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Stromusc GW501516 (Cardarine) 10Mg rau Case: 317318-70-0

Stromusc GW501516 (Cardarine) 10Mg rau Case: 317318-70-0

GW501516 (Cardarine) yog kev tshawb fawb tshawb xyuas tsis pom zoo rau tib neeg siv los ntawm txhua lub cev tswj hwm lub cev (FDA, EMA, thiab lwm yam). Cov kev tshawb fawb tseem ceeb preclinical, tshwj xeeb los ntawm Asmeskas Kev tsim kho Cancer National Cancer hauv ntau hom tsiaj ntawm ntau cov tsiaj uas muaj feem xyuam rau tib neeg siv. Nws txoj kev loj hlob rau kev kho kev siv tau raug tso tseg vim tsis muaj kev pheej hmoo carcinogenable kev pheej hmoo. Qhov kev tshawb fawb no tau nthuav tawm ib leeg tsuas yog rau cov ntaub ntawv thiab kev nkag siab kev nkag siab hauv zej zog kev ua kom lub zej zog. Tus kheej - kev tswj hwm yog muaj zog poob siab thiab muaj kev phom sij.

Xa kev nug
Hauj lwm lawm

Dab tsi yog GW501516 (Cardarine)?

GW501516, feem ntau hu ua cardarine, yog synthetic peroxisome proliferator - ushing} ushing} ua haujlwm recta (pparΔ) agonist. Ameslikas tau tsim los ntawm xyoo 1990 los ntawm GlaxosmithKline (GSK) thiab Ligand Pharmeticals, nws qhov kev tshawb fawb txog dyslipic) / triglycal ntau qib), thiab rog. PARDΔ yog cov protein nuclear recein uas tswj hwm cov ntsiab lus ntawm cov txheej txheem ntawm cov txheej txheem cellular, feem ntauLiipid metabolism thiab lub zog siv.Ua kom muaj ntawm Parpently Fundamentally reprograms hlwb, kom haum cov leeg leeg cov roj thiab txhim kho roj ua haujlwm thiab cov roj biogenesis (tsim cov khoom siv cellular cellular).

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Nta ntawm GW501516 (Cardarine)

● Mechanism ntawm kev nqis tes ua:Xaiv thiab muaj zog ppparΔ agonist. Nws khi rau pparΔ hauv lub cell nucleus, sib sau ua ke uas khi rau cov ntaub ntawv DNA (PPP cov ntsiab lus ntawm lub hom phiaj.

● Metabolic reprogramming:Hloov Cellular lub zog nyiam los ntawm cov piam thaj qabzib (carbohydrates) ntawm fatty acid oxidation (hlawv rog). Qhov no tshwm sim feem ntau hauv cov leeg pob txha, cov leeg nqaij lub plawv, thiab daim siab.

● Qhov Endaully Txhim Kho:Dramatically nce kev tawm dag zog thiab nkees tsis kam nyob rau hauv cov qauv tsiaj los ntawm kev txhim kho cov leeg nqaij ua kom zoo thiab tawm tsam glycogen khw.

At Lipid Hloov:Lowers LDL ("Phem"))))) ("triglycerides thaum nce HDL (" Zoo ") (cholesterol).

Insulin insulin rhiab:Txhim kho cov kua qaub thiab kev siv hauv cov leeg nqaij, txhim kho insulin rhiab.

● Cov androgenicity tsawg:Tsis yog tshuaj hormones (steroid lossis prohormone). Tsis khi rau androgen receptors. Tsis ua rau Androgenic phiv (Pob txuv, cov plaub hau poob, teeb meem prostate, muaj kev phom sij rau cov poj niam).

● Tshuaj lom neeg Xwm:Tsis - hormonal, cov tshuaj me. Ruaj khov nyob rau hauv chav tsev kub.

