Siab -Quality STROMUSC MENT (Trestolone Acetate) 50mg/ml Rau Bodybuilding CAS: 6157-87-5
Trestolone Acetate, paub sib tham nyob rau hauv bodybuilding lub voj voog raws li MENT, sawv cev rau ib qho ntawm cov muaj zog tshaj hluavtaws anabolic -androgenic steroids puas tau tsim. Lub ntsiab lus ntawm MENT yog muab los ntawm nws cov tshuaj nomenclature-7 -Methyl-19-Nortestosterone-qhov twg "M" txhais tau hais tias pawg methyl ntawm 7 txoj hauj lwm, "E" hais txog estrane puag qauv, "N" qhia tias tsis muaj 19th carbon (tsis yog nws qhov kev teeb tsa). Ua ntej synthesized nyob rau hauv 1963, lub compound tseem tsis nco qab lawm ntau xyoo mus txog rau thaum cov paj paj resurrive nws rau tej kev siv kho mob.
Lub Compound's Identity thiab Keeb Kwm
Trestolone Acetate, paub sib tham nyob rau hauv bodybuilding lub voj voog raws li MENT, sawv cev rau ib qho ntawm cov muaj zog tshaj hluavtaws anabolic -androgenic steroids puas tau tsim. Lub ntsiab lus MENT yog muab los ntawm nws cov tshuaj nomenclature -7 -Methyl-19-Nortestosterone- qhov twg "M" qhia txog pawg methyl ntawm 7 txoj hauj lwm, "E" hais txog cov qauv estrane, "N" qhia qhov tsis muaj 19 carbon (tsis yog kev teeb tsa), thiab "T" qhia txog nws cov testosterone- rov qab los. Ua ntej synthesized nyob rau hauv 1963, lub compound tseem tsis nco qab lawm ntau xyoo mus txog rau thaum cov paj paj resurrive nws rau tej kev siv kho mob.
Chemically xaiv raws li 7 -methylestr-4-en-17 -ol-3-ib 17 -acetate, Trestolone Acetate yog 19-tsis yog derivative uas muaj nyob rau tib tsev neeg steroid li Nandrolone thiab Trenbolone. Txawm li cas los xij, nws muaj qhov sib txawv tseem ceeb uas ua rau nws sib nrug ntawm lwm tus 19-tsis yog: 7 - pawg methyl tiv thaiv 5 - txo qis thaum ib txhij txhim kho androgen receptor binding affinity. Qhov kev hloov kho cov qauv no yog lub hauv paus ntawm nws qhov muaj zog tshaj plaws.
Raws li ib tug prodrug, Trestolone Acetate undergoes sai hydrolysis tom qab kev tswj hwm, hloov mus rau lub active compound Trestolone (MENT). Cov acetate ester txuas ntawm C17 txoj haujlwm hloov kho nws cov tshuaj pharmacokinetics, muab kev tswj kev tso tawm thiab txhim kho bioavailability tom qab txhaj tshuaj intramuscular. Qhov 50mg / mL concentration yog qhov feem ntau ntsib kev npaj hauv qhov tsis yog -kev kho mob, feem ntau nthuav tawm hauv 10mL multidose vials.


Pharmacological nta thiab Mechanism of Action
Androgen Receptor Affinity
Pharmacological profile ntawm MENT tsis muaj dab tsi luv luv ntawm qhov zoo tshaj plaws. Nws cov androgen receptor binding affinity tau tshaj tawm tias muaj kwv yees li 2.6 npaug ntawm 5 -dihydrotestosterone (DHT), nrog rau cov khoom siv hluav taws xob uas txuas ntxiv rau nws cov teebmeem. Lub 7 -methylation ua hauj lwm rau ntau lub hom phiaj: nws nce androgen receptor affinity, cuam tshuam metabolic inactivation los ntawm kev txo qis ntawm delta -4 daim ntawv cog lus, thiab txo affinity rau kev sib deev hormone-binding globulin (SHBG). Qhov no txhais tau hais tias ib qho kev faib ua feem ntau ntawm cov compound tseem tsis pub dawb thiab ua haujlwm lom neeg hauv kev ncig.
