
FIERCE Letrozole (Femara) 2.5mg Bodybuilding CAS: 112809-51-5
Letrozole (Femara) thiab Arimidex yog ob qhov nrov tshaj plaws aromatase inhibitors ntawm 3 loj AIs, nrog Letrozole yog qhov thib ob nrov tshaj plaws. Letrozole tau pom qee qhov ua tau zoo kawg nkaus hauv kev txo cov tshuaj Estrogen, ntau dua li ob qhov loj aromatase inhibitors. Hauv kev sib piv nrog Arimidex, Letrozole tau pom tias yog 10 - 20 npaug ntawm lub zog ntawm Arimidex, thiab txawm hais tias Letrozole koob tshuaj muaj txiaj ntsig zoo ib yam li Aromasin, nws ua haujlwm los ntawm txoj kev sib txawv kom ua tau zoo ntawm nws tus kheej txoj cai[1 ]. Txawm li cas los xij, cov ntsiab lus hais tias anabolic steroid siv cov neeg ncaws pob lossis tus kws tsim lub cev sib txawv me ntsis los ntawm kev kho mob thiab kev kho mob daim ntawv thov ntawm Letrozole lossis ib qho aromatase inhibitor, thiab qhov no yog dab tsi cov neeg siv tshuaj anabolic steroid feem ntau txhawj xeeb nrog: cov koob tshuaj Letrozole kom zoo rau kev tswj Estrogen, yuav ua li cas. Txhawm rau siv cov koob tshuaj Letrozole, thiab cov cwj pwm sib txawv uas cov koob tshuaj Letrozole tuaj yeem siv tau.
yog dab tsiLetrozole?
Nws yuav tsum xub to taub tias Letrozole yog ib qho aromatase inhibitor, nrog rau ntau yam kev siv nyob rau hauv cov nqe lus ntawm Estrogen tswj. Raws li aromatase inhibitor, nws tuav lub peev xwm los tswj hwm qhov tseeb ntawm txhua qhov muaj peev xwm Estrogenic phiv uas cov neeg siv tshuaj anabolic steroid sim zam lossis tshem tawm. Tus txheej txheem raws tu qauv (los yog txoj cai dav dav) rau kev sivtag nrhoaromatase inhibitors yuav tsum yog cov hauv qab no:
Sim zam kev siv cov aromatase inhibitors ntawm txhua tus nqi tshwj tsis yog tias tsim nyog. Yog tias kev siv cov aromatase inhibitor yog qhov tsim nyog, siv nws tsuas yog thaum xav tau, thiab sim ua kom qis tshaj qhov ua tau zoo rau lub hom phiaj ntawm kev tswj hwm Estrogen es tsis yog kev tshem tawm cov tshuaj estrogen.
Qhov no yog qhov tseem ceeb heev thiab yuav tsum nco ntsoov los ntawm txhua tus neeg nyeem tshawb xyuas kev siv aromatase inhibitors. Qhov tseeb ntawm qhov teeb meem yog tias kev siv aromatase inhibitors, txawm tias nws yog peb lub hauv paus AIs (Arimidex, Aromasin, thiab Letrozole) lossis lwm yam, yuav ua rau muaj kev cuam tshuam tsis zoo rau lub cev yog siv thaum lawv tsis xav tau, lossis thaum lawv siv. Kev siv ntau dhau ntawm Letrozole koob tshuaj uas siab dhau lawm.
Nco ntsoov tias yog vim li cas rau kev siv cov aromatase inhibitor yuav tsum nyob rau txhua lub sijhawm yog rau lub hom phiaj ntawm Estrgentswjtsis yog Estrogentshem tawm, raws li qhov ua tiav thiab tag nrho txo qis ntawm tag nrho cov qib Estrogen hauv lub cev tuaj yeem ua rau muaj kev cuam tshuam rau tib neeg lub cev. Qhov no yuav piav qhia ntxiv nyob rau hauv cov kev mob tshwm sim ntawm qhov profile no, tab sis cov lus piav qhia dav dav yog tias cov tshuaj no (aromatase inhibitors) ua rau lub cev tsis zoo ntawm cov tshuaj hormones tseem ceeb (Estrogen) uas yog qhov tseem ceeb rau ntau yam tseem ceeb ntawm lub cev ua haujlwm ntawm lub cev ib txwm muaj.