Asn nyaj pheej txaus ntshai loj:Pov thawj carcinogenicity nyob rau hauv cov tsiaj qauv thoob plaws ntau lub plab thiab hom tsiaj ntawm kev kho cov koob tshuaj. Qhov no yog nws lub ntsiab lus thiab tsis tsim nyog feature.

Purported daim ntawv thov hauv kev ua kom lub cev (raws li kev siv hluav taws xob & anecdote)

● Rog Rog Catalyst:Los ntawm kev yuam cov leeg pob txha los xum oxidize fatty acids rau lub zog, txawm tias muaj kev sib tw nrawm nrawm dua li acceler {1} {{1} {1} {1} Puas muaj kev nrawm nrawm, ua rau lub cev nqaij ntuag qis dua.

● Qhov AVURITUR Accevion & Cov Khoom Siv Muaj Peev Xwm Ua Haujlwm:Lub glycogen - Cov txiaj ntsig sparing yog cov nyhuv uas muaj lub cev ua haujlwm los cob qhia kev nyuaj, thiab ntau dua, thiab ntau zaus. Siab - rec teeb, thiab tag nrho cov ntim ntim yuav muaj peev xwm nce ntxiv, kov yeej cov tawv nqaij tsis muaj zog. Qhov no yog nws feem ntau cov nyhuv tshaj tawm hauv Anecdotal cov account.

● Rov qab soj ntsuam:Txhim kho mitochondrial muaj nuj nqi thiab txo cov mob ppparδ

● "Cov leeg nqaij" - sparing "thaum txiav:Los ntawm muab lwm txoj hauv kev, cov zog siv tau zoo (rog), nwstej zaumPab kom txuag cov leeg nqaij ntshiv thaum muaj kev tiv thaiv kab mob calorie los ntawm txo lub cev lub cev xav tau kom catabolize cov nqaij protein rau lub zog (gluconeogenesis).

● Txhim kho Lipid Profile:Thaum lub sij hawm feem ntau yog cov cim kev noj qab haus huv, qis dua HDL tuaj yeem txhawb nqa theem, txawm tias qhov no yog qhov tseem ceeb tshaj plaws los ntawm kev muaj mob cancer.

Insulin Insulity Txhawb Nqa:Tej zaum yuav pab tau cov zaub mov muaj kev faib tawm, muaj peev xwm coj tau ntau cov as-ham rau cov leeg nqaij, qhov tseem ceeb tshaj plaws hauv hypercaloric (bulking) theem.

Purported cov txiaj ntsig (nyob rau hauv cov ntsiab lus ntawm lub homphiaj ntawm lub hom phiaj)

● Txhim kho cov txhais lus:Ua kom muaj roj ua kom nrawm pom pom cov leeg cov leeg thiab sib cais.

Ulder Cov ntim ntau ntxiv & kev siv:Tso cai rau kev teeb tsa ntau dua, reps, thiab cov thauj khoom hnyav dhau sijhawm vim kev txo qis.

Muab cov teeb meem zoo tshaj plaws:Ua kom siab siab -}}} {{-} Lub Xeev Cardio Ntau Metable thiab siv tau zoo rau kev poob rog.

● Cov leeg muaj peev xwm tuav tseg:Tej zaum yuav pab tswj cov tawv tawv - khwv tau cov leeg nqaij thaum lub cev muaj roj ua kom nruj.

● Tsis - hormonal:Zam kev cuam tshuam kev phiv los ntawm anabolic steroids (androgenic, estrogenic, hepatotoxic).

● Ceev xwm ceev:Qhov cuam tshuam ntawm kev ua siab ntev yog feem ntau qhia nyob rau hauv cov hnub.