Lub Aromatization Paradox
Tej zaum qhov tshwj xeeb tshaj plaws ntawm MENT yog nws txoj kev sib raug zoo nrog estrogen. Tsis zoo li lwm yam 19-tsis muaj cov tshuaj xws li Nandrolone thiab Trenbolone, uas tsis aromatize ntau, MENT hloov mus rau 7 -methylestradiol- muaj zog estrogenic metabolite. Cov cuab yeej no ua rau MENT ib qho kev sib xyaw ua ke: nws muab Trenbolone zoo li androgenic zog thaum ib txhij muab nws tus kheej estrogenic teeb liab. Cov yam ntxwv no tau coj qee cov neeg siv qib siab los ua haujlwm MENT ua ib qho chaw nyob ib leeg yam tsis muaj testosterone puag, vim nws tuaj yeem ua raws li qhov xav tau ntawm androgenic thiab estrogenic rau kev ua haujlwm ntawm lub cev.
Progestogenic Activity
Raws li 19-tsis yog derivative, MENT nthuav tawm cov haujlwm progestogenic, ua tus agonist ntawm progesterone receptor nrog khi affinity piv rau progesterone nws tus kheej. Qhov no progestogenic tivthaiv, ua ke nrog nws cov estrogenic metabolite, tsim ib tug complex hormonal milieu uas yuav tsum tau ceev faj tswj.
Tsis-5-Alpha txo qhov xwm txheej
MENT tsis cuam tshuam nrog 5-alpha reductase enzyme thiab yog li tsis tuaj yeem hloov mus rau dihydrotestosterone (DHT). Nws cov teebmeem androgenic yog tag nrho ncaj qha, kho los ntawm androgen receptor nws tus kheej. Qhov no txhais tau hais tias DHT-txog cov kev mob tshwm sim xws li prostate o thiab txiv neej qauv baldness tshwm sim los ntawm ib tug sib txawv mechanism tshaj nrog cov tebchaw uas hloov mus rau DHT.
Cov kev siv hauv Bodybuilding
Cov leeg nqaij hypertrophy thiab muaj zog
Hauv cov ntsiab lus ntawm kev tsim lub cev, MENT tau txais lub koob npe nrov rau kev tsim cov khoom lag luam nrawm thiab tseem ceeb hauv cov leeg nqaij thiab lub zog. Cov ntaub ntawv tshawb fawb qhia tias nws lub zog anabolic tuaj yeem nce mus txog kaum npaug ntau dua li testosterone. Lub compound tsim ib qho chaw anabolic heev los ntawm kev sib txuas ntawm cov protein ntau thiab txhim kho nitrogen tuav hauv cov leeg nqaij.
Cov txiaj ntsig tau tsim los ntawm MENT feem ntau tau piav qhia tias "ntub" vim yog cov dej estrogenic khaws cia, ua rau cov nqaij ntshiv loj thiab loj. Cov neeg siv tshaj tawm cov twj tso kua mis hnyav thaum lub sijhawm kev cob qhia thiab kev hloov pauv sai sai uas tuaj yeem pom hauv thawj lub lis piam ntawm kev tswj hwm.
Qhov "Tag nrho-hauv-Ib" Phenomenon
MENT lub peev xwm los muab ob qho tib si nws tus kheej androgenic -anabolic teeb liab thiab nws tus kheej estrogen tau ua rau nws siv los ua qhov muaj peev xwm hloov pauv rau testosterone. Cov kev tshawb fawb soj ntsuam tau tshawb xyuas MENT li txiv neej cov tshuaj tiv thaiv kab mob thiab ua lwm txoj hauv kev kho testosterone hloov. Nyob rau hauv lub bodybuilding sphere, qhov no tau txhais mus rau hauv lub voj voog uas MENT yog khiav solo los yog thawj tus neeg sawv cev anabolic yam tsis muaj ib txwm siv testosterone puag-ib qho kev coj ua uas tseem muaj teeb meem tab sis nce ntau ntawm cov neeg siv qib siab.