Kev kho mob Letrozole Dosage
Letro tau pom zoo los ntawm FDA rau kev kho mob ntawm cov poj niam cev xeeb tub tom qab yug me nyuam cov neeg mob qog noj ntshav raws li kev kho mob ntxiv thaum cov kev kho thawj kab (xws li Nolvadex) ua tsis tiav. Nws kuj tau pom zoo rau kev kho mob txuas ntxiv rau cov poj niam cev xeeb tub tom qab mob qog noj ntshav tom qab 5 xyoos ntawm Nolvadex tswj hwm. Letrozole kuj tau txais kev pom zoo rau kev kho mob ntawm cov poj niam tom qab yug me nyuam cov poj niam mob qog noj ntshav uas muaj cov tsos mob ntawm Estrogen receptor tsis paub txog mob qog noj ntshav. Qhov no yog ib qho mob qog noj ntshav hauv lub mis uas qhov kev kuaj mob qhia tias nws tsis paub tias Estrogen yog tus neeg ua txhaum, lossis puas yog mob qog noj ntshav mis hnyav dua los ntawm Estrogen. Thaum kawg, nws kuj tau txais kev pom zoo rau kev kho mob ntawm cov poj niam cev xeeb tub tom qab mob qog noj ntshav mis rau cov neeg mob uas tag nrho lwm cov tshuaj tiv thaiv Estrogen tsis tau ua haujlwm (qhov no suav nrog SERMs thiab tag nrho lwm yam AIs). Letrozole feem ntau yog qhov chaw zaum kawg thiab kev kho mob zaum kawg rau cov neeg mob qog noj ntshav thaum txhua yam ua tsis tiav.
Cov koob tshuaj Letrozole rau kev kho mob qog noj ntshav hauv txhua kis yog 2.5mg ib hnub.
Letrozole Dosage Thaum siv Anabolic Steroid
Letrozole tshwj xeeb tsis tuaj yeem muab faib ua peb theem ntawm cov neeg siv (pib, nruab nrab, thiab qib siab) raws li ib txwm tau teev tseg thiab teev nyob rau hauv cov ntaub ntawv sib txawv ntawm cov tshuaj sib txawv thiab tshuaj. Qhov no yog vim qhov tseeb tias Letrozole yog ib qho tshuaj ntxiv uas tsis yog siv tshwj xeeb rau lub hom phiaj ntawm kev txhim kho kev ua tau zoo, tab sis nws yog siv los tawm tsam lossis txo ntau yam kev mob tshwm sim ntawm Estrogen thaum siv aromatizable anabolic steroids.
Qee qhov xwm txheej, Letrozole koob tshuaj kuj tseem tuaj yeem siv los ua kom cov tshuaj tiv thaiv endogenous ntawm Testosterone hauv cov txiv neej, uas tso cai rau cov tshuaj no siv los ua cov tshuaj ntxiv thaum PCT (Post Cycle Therapy) theem tom qab kawg ntawm lub voj voog anabolic steroid, tab sis. kev siv ntawm nws tus kheej rau lub hom phiaj no tsis yog ntau heev thiab tsis zoo li yuav ua rau pom kev ua tau zoo txhawb cov teebmeem. Letrozole txoj kev siv los ua ib qho endogenous Testosterone stimulating tus neeg saib xyuas yuav raug them ntxiv nyob rau hauv kom meej sai sai.
