
STADA Testosterone Acetate Rau Bodybuilding CAS: 1045-69-8
Testosterone acetate yog ib qho hluavtaws androstane steroid thiab testosterone ester. Nws yog siv feem ntau rau kev kho tshuaj hormone hloov pauv (HRT) hauv cov txiv neej nrog hypogonadism thiab rau qee hom mob qog noj ntshav hauv cov poj niam. Raws li daim ntawv esterified ntawm testosterone, nws yog tus cwj pwm los ntawm nws cov tshuaj pharmacokinetics, kev siv tshuaj kho mob, thiab cov teebmeem ntawm lub cev. Hauv qab no yog cov lus sib tham txog testosterone acetate, npog nws cov khoom, kev siv, cov txiaj ntsig, ntau npaum li cas, ib nrab-lub neej, ncig, thiab ntau dua.
Cov khoom ntawm Testosterone Acetate
Chemical Structure thiab Formula:
IUPAC lub npe:(17) -3-Oxoandrost-4-en-17-yl acetate
Molecular Formula: C21H30O3
Molecular Luj:330.46 g / mol
Chemical Structure:
Lub cev muaj zog:
Qhov tsos:Dawb los yog tawm-dawb crystalline hmoov
Melting Point:137-140 degree
Solubility:Soluble nyob rau hauv cawv, acetone, thiab lwm yam organic solvents; xyaum insoluble hauv dej.
Pharmacological Properties:Testosterone acetate yog Testosterone ester, uas txhais tau hais tias nws yog testosterone khi rau ib qho acetate ester los pab txhawb nws tso rau hauv cov hlab ntsha nyob rau lub sijhawm. Qhov esterification no hloov pauv cov tshuaj pharmacokinetics ntawm testosterone, tso cai rau kev tso tawm qeeb qeeb ntawm qhov chaw txhaj tshuaj, yog li ncua sijhawm ntawm nws cov teebmeem.


Kev siv Testosterone Acetate
Kev siv kho mob:
1. Hypogonadism hauv txiv neej:
Testosterone acetate feem ntau yog siv rau hauv testosterone hloov kho (TRT) los kho hypogonadism, ib qho mob uas muaj cov qib testosterone tsawg hauv cov txiv neej. Cov tsos mob ntawm hypogonadism suav nrog txo libido, erectile kawg, qaug zog, kev nyuaj siab, thiab poob ntawm cov leeg nqaij.
2.Delayed Puberty hauv Cov Tub:
Nws tuaj yeem siv los kho cov tub hluas nrog ncua kev puberty, pab txhawb kev loj hlob ntawm kev sib deev yam ntxwv xws li kev sib sib zog nqus ntawm lub suab, kev loj hlob ntawm lub ntsej muag thiab lub cev plaub hau, thiab nce cov leeg nqaij.
3. Mob cancer mis hauv poj niam:
Qee zaum, testosterone acetate yog siv los kho qee yam mob qog noj ntshav hauv cov poj niam. Nws pab los ntawm inhibiting kev loj hlob ntawm estrogen-dependent cancer hlwb.
4.Gender Dysphoria:
Testosterone acetate tuaj yeem raug sau rau cov txiv neej hloov pauv (poj niam-rau-txiv neej) ua ib feem ntawm kev kho tshuaj hormone hloov mus ua kom tus txiv neej.
Cov txiaj ntsig ntawm Testosterone Acetate
1. Txhim kho Libido thiab kev sib deev muaj nuj nqi:
Testosterone yog qhov tseem ceeb rau kev ua haujlwm ntawm kev sib deev hauv cov txiv neej. Ntxiv nrog rau testosterone acetate tuaj yeem txhim kho libido, txhim kho kev sib deev, thiab kho erectile kawg.