Kev txiav txim siab stacking
MENT feem ntau muab tso rau hauv pawg nrog rau lwm cov tebchaw. Kev sib koom ua ke muaj xws li testosterone (thaum txo koob tshuaj), Nandrolone, thiab ntau qhov ncauj. Qee cov neeg siv MENT ua tus neeg saib xyuas "kev pub dawb" es tsis yog thawj tus neeg tsav tsheb hypertrophic, siv nws los txhawb cov teebmeem ntawm lwm cov tebchaw. Qhov sib xyaw ua ke txhais tau hais tias nws tuaj yeem hloov kho rau ntau yam kev sib koom ua ke nyob ntawm tus kheej lub hom phiaj thiab kev ua siab ntev.
Cov txiaj ntsig: Dab tsi Cov Neeg Siv Qhia
Rapid Mass Acretion
Qhov feem ntau hais txog qhov txiaj ntsig ntawm MENT yog qhov nrawm nrawm ntawm cov txiaj ntsig. Cov neeg siv tsis tu ncua qhia txog kev nce qib hauv qhov loj thiab lub zog uas tshwm sim sai dua nrog rau feem ntau lwm cov tebchaw. Cov lus teb ceev ceev no ua rau MENT txaus nyiam rau luv luv los yog rau kev tawg ntawm stagnation theem.
Sense of Well{0}}Ua thiab Libido
Tsis zoo li Trenbolone- uas yog qhov tsis zoo rau kev ua rau muaj kev ntxhov siab, ntxhov siab, thiab pw tsaug zog cuam tshuam -MENT feem ntau cuam tshuam nrog kev nkag siab zoo- ua, kev ntseeg siab, thiab nce libido. Kev sib xyaw ua ke ntawm lub zog androgen receptor activation thiab txaus estrogenic kev ua haujlwm zoo li tsim kom muaj lub siab zoo rau ntau tus neeg siv.
Kev Noj Qab Haus Huv
Cov tshuaj estrogenic metabolite 7 -methylestradiol tuaj yeem pab txhawb kev noj qab haus huv los ntawm nws cov teebmeem ntawm collagen synthesis thiab synovial kua. Qhov no yog qhov sib piv rau cov uas tsis yog - aromatizing compounds uas tuaj yeem ua rau kev sib koom ua ke tsis zoo vim yog qhov tsis muaj tshuaj estrogen.
Lipid Profile
Qee cov ntawv ceeb toom qhia tias MENT muaj qhov cuam tshuam zoo rau lipid profile piv rau lwm cov androgens muaj zog. Txawm li cas los xij, qhov no yuav tsum tau txhais nrog ceev faj, vim tias cov lus teb ntawm tus kheej sib txawv heev, thiab qhov sib xyaw ua ke ntawm cov tshuaj estrogenic tuaj yeem cuam tshuam lipoprotein metabolism hauv txoj hauv kev nyuaj.
Cov lus qhia noj tshuaj
Beginner Range
Rau thawj - cov neeg siv sijhawm, kev siv tshuaj tiv thaiv tau qhia zoo. Ib qho pib pib yog 25mg muab txhua hnub (ED). Qhov no tso cai rau tus neeg siv los ntsuas tus kheej kam rau ua thiab ntsuas qhov sib xyaw ua ke ua ntej txiav txim siab ntau npaum li cas. Qee qhov chaw pom zoo kom pib qis dua, ntawm kwv yees li 10-20mg muab txhua ob mus rau peb hnub.
Nruab Nrab
Tus qauv zoo npaum li cas rau cov neeg siv feem ntau poob ntawm 25-75mg txhua hnub (ED) lossis txhua hnub (EOD), tag nrho 175-525mg ib lub lis piam. Rau ntau tus neeg, 25-50mg ED ua pov thawj ntau tshaj qhov txaus kom ua tiav cov txiaj ntsig zoo. Qhov 50mg / mL concentration ua rau kev siv ntau npaum li cas ncaj nraim: 0.5mL txog 1.0mL rau ib qho tshuaj nyob ntawm cov tshuaj xaiv.