Qhov teeb meem tseem ceeb: kev siv tshuaj (10mg tshwj xeeb) & carcinogenicity

Qhov no yog lub crux ntawm qhov txaus ntshai. Tus10mg noj ntau npaum li cas tau muab tso tseg anecdotallynyob rau hauv lub cev lub voj voog. Txawm li cas los xij, kev nkag siab nws cov keeb kwm thiab kev pheej hmoo yog qhov tseem ceeb tshaj plaws:

Keeb Kwm:Txwv tib neeg chaw kuaj mob (theem I / II) rau cov kab mob metabolic siv tau xaim hluav taws xob los ntawm2.5mg rau 10mg txhua hnubCov. Qee qhov kev tshawb fawb pom tias yuav cuam tshuam lipid zoo li 10mg. Qhov no tau tsim tawm 10mg koob tshuaj nyob hauv kev tshawb fawb Lexicon, uas yog tom qab ntawd saws (recklessly) los ntawm kev ua haujlwm txhim kho zej zog.

Cov kab mob rau kev mob cancer:TusFDA cov ncauj lus kom ntxaws ntawm GSK cov ntaub ntawv ua ntejqhia cov txiaj ntsig pom tseeb:

○ Qhov pib pib ntawm cov qog hauv ntau cov ntaub so ntswg (mob siab, lub plab, tawv nqaij, lub plab, lub plab, hauv plab) hauv nas thiab nas.

○ hlav tau tshwm sim ntawmTag nrho cov koob tshuaj kuaj, suav nrog koob tshuajqi duatshaj li 10mg / hnub nyob rau mg / kg hauv paus.

○ Tus nqi carcinogenic tau pomhauv lub lis piamnyob rau hauv qee qhov kev tshawb fawb.

    ○Mechanism:PARKTδ agonism nws tus kheej yog cuam tshuam hauv cov qog nqaij hlav thiab kev nce qib, tshwj xeeb yog cov ntaub so ntswg epithelial. Mob mob rau kev ua kom muaj kev cuam tshuam ntawm kev cai cellular.

Tib neeg txoj kev pheej hmoo tsis paub (tab sis feem ntau):Thaum ntev {- sij hawm kawm tib neeg cov kev tshawb fawb), tus kws twv tsis tau muaj txiaj ntsig), cov kev tshawb pom zoo ib yam nyob hauv tib neeg cov koob tshuaj ntawm cov koob tshuaj no.Tsis muaj kev nyab xeeb lossis tsim kev tshuaj rau tib neeg kev siv.Siv 10MG txhua hnub yog ua si Lavxias teb Lavxias roulette nrog kev pheej hmoo mob cancer raws cov tsiaj cov ntaub ntawv.

Kev voj voog (siv qauv - theoretical & heev pheej hmoo)

Txawm hais tias muaj kev pheej hmoo, cov qauv tau sib tham txog:

● Rog poob / txiav lub voj voog:Feem ntau 6-8 lub lis piam ntawm 10-20mg / hnub (feem ntau cais AM / PM). Lub hom phiaj yog nrawm ua rog poob thiab ua kom ntev rau kev noj haus / cardio.

● Xaus / Ua tau zoo Ciaje:Feem ntau 4-6 lub lis piam ntawm 10-20mg / hnub, tsom lub peev xwm ntawm kev cob qhia muaj peev xwm.

● "Choj" ntawm Steroid Cycles:Siv thaum tawm - lub sij hawm los ntawm cov tshuaj steroids los ntawm kev ua kom ntev thiab muaj roj ploj, ntau zaus rau ncua sijhawm (txaus ntshai).

● Tseem ceeb tebeats:Lub voj voog ntev dua nce qib kev ua haujlwm carcinogen. Stacking nrog lwm cov tebchaw (zoo li sarms lossis steroids) ntxiv kev tsis paub kev pheej hmoo txaus ntshai thiab metabolic quav.Txhua lub voj voog uas muaj Cardarine nqa cov mob cancerable.

Ib nrab - lub neej thiab noj suing

Ib nrab - lub neej:GW501516 muaj ntev ntev ib nrab - lub neej nyob hauv tib neeg, kwv yees yuavKwv yees li ntawm 16-24 teevraws li cