
SARMS LGD3303 HMOOV RAU LUB CAIJ BODYBUDING CAS: 1196133-39-7
Selective Androgen Receptor Modulators (SARMs) are a class of therapeutics designed to mimic the muscle-building effects of anabolic steroids while minimizing androgenic side effects. LGD-3303, developed by Ligand Pharmaceuticals, is a potent, nonsteroidal SARM initially investigated for conditions like muscle wasting and osteoporosis .
Taw qhia rau sarms thiab lgd -3303
Selective Androgen Receptor Modulators (SARMs) are a class of therapeutics designed to mimic the muscle-building effects of anabolic steroids while minimizing androgenic side effects. LGD-3303, developed by Ligand Pharmaceuticals, is a potent, nonsteroidal SARM initially investigated for conditions like muscle wasting and osteoporosis .} tsis zoo li steroids, nws xaiv cov khoom siv thiab pob txha, muab cov phiaj xwm ua kom zoo rau kev txhim kho lub cev thiab kev ua haujlwm {{}


Kev Tshawb Nrhiav thiab Kev Loj Hlob
LGD -3303 tawm los ntawm cov tshuaj ntsuam ligand uas tseem ceeb tshaj plaws rau cov ntaub so ntswg zoo li ostarine ua ntu zus los ntawm ostarine (mk {}) {4 {4} Txawm hais tias theem kuv tau sim ua kom muaj txiaj ntsig zoo, tawm hauv cov kev tshawb fawb hauv kev tshawb fawb ua "tus qauv share sharm."
Cov qauv tshuaj lom neeg thiab cov kws muag tshuaj
LGD-3303's structure features a quinoline core, enhancing AR binding specificity. It exhibits a 10:1 anabolic-to-androgenic ratio in preclinical models, compared to testosterone's 1:1 ratio. This selectivity reduces risks of prostate enlargement or hair loss. Yam tsis zoo li cov tshuaj steroids, nws tsis ua kom tawg rau hauv estrogen, mitigating gynecomastia txaus ntshai {}}
Mechanism ntawm Kev Ua
LGD -3303 activ activ activ activ ar ar {} Nws xaiv cov txiaj ntsig. Nws muaj kev vam meej - gonadal (HPG) Axis supression pom nrog cov tshuaj steroids, nws muaj ib qho kev nyab xeeb profile, txawm tias qhov kev nyab xeeb me me tseem muaj peev xwm ua tau ntawm cov tshuaj siab .
Cov Nta Tshwj Xeeb Ntawm LGD -3303
● Cov Bioavility Siab: Kev tswj hwm qhov ncauj nrog ~ 90% nqus .
● Ntev ib nrab-lub neej: ~ 24-30 teev, ua kom muaj kev phom sij ib zaug .
● Nonsteroidal Xwm: Zam kev hepatotoxicity txuas rau 17 -} alkylated steroids .
● Nqaij-TSHWJ XEEB Hypertrophy: Txhawb kev ntshiv rog uas tsis muaj dej khaws cia .
Cov ntawv thov hauv kev ua haujlwm ntawm lub cev
Rulkers Bulking Cycles: Txhim kho cov ntshiv loj nce (5-10 lbs ntau tshaj 8 lub lis piam) .
● Txiav kauj tshuag: Khaws cov leeg nqaij thaum lub sijhawm muaj nqi caloric .
Recomposition: Fixataneous rog poob thiab cov leeg kev loj hlob .
● Kev raug mob rov qab: Kho kom nrawm dua ntawm cov ntaub so ntswg sib txuas .
Cov Ntawv Pov Thawj Cov Nyiaj Pab
● Cov leeg kev loj hlob: Cov ntaub ntawv preclinical qhia 6-8% leeg loj nce hauv 4 lub lis piam .
HeCS Ecce EcSet Enj zuj zus: Cov neeg siv daim ntawv tshaj tawm 15-20% boosts nyob rau hauv nqa zoo li lub rooj ntev xovxwm {2.
● Rog oxidation: Upregulates meabolic enzymes, ib pab lipolysis .
● Cov pob txha ceev: Kev tiv thaiv kab mob osteoporosis tiv thaiv .
Muab thiab tswj hwm
● Pib Pib: 5-10 mg / hnub, coj tus yuam sij nrog rog rau nqus .