Advanced Range
Cov neeg siv kev paub dhau los tuaj yeem thawb ntau npaum li cas mus rau 100mg txhua hnub, txawm hais tias qhov no feem ntau tsis pom zoo rau cov tsis paub nrog qhov sib xyaw. Tag nrho cov koob tshuaj txhua lub lim tiam hauv 350-700mg ntau tau ntsib ntawm cov neeg siv siab heev, txawm hais tias kev tswj cov kev mob tshwm sim dhau los ua qhov nyuaj ntawm cov qib no.
Kev tswj hwm zaus
Vim yog cov acetate ester luv luv ib nrab- lub neej, kev tswj hwm nquag yog tsim nyog los tswj cov ntshav plasma kom ruaj khov. Kev txhaj tshuaj txhua hnub (ED) yog cov txheej txheem ntau tshaj plaws, txawm tias qee cov neeg siv xaiv rau txhua -lwm-hnub (EOD) kev tswj hwm. EOD koob tshuaj ntawm 50mg tau tshaj tawm, tab sis qhov no yuav ua rau muaj kev hloov pauv ntawm hormonal ntau dua.
Cycle Design thiab Duration
Lub voj voog ntev
Hom MENT cycles li ntawm 4 mus rau 12 lub lis piam. Lub voj voog luv luv ntawm 4-6 lub lis piam feem ntau pom zoo rau cov neeg siv thawj zaug lossis cov neeg nrhiav kom txo qis cov kev mob tshwm sim. Longer cycles of 8-12 weeks are employed by more experienced users aiming for maximum tissue accretion.
First Cycle Protocol
Ib txoj hauv kev ua kom zoo rau thawj lub voj voog MENT suav nrog pib nrog 25mg txhua hnub rau thawj ob lub lis piam, tom qab ntawd maj mam nce mus rau 50mg txhua hnub yog tias cov kev mob tshwm sim tseem tswj tau. Lub voj voog yuav tsum tsis pub tshaj 4-6 lub lis piam rau kev pib ua haujlwm.
Stacked Cycle Piv txwv
Rau cov neeg koom nrog MENT rau hauv ib pawg, cov txheej txheem hais txog feem ntau suav nrog kev khiav 25mg / hnub lossis 50mg EOD ntawm MENT rau 3-4 lub lis piam, tom qab ntawd cov tshuaj ntxiv xws li Nandrolone Phenylpropionate (NPP) ntawm 25mg / hnub lossis 50mg EOD tuaj yeem qhia. Lub sijhawm tag nrho lub voj voog feem ntau txuas mus rau 8-10 lub lis piam hauv cov xwm txheej zoo li no.
Ntawm -Cycle Support
Muab rau MENT's estrogenic thiab progestogenic kev ua haujlwm, ntawm -cov tshuaj tiv thaiv kab mob yog qhov tseem ceeb. Aromatase inhibitors xws li Anastrozole lossis Exemestane feem ntau ua haujlwm los tswj cov tshuaj estrogenic. Kev tswj hwm prolactin nrog cov tshuaj xws li Cabergoline lossis Pramipexole kuj tseem yuav tsim nyog vim MENT txoj kev nyiam ua kom cov ntshav prolactin nce. Kev soj ntsuam ntshav siab yog qhov tseem ceeb, vim tias MENT tuaj yeem ua rau muaj kev nce siab hauv systolic ntshav siab.
Ib nrab-Lub Neej thiab Pharmacokinetics
Cov tshuaj Acetate Ester
Cov acetate ester txuas rau trestolone molecule dictates nws cov pharmacokinetic profile. Acetate esters yog luv luv -chain esters uas ua rau kom nqus tau sai, siab tshaj ntshav plasma, thiab kev tshem tawm sai heev. Qhov no yog qhov sib piv rau cov esters ntev dua xws li enanthate lossis cypionate, uas muab cov ntaub ntawv tso tawm ntau dua.
Ib nrab-Kev kwv yees lub neej
Ib nrab -Lub neej ntawm Trestolone Acetate tau raug kev sib cav ntau hauv zej zog tsim lub cev. Qee qhov chaw qhia tias ib nrab luv luv heev -lub neej ntsuas hauv feeb, thaum cov chaw kho mob qhia txog qhov ntev dua ntawm 1-2 hnub. Qhov tsis sib xws yuav qhia txog qhov sib txawv ntawm qhov sib xyaw ua ke ntawm lub cev ib nrab-lub neej thiab lub sijhawm ua haujlwm ntawm kev ua haujlwm tom qab kev tswj hwm intramuscular.