Rau lub hom phiaj ntawm kev tswj Estrogen thaum lub voj voog: Letrozole yog qhov zoo tshaj plaws aromatase inhibitor siv los txo cov qib ntawm Estrogen hauv lub cev thaum lub voj voog uas muaj kev siv cov aromatizable androgens (anabolic steroids uas muaj kev sib raug zoo los khi rau aromatase enzyme thiab nkag mus rau aromatization rau hauv Estrogen). Qhov no tau piav qhia yav dhau los hauv qhov kev taw qhia. Cov koob tshuaj Letrozole rau lub hom phiaj no npog ntau yam, thiab ntau npaum li cas Letrozole yuav tsum tau (thiab ntau npaum li cas) kuj tseem nyob ntawm ntau npaum li cas ntawm aromatizable anabolic steroids siv, tus neeg mob siab rau aromatase inhibitors, thiab tus nqi ntawm aromatization ntawm anabolic. steroids siv. Nrog rau qhov no tau hais, qhov dav dav ntawm Letrozole koob tshuaj yog kwv yees li 1.25mg - 2.5mg ib hnub. Muaj cov npoo loj heev rau kev hloov kho thiab cov neeg siv nyiam thaum nws los txog rau Letrozole ntau npaum, vim txhua tus neeg yuav tsum maj mam kho lawv cov koob tshuaj nyob ntawm seb lawv xav tias lub cev teb li cas. Qhov no tshwj xeeb tshaj yog rau Letrozole, uas yog lub zog tshaj plaws thiab muaj zog AI ntawm peb. Txawm hais tias 1.25mg ib hnub yog ntau dhau rau ntau tus neeg siv tshuaj anabolic steroid, thiab feem ntau cov koob tshuaj pom zoo yog 1.25mg txhua hnub, thiab feem ntau tuaj yeem ua tau tsawg dua tshwj xeeb tshaj yog xav txog ib nrab-lub neej ntawm Letrozole yog 2 - 4 hnub. Cov koob tshuaj Letrozole tuaj yeem hloov kho tau yooj yim yog tias tus neeg siv xav tias nws tsis ua haujlwm zoo txaus, lossis yog tias nws txo qis Estrogen ntau dhau.
Nco ntsoov tias lub tswv yim nrog kev siv cov aromatase inhibitors yog tswj cov qib Estrogen thiab coj lawv rov qab mus rau qhov qub physiological theem tsis zoo li kev txo qis thiab / lossis tshem tawm ntawm lawv, uas yuav ua rau muaj teeb meem hauv lub cev.
Poj niam Letrozole Dosage
Cov poj niam anabolic steroid cov neeg siv tsis tshua xav tau kev txhawj xeeb txog kev nce qib Estrogen, tab sis rau cov neeg uas muaj kev sib tw cev nqaij daim tawv uas yuav tsum tshem tawm cov dej tuav cuam tshuam nrog cov tshuaj Estrogen uas ua rau lub pliaj plob tsis so tswj, kev siv cov aromatase inhibitor xws li Letrozole (Femara) yuav tsim nyog. . Txawm li cas los xij, vim muaj lub zog loj ntawm Letrozole, nws raug pom zoo tias cov poj niam sim siv ib qho ntawm ob qho loj aromatase inhibitors ua ntej yuav siv Letrozole. Qhov no yog vim hais tias nws tau pom kev kho mob tias aromatase inhibitors qhov tseeb ua rau txo qis Estrogen hauv cov poj niam ntau dua li cov txiv neej.
Nws yog ib qho tseem ceeb uas yuav tsum nco ntsoov tias kev kho mob, Letrozole tau pom zoo siv rau cov poj niam tom qab yug me nyuam nkaus xwb, uas muaj qhov sib txawv ntawm cov tshuaj hormones piv rau cov poj niam ua ntej menopausal. Txawm hais tias ntawm cov poj niam cev xeeb tub tom qab mob qog noj ntshav mis, Letrozole yog siv los ua qhov chaw kawg kawg ntawm kev tiv thaiv kab mob qog noj ntshav tom qab tag nrho lwm yam kev kho mob thiab tshuaj tsis ua tiav. Vim tias cov ntaub ntawv kho mob tau qhia tias aromatase inhibitors muaj txiaj ntsig zoo rau cov poj niam ntau dua li cov txiv neej (nyob ntawm aromatase inhibitor hauv nqe lus nug siv),Cov koob tshuaj Letrozolentawm 1.25mg txhua hnub lossis ib zaug txhua ob hnub yuav tsum txaus thiab qhov tseeb ntau zaus dhau los, nyob rau hauv rooj plaub no tus neeg yuav xav tias yuav tsum tau kho kom tsawg dua lossis tsawg dua ntawm kev tswj hwm.