2. Ua kom cov leeg nqaij thiab muaj zog:
Testosterone muaj cov teebmeem anabolic, txhawb cov protein synthesis thiab cov leeg nqaij. Qhov no ua rau nws muaj txiaj ntsig zoo rau kev nce cov leeg nqaij thiab lub zog, uas yog tshwj xeeb tshaj yog muaj txiaj ntsig zoo rau cov tib neeg uas muaj cov nqaij ntshiv.
3. Txhim kho lub siab thiab lub zog theem:
Tsawg testosterone qib feem ntau cuam tshuam nrog kev xav tsis zoo xws li kev nyuaj siab thiab qaug zog. Testosterone acetate tuaj yeem txhim kho kev xav, nce qib zog, thiab txhim kho kev noj qab haus huv tag nrho.
4. Kev txhim kho pob txha pob txha:
Testosterone plays lub luag haujlwm tseem ceeb hauv cov pob txha metabolism. Nws supplementation pab nyob rau hauv ua kom cov pob txha ntxhia pob zeb ceev, yog li txo qhov kev pheej hmoo ntawm osteoporosis thiab pob txha.
5. Mob plawv:
Testosterone tau pom tias muaj txiaj ntsig zoo rau kev noj qab haus huv ntawm cov hlab plawv, suav nrog kev txhim kho lipid profile, txo cov roj visceral, thiab txhim kho endothelial muaj nuj nqi.
Dosage ntawm Testosterone Acetate
Qhov ntau npaum ntawm testosterone acetate txawv nyob ntawm tus neeg mob, hnub nyoog, thiab cov lus teb rau kev kho mob. Nws yog siv los ntawm kev txhaj tshuaj intramuscular. Cov koob tshuaj ib txwm muaj xws li:
Rau Hypogonadism:
● Thawj koob tshuaj:50-100 mg muab tshuaj txhua txhua 2-4 lis piam.
● Kev Kho Kom Zoo:Kho raws li cov qib testosterone hauv cov ntshav, feem ntau yog 50-200 mg txhua 2-4 lub lis piam.
Rau Delayed Puberty:
● Thawj koob tshuaj:50 mg muab txhua txhua 2-4 lub lis piam rau 4-6 hli.
● Kev Kho Kom Zoo:Kho raws li cov lus teb thiab kev loj hlob ntawm kev puberty.
Rau Mob Cancer:
● koob tshuaj:50-100 mg muab tshuaj txhua 1-2 lub lis piam, nyob ntawm cov lus teb thiab cov kev mob tshwm sim.
Rau Poj Niam Dysphoria:
● koob tshuaj:50-200 mg muab tshuaj txhua 1-2 lub lis piam, nyob ntawm tus neeg xav tau kev pab thiab teb rau kev kho mob.
Ib nrab-Lub neej thiab kev ncig
Ib nrab neej:
●Lub neej ib nrab ntawm testosterone acetate yog luv luv piv rau lwm yam testosterone esters. Nws yog kwv yees li 3 hnub. Ib nrab-lub neej luv luv yuav tsum tau noj ntau zaus kom tswj cov ntshav siab.
Kev ncig:
● Thaum txhaj tshuaj intramuscular, testosterone acetate maj mam nqus mus rau hauv cov hlab ntsha. ester daim ntawv cog lus yog hydrolyzed los ntawm esterases, tso tawm dawb testosterone. Tus dawb testosterone ces exerts nws physiological teebmeem los ntawm khi rau androgen receptors nyob rau hauv ntau yam ntaub so ntswg.
●Testosterone feem ntau metabolized nyob rau hauv daim siab, qhov uas nws hloov mus rau hauv dihydrotestosterone (DHT) thiab estradiol. DHT yog ib qho muaj zog dua androgen, thaum estradiol yog ib qho tshuaj estrogen. Ob leeg metabolites pab txhawb rau tag nrho cov teebmeem ntawm testosterone.
Pharmacodynamics
Testosterone exerts nws cov teebmeem los ntawm ntau yam mechanisms:
1. Androgen Receptor Binding:
Testosterone khi rau androgen receptors nyob rau hauv lub hom phiaj cov ntaub so ntswg xws li cov leeg, pob txha, thiab lub cev xeeb tub. Qhov kev khi no ua rau lub receptor, ua rau muaj kev hloov pauv ntawm cov noob qhia thiab cov teebmeem ntawm tes.