Cov acetate ester muab ib nrab - lub neej uas tsim nyog txhua hnub lossis txhua -lwm- hnub tswj hwm kom tswj cov ntshav kom ruaj khov. Qhov kev tshem tawm sai sai no yog qhov txiaj ntsig zoo rau cov neeg siv uas muaj kev cuam tshuam tsis zoo, vim tias kev txiav tawm tso cai rau qhov sib xyaw kom tshem tawm qhov system nrawm.
Kev kuaj pom thiab tshem tawm
Ib nrab luv luv -lub neej txhais tau hais tias MENT raug tshem tawm ntawm lub cev sai dua li ntev dua - estered compounds. Thaum qhov no pab txhawb kev rov qab sai ntawm cov tshuaj hormones endogenous tom qab kev tso tseg, nws kuj txhais tau hais tias kev tswj hwm zoo ib yam yuav tsum tau tswj xyuas cov teebmeem anabolic. Ua kom tiav kev tshem tawm ntawm lub cev feem ntau tshwm sim nyob rau hauv ob peb hnub ntawm kev txhaj tshuaj zaum kawg, txawm hais tias cov tshuaj tiv thaiv metabolite yuav ntev dua.
Ncej -Cycle Therapy (PCT)
Kev Sib Tw Sib Tw
MENT yog ib qho kev tawm tsam loj heev, muaj peev xwm ua kom nrawm thiab ua tiav kev kaw ntawm hypothalamic{0}}pituitary-gonadal (HPG) axis. Nws lub zog suppressive yog piv rau kev sib xyaw ntawm testosterone thiab etonogestrel. Qhov kev tawm tsam no yog kho los ntawm ntau lub tswv yim: estrogens tawm tswv yim tsis zoo ntawm pituitary, androgens thiab estrogens qeeb hypothalamic GnRH secretion, thiab cov khoom sib xyaw ua haujlwm progestogenic ntxiv dag zog rau cov teeb liab suppressive.
PCT Initiation
Muab MENT ib nrab luv luv -lub neej, PCT yuav tsum pib sai sai tom qab kev tswj hwm zaum kawg. Rau acetate ester, lub sijhawm tos ntawm 3-7 hnub tom qab txhaj tshuaj kawg yog qhov ua ntej pib PCT. Qhov no tso cai rau lub sij hawm txaus rau lub exogenous compound kom meej thiab rau endogenous suppression yuav tsum tau hais.
Standard PCT raws tu qauv
Ib txoj hauv kev zoo PCT rau MENT suav nrog kev siv cov tshuaj estrogen receptor modulators (SERMs) los txhawb kev tsim cov tshuaj endogenous testosterone. Cov txheej txheem raug suav hais tias feem ntau suav nrog Tamoxifen ntawm 20mg txhua hnub rau ob lub lis piam, ua raws li 10mg txhua hnub rau ob lub lis piam ntxiv. Qee cov neeg siv koom nrog tib neeg chorionic gonadotropin (hCG) thaum lub sijhawm kawg ntawm lub voj voog lossis lub sijhawm hloov pauv ua ntej SERM txoj kev kho kom txhawb nqa Leydig cell function.
Extended Recovery Considerations
Qhov kev tawm tsam loj heev tshwm sim los ntawm MENT txhais tau hais tias kev rov qab los ntawm kev tsim cov tshuaj testosterone ntuj yuav nyuaj dua li cov tshuaj tiv thaiv tsawg dua. Qee cov neeg siv tau tshaj tawm tsis tu ncua txawm tias tom qab tus qauv PCT raws tu qauv. Qhov no tau ua rau qee tus tub ceev xwm pom zoo kom ncua sijhawm PCT lossis siv cov txheej txheem nruj dua uas suav nrog ntau yam SERMs lossis kev kho ua ke.