Letrozole Dosage rau nce Endogenous Testosterone Secretion thiab PCT (Post Cycle Therapy)
Nws tau hais yav dhau los hais tias Letrozole tuav lub peev xwm los nce qib endogenous ntawm Testosterone hauv cov txiv neej. Qhov no yog los ntawm qhov kev tawm tswv yim tsis zoo ntawm HPTA (Hypothalamic Pituitary Testicular Axis), uas tau pom tias ntau dhau ntawm Estrogen hauv cov txiv neej tuaj yeem ua rau txo qis cov zis ntawm endogenous Testosterone, ua rau hypogonadism. Letrozole tshwj xeeb hauv ntau cov kev tshawb fawb tau pom tias tuav lub peev xwm nce qib Testosterone los ntawm kev txo qis ntawm Estrogen. Ib txoj kev tshawb fawb tshwj xeeb tau soj ntsuam ib tus txiv neej laus uas pom cov teeb meem kev sib deev tsis zoo uas tshwm sim los ntawm qhov tsis tshua muaj endogenous androgen ntau lawm uas tau tswj hwm nrog cov koob tshuaj Letrozole, thiab txoj kev tshawb fawb tau xaus lus tias Testosterone qib tau rov zoo li qub physiological theem thiab kev ua haujlwm ntawm kev sib deev tau rov qab los. Nyob rau hauv txoj kev tshawb no, LH (Luteinizing Hormone) thiab FSH (Follicle Stimulating Hormone) tau nce, thaum SHBG (Sex Hormone Binding Globulin) tau txo qis. LH thiab FSH yog ob qho tseem ceeb gonadotropins uas taw qhia cov qe ntshav kom pib tsim Testosterone, thaum SHBG yog cov protein uas khi rau androgens thiab ua rau lawv tsis ua haujlwm (ntau yam tib yam aromatase inhibitors yuav khi rau aromatase enzyme thiab ua rau nws tsis ua haujlwm) . Tib txoj kev tshawb fawb tau txiav txim siab tias Letrozole ua tau zoo heev ntawm kev txo cov tshuaj Estrogen hauv cov txiv neej uas qhov kev xeem cov qib Estrogen yog qhov tseeb tsis tuaj yeem kuaj pom.
Ib qho tuaj yeem xaus lus yooj yim, raws li cov ntaub ntawv tau muab, tias Letrozole yuav yog qhov zoo ntxiv rau qhov tsim nyog nce ntxiv hauv Testosterone xav tau thaum lub sij hawm tom qab lub lis piam tom qab kev siv tshuaj anabolic steroid. Muaj ib qhov teeb meem nrog qhov sib ntxiv ntawm Letrozole hauv PCT program uas suav nrog kev siv SERMs xws li Nolvadex thiab Clomid, uas yog lub npe hu ua cov khoom tseem ceeb rau PCT program. Qhov teeb meem tib yam no tshwm sim hauv Arimidex, tab sis tsis yog hauv Aromasin (Exemestane). Qhov teeb meem yog tias Letrozole thiab Nolvadex (nrog rau Arimidex thiab Nolvadex) ob leeg ncaj qha tawm tsam ib leeg. Ib txoj kev tshawb fawb tau pom tias thaum Letrozole siv nrog Nolvadex, Nolvadex yuav txo cov ntshav plasma concentration ntawm Letrozole (nrog rau Arimidex, lwm yam siv aromatase inhibitor).