2. Kev hloov pauv rau DHT:
Testosterone hloov mus rau DHT los ntawm enzyme 5 -reductase. DHT khi rau androgen receptors nrog ntau dua affinity dua testosterone, ua rau muaj zog androgenic cuam tshuam ntau dua.
3. Kev hloov pauv rau Estradiol:
Testosterone yog aromatized rau estradiol los ntawm enzyme aromatase. Estradiol khi rau cov tshuaj estrogen receptors, kho qee qhov cuam tshuam ntawm testosterone, tshwj xeeb tshaj yog ntawm pob txha ntom thiab libido.
Cov Kev Phem Phem thiab Kev Phem
Zoo li txhua yam tshuaj, testosterone acetate muaj kev pheej hmoo ntawm kev phiv. Cov no tuaj yeem sib txawv hauv qhov hnyav thiab ntau zaus thiab tuaj yeem suav nrog:
Cov teebmeem Estrogenic:
● Gynecomastia (kev loj hlob ntawm lub mis hauv cov txiv neej)
● Dej tuav thiab edema
Cov teebmeem ntawm Androgenic:
● Pob txuv thiab oily daim tawv nqaij
● Cov plaub hau poob (nyob rau hauv cov tib neeg predisposed rau txiv neej qauv baldness)
● Nce lub cev thiab lub ntsej muag cov plaub hau loj hlob
Kev saib xyuas thiab ua raws
Kev saib xyuas tsis tu ncua yog qhov tseem ceeb los xyuas kom muaj kev nyab xeeb thiab siv tau zoo ntawm testosterone acetate. Qhov no suav nrog:
Ntshav Testosterone Qib:Txhawm rau kho ntau npaum li cas thiab xyuas kom muaj kev kho mob.
Lipid Profile:Txhawm rau soj ntsuam cov roj cholesterol.
Kev kuaj lub siab ua haujlwm:Txhawm rau txheeb xyuas qhov muaj peev xwm hepatotoxicity.
Ua kom tiav ntshav suav (CBC):Txhawm rau soj ntsuam cov qib hematocrit thiab hemoglobin.
Prostate-Specific Antigen (PSA):Txhawm rau tshuaj xyuas kev noj qab haus huv prostate hauv cov txiv neej.
Cov ntaub ntawv kho mob
| Hom |
STADA |
|
Cov npe lag luam |
Aceto-Sterandryl, Aceto-Testoviron, Amolisin, Androtest A, Deposteron, Farmates, Perandrone A |
|
CAS |
1045-69-8 |
|
Molar loj |
330.468 |
|
Formula |
C21H30O3 |
|
Purity |
Tshaj 98% |
|
Yam khoom |
75 mg/ml |
Txhua yam kev xav tau, thov hu rau peb
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Xaus
Testosterone acetate yog ib qho tseem ceeb kho tus neeg sawv cev rau kev kho mob ntawm ntau yam mob uas muaj feem xyuam rau testosterone deficiency. Nws muaj peev xwm muab cov qib testosterone ruaj khov ua rau nws tsim nyog rau kev kho tshuaj hormone hloov. Txawm li cas los xij, zoo li txhua yam tshuaj, nws yuav tsum tau ua tib zoo xav txog cov txiaj ntsig thiab kev pheej hmoo, kev siv tshuaj kom tsim nyog, thiab kev saib xyuas tsis tu ncua kom ntseeg tau tias tus neeg mob muaj kev nyab xeeb thiab ua tau zoo. Raws li nrog rau kev kho tshuaj hormones, kev kho tus kheej ntawm kev kho mob raws li cov neeg mob tshwj xeeb yog qhov tseem ceeb rau kev ua tiav cov txiaj ntsig zoo.
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