Kev soj ntsuam thiab kev hloov kho
Muab qhov sib txawv ntawm tus kheej cov lus teb, cov ntshav ua haujlwm yog qhov tseem ceeb rau kev coj PCT. Kev soj ntsuam tag nrho cov testosterone, dawb testosterone, LH, FSH, thiab estradiol qib tso cai rau kev soj ntsuam lub hom phiaj ntawm kev rov qab los thiab kev hloov kho ntawm PCT raws tu qauv.
Kev xav txog kev pheej hmoo
Cov teebmeem Estrogenic
MENT qhov kev hloov pauv mus rau 7 -methylestradiol tsim muaj peev xwm loj rau cov kev mob tshwm sim estrogenic xws li gynecomastia, dej tuav, thiab ntshav siab. Cov tshuaj estrogenic metabolite tau tshaj tawm tias muaj zog, thiab qee cov neeg siv piav qhia MENT li tsim cov tshuaj estrogen ntau dua li lwm yam steroid.
Prolactin{0}}Cov teeb meem ntsig txog
Kev ua haujlwm progestogenic ua ke nrog kev nce qib ntawm prolactin tuaj yeem ua rau prolactin -induced gynecomastia thiab kev sib deev tsis zoo. Qhov no "ob chav whammy" ntawm estrogen thiab prolactin yuav tsum muaj kev tswj hwm cov tswv yim.
Cov ntaub ntawv kho mob
| Hom | STROMUSC |
|
Cov npe lag luam |
Orgasteron acetate; MENT acetate; CDB-903; NSC-69948; U-15614; 7 -Methyl-19-nortestosterone 17 -acetate; 7 -Methylestr-4-en-17 -ol-3-one 17 -acetate |
|
CAS |
6157-87-5 |
|
Molar loj |
330.468 |
|
Formula |
C21H30O3 |
|
Purity |
Tshaj 98% |
|
Yam khoom |
50 mg/ml |
Txhua yam kev xav tau, thov hu rau peb
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Xaus
Trestolone Acetate (MENT) ntawm 50mg / mL sawv cev rau ib qho ntawm cov muaj zog tshaj plaws anabolic agents muaj nyob rau hauv tsis yog-sphere soj ntsuam. Nws qhov tshwj xeeb pharmacological profile- sib txuas cov tshuaj androgen receptor affinity, aromatization rau lub zog estrogen, thiab progestogenic kev ua si-tsim ib tug compound ntawm extraordinary hwj chim thiab complexity. Kev nce nrawm hauv cov leeg nqaij thiab lub zog yog sib npaug los ntawm cov kev sib tw tseem ceeb hauv kev tswj cov kev mob tshwm sim thiab tom qab- rov qab mus.
Lub tebchaw keeb kwm raws li ib tug txiv neej muaj peev xwm tiv thaiv kab mob thiab TRT lwm txoj hauv kev qhia txog nws cov teebmeem muaj zog ntawm HPG axis. Tib yam khoom no uas ua rau nws siv tau rau kev tiv thaiv kab mob ua rau nws yog ib qho nyuaj tshaj plaws rau kev xa rov qab - voj voog rov qab. Cov acetate ester luv luv muab qhov zoo ntawm kev tshem tawm sai sai yuav tsum muaj kev cuam tshuam tsis zoo tshwm sim, tab sis kuj xav tau cov txheej txheem kev tswj hwm.
Rau cov neeg uas xaiv los ua haujlwm MENT, kev npaj txhij txhua- suav nrog kev nthuav dav ntawm - kev txhawb nqa lub voj voog, kev ntsuas ntshav siab, thiab lub qhov dej -tsim PCT raws tu qauv- tsis yog xaiv tab sis tseem ceeb. Lub zog lub zog xav tau kev hwm, thiab nws cov kev pheej hmoo yuav tsum tau tswj xyuas kom zoo. Raws li nrog tag nrho cov muaj zog anabolic agents, qhov kev txiav txim siab siv MENT yuav tsum tau ua nrog tag nrho cov kev paub txog ob qho tib si nws muaj peev xwm zoo kawg thiab nws cov peev xwm tseem ceeb rau kev puas tsuaj.
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