Huaj vam: 15-20 mg / hnub (decit koob tshuaj vim ntev ib nrab-lub neej) .
● Kev voj voog ntev: 8-12 lub lis piam, ua raws PCT .
* Nco tseg: Tib neeg cov kev sim siv 1-3 mg / hnub; Cov koob tshuaj ntau dua yog anecdotal . *
Kev voj voog studing tswv yim
● Cov tsev loj: Tshooj nrog Mk -677} (ibtamoren) rau i{-1.
● Kev txiav: Sib txuas nrog cardarine (gw -501516}) rau kev ua kom ntev.
PCT PCT Cov khoom tseem ceeb: Suav nrog nolvadex (20 mg / hnub) rau 4 lub lis piam tom qab-voj voog .
Ib nrab-lub neej thiab koob zaus
Nrog 24 - {30- teev ib nrab-lub neej, ib hnub txhua hnub nyob ruaj khov {}}} .
Tom qab kev cobqhy (Pct)
Txawm tias metoids tshaj cov tshuaj steroids, lgd -3303 sudpresses Nature Testosterone}}} pcct raws nrho:
● Nolcadadex: 20 mg / hnub (lub lis piam 1-2), 10 mg / hnub (lis piam 3-4) .
FandingMhene: 12 {{.}} 5 mg / hnub rau 4 lub lis piam (ua tau zoo rau lh / fsh rov qab).
Kev Nyab Xeeb thiab Kev Mob tshwm sim
● Muaj ntau: Yias SOARCE (30-50% Testosterone poob) .
Tsis tshua muaj: Mob taub hau, lipid profile hloov (HDL txo) .
Kev rho me nyuam: Daim siab txhawb nqa (NAC), roj tswj kav (Omega -3 s) .
Raws cai
LGD -3303 Tsis yog FDA-tau pom zoo thiab raug muag los ntawm Wada {2} Zoo} Kev Tshawb Fawb Raws Li Kev Tshawb Fawb, "nws txoj cai sib txawv; txwv nyob hauv Australia, tsis ntseeg nyob rau hauv lub u . s {} Tab sis tsis rau tib neeg .
Cov neeg siv kev paub
Anecdotal qhia nthuav dav lub zog nce thiab vascularity, txawm hais tias qee cov ntawv sau tseg} {lbs {1} .
Cov chaw kuaj mob tshawb nrhiav kev pom
Ib qho kev kawm 2010 nyob rau hauvPhau Ntawv Journal ntawm Pharmacologypom lgd -3303 muaj ntau zuj zus los ntawm 9% ntawm cov nas hauv pawg neeg. Cov ntaub ntawv hauv tib neeg nyob tsis muaj, hais txog kev ceev faj
Piv rau lwm tus sarms
Vs . lgd -4033: Lgd -3303 Tau ntau dua archinity tab sis kev tsim kho cov keeb kwm kev txhawb ntxiv {}}
Vs . rad -140: Tsawg dua Androgenic, ua rau nws preferable rau kev txiav .
Kev Txiav Txim Siab
Thaum sarms muab txoj kev nyab xeeb rau cov tshuaj steroids, lawv cov kev tsis muaj kev siv tau siv cov kev txhawj xeeb ntev thiab kev ncaj ncees hauv cov kis las.
Yav tom ntej zeem muag
Kev tshawb fawb txuas ntxiv mus rau hauv cov ntaub so ntswg yuav ua kom lub LGD -3303}} rau kev kho cachexia {}}
Cov ntaub ntawv kho mob
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Kev Lag Luam Npe |
LGD3303 |
|
Cas |
1196133-39-7 |
|
Tus hniav loj |
342.75 |
|
Mf |
C16H14Tus nplais3N2O |
|
Kev coj dawb huv |
Saum toj no 98% |
|
Kev tsim nyog |
Dawb Cyrstalline Hmoov |
Kev xav tau, thov hu rau peb
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Tag
LGD -3303 nthuav tawm kev xaiv lub cev rau lub cev thiab tsis muaj kev cuam tshuam rau cov leeg, hais txog PCT thiab kev saib xyuas PCT thiab Kev Noj Qab Haus Huv.
Cim npe nrov: SARMS LGD3303 HMOOV RAU LUB CAIJ BODYBUDING CAS: {{}}}} {{{{} Cov chaw tsim khoom, cov chaw tsim khoom, Hoobkas