Qhov xaus ntawm no yog tias kev siv Letrozole thiab Nolvadex ua ke yog lub tswv yim phem heev. Yog li ntawd, Letrozole txoj kev siv los ua PCT feem ntau txwv yog siv nrog Nolvadex. Hloov chaw, nws siv nrog HCG yuav muaj txiaj ntsig zoo dua, tab sis qhov no kuj nthuav tawm qhov teeb meem ntawm qhov tseem ceeb ntawm SERM rau lub hom phiaj ntawm endogenous Testosterone stimulation tsis tuaj. Yog li ntawd, ib qho kev xaiv zoo dua aromatase inhibitor rau PCT es tsis txhob Arimidex yuav yog Aromasin (Exemestane), vim hais tias tsis zoo li Letrozole, Aromasin tsis tau pom muaj nws cov txiaj ntsig tau tshem tawm lossis txo los ntawm Nolvadex raws li qhia hauv kev tshawb fawb.
Kev Tswj Xyuas Kom Zoo thiab Lub Sijhawm ntawm Letrozole Dosages
Tsis muaj kev txiav txim siab tshwj xeeb nrog kev tswj hwm ntawm cov koob tshuaj Letrozole, thiab nws tuaj yeem noj txhua lub sijhawm ntawm nruab hnub (thaum sawv ntxov, hmo ntuj, ua ntej, thaum, lossis tom qab noj mov).
Ib qho tseem ceeb uas yuav tsum tau ua nrog cov koob tshuaj Letrozole yog qhov tseeb nws yuav siv sijhawm 60 hnub ua ntej cov ntshav plasma qib ntawm Letrozole tau mus txog qib siab tshaj plaws, txawm tias nws lub neej ib nrab yog kwv yees li 2 - 4 hnub. Letrozole muaj lub qhov rais ntev tshaj plaws ntawm lub sijhawm rau cov ntshav plasma kom ncav cuag qhov siab tshaj plaws ntawm tag nrho peb qhov loj aromatase inhibitors (hloov, Arimidex thiab Aromasin xav tau 7 hnub txhawm rau kom pom cov ntshav ntshav siab kom ncav cuag).
Cov ntaub ntawv kho mob
| Hom | FIERCE |
|
Cov npe lag luam |
Femara, letrozole |
|
CAS |
112809-51-5 |
|
Molar loj |
285.310 |
|
Formula |
C17H11N5 |
|
Purity |
Tshaj 98% |
|
Yam khoom |
2.5mg * 50 |
Txhua yam kev xav tau, thov hu rau peb
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Kev cia siab thiab txiaj ntsig los ntawm Letrozole Dosages
Vim tias Letrozole yog nyob deb ntawm qhov zoo tshaj plaws aromatase inhibitor nrog lub peev xwm los txo cov qib Estrogen mus rau qib tsis tuaj yeem kuaj pom, cov neeg siv yuav tsum tau ceev faj kom ntseeg tau tias cov qib Estrogen no tsis poob qis dhau los ua kev noj qab haus huv. Raws li Estrogen qib poob qis, lub cev yuav siv sij hawm ntau dua 'grainier' thiab 'ripped' saib vim qhov poob dej tuav los ntawm Estrogen. Qhov no ua rau muaj tsawg heev rau tsis muaj cov kua dej subcutaneous, uas yuav nthuav tawm cov pob txha hauv qab kom pom tseeb dua. Ib qho kev zam rau qhov teeb meem ntawm kev tshem tawm Estrogen tiav yog nyob rau hauv kev sib tw bodybuilders uas yuav tsum tau yuav luag tag nrho tshem tawm cov dej tuav nyob rau hnub sib tw. Nyob rau hauv cov xwm txheej zoo li no, Letrozole tej zaum yuav yog qhov zoo tshaj plaws aromatase inhibitor siv saum toj no tag nrho lwm cov AIs ntawm tag nrho cov koob tshuaj siv los ntawm cov neeg ncaws pob sib tw tsuas yog hnub ua rau muaj kev sib tw rau lub cev hloov cov laj thawj yav dhau los. Kev txo qis ntawm Estrogen yuav tsum tsis txhob khaws cia ntev dua 48 teev rau kev noj qab haus huv.
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