rau cov zis metabolite yog 3 -hydroxy-1-methylene-5 -androstan-17-one. Sulfated metabolites tuaj yeem kuaj pom hauv cov zis rau lub sijhawm txuas ntxiv, nrog qee cov cim tseem ceeb tuaj yeem kuaj tau ntev txog 17 hnub thiab lwm tus muaj peev xwm ntev dua.
Ncej -Cycle Therapy
Tom qab-kev kho lub voj voog (PCT) yog qhov yuav tsum tau ua tom qab muaj kev cuam tshuam anabolic steroid voj voog, thiab methenolone enanthate tsis muaj qhov zam. Txawm hais tias nws lub koob npe nrov li "mob", nws suppresses endogenous testosterone ntau lawm, tshwj xeeb tshaj yog nyob rau hauv cov koob tshuaj siv nyob rau hauv bodybuilding ntsiab lus. PCT lub hom phiaj los kho cov hypothalamic -pituitary-gonadal axis kom ua haujlwm zoo li sai thiab nyab xeeb li sai tau.
Tus txheej txheem PCT raws tu qauv tom qab lub voj voog methenolone enanthate suav nrog kev xaiv tshuaj estrogen receptor modulator (SERM). Nolvadex (tamoxifen citrate) feem ntau yog siv ntawm 20 mg ib hnub twg rau plaub lub lis piam, qee zaum nrog lub tswv yim tapering ntawm 20/20/10/10 mg tshaj plaub lub lis piam. Clomid (clomiphene citrate) yog lwm qhov kev xaiv, feem ntau noj ntawm 50 mg txhua hnub rau plaub lub lis piam. Qee cov kws kho mob nyiam enclomiphene, lub hom phiaj ntau dua ntawm clomiphene, ntawm 25 mg ib hnub rau ob lub lis piam tom qab 12.5 mg ib hnub rau plaub lub lis piam thiab tom qab ntawd 12.5 mg txhua hnub rau ib lub lis piam.
Lub sijhawm ntawm PCT pib yog qhov tseem ceeb. Vim hais tias methenolone enanthate muaj ib nrab -lub neej ntawm kwv yees li 10.5 hnub, nws yuav siv sij hawm kwv yees li tsib ib nrab -lub neej-txog 50 hnub-rau cov compound yuav luag tag nrho tshem tawm ntawm lub system. Txawm li cas los xij, feem ntau cov txheej txheem siv tau pib PCT kwv yees li 14-18 hnub tom qab kev txhaj tshuaj zaum kawg, thaum cov qib circulating tau poob qis txaus kom tso cai rau SERM los txhawb kev tso tawm gonadotropin yam tsis tau cuam tshuam los ntawm kev tawm tsam androgen.
Thaum PCT, cov neeg siv yuav tsum saib xyuas cov cim qhia ntawm testosterone qis: qaug zog, tsis muaj libido, kev puas siab puas ntsws, thiab mob pob qij txha. Cov ntshav ua haujlwm- suav nrog tag nrho cov testosterone, luteinizing hormone, follicle-stimulating hormone, thiab estradiol- tuaj yeem muab lub hom phiaj kev pom zoo ntawm kev rov zoo. Kev kho kom rov zoo tag nrho yuav siv li ob peb lub lis piam mus rau ob peb lub hlis, nyob ntawm tus neeg thiab lub sijhawm ntawm lub voj voog ua ntej.
Cov ntaub ntawv kho mob
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Hom |
STROMUSC |
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Cov npe lag luam |
Metenolone enanthate, Nibal Txhaj Tshuaj, Primobolan Depot Metenolone 17 -enanthate; NSC-64967; SH-601; SQ-16374; |
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CAS |
303-42-4 |
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Molar loj |
414.630 |
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Formula |
C27H42O3 |
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Purity |
Tshaj 98% |
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Peev Xwm / Lub raj mis |
200 mg/ml |
Txhua yam kev xav tau, thov hu rau peb
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Xaus
Methenolone enanthate 200 mg / ml yog qhov sib xyaw ua ke uas muab nqi zog rau kev ua siab ntev thiab kev ua haujlwm siab. Nws yuav tsis xa cov txiaj ntsig loj heev ntawm testosterone lossis nandrolone, tab sis nws muaj qee yam muaj txiaj ntsig zoo rau lub cev - tsom mus rau kis las: zoo. Cov txiaj ntsig yog lean, sab - cuam tshuam profile yog qhov zoo sib xws, thiab qhov tsis yog - aromatizing xwm simplifies lub voj voog kev tswj hwm ntau. Nws ntev ib nrab-lub neej ua rau ob zaug- noj tshuaj txhua lub lim tiam, thiab nws tus cwj pwm androgenic me me ua rau nws yog ib qho ntawm ob peb cov tshuaj anabolic steroids uas tuaj yeem txiav txim siab rau poj niam siv nrog kev ceev faj kom tsim nyog. Tsis muaj qhov no txhais tau hais tias lub compound tsis muaj teeb meem. Kev tawm tsam ntawm kev tsim cov tshuaj testosterone ntuj yog tiag tiag, cov teebmeem ntawm cov hlab plawv thiab lipid yuav tsum tau saib xyuas, thiab cov khoom sib xyaw tseem yog cov tshuaj tswj hwm hauv feem ntau cov cai. Siv lub luag haujlwm, txawm li cas los xij, methenolone enanthate tseem yog cov cuab yeej tshwj xeeb thiab muaj txiaj ntsig nyob rau hauv lub cev tsim tshuaj tshuaj repertoire.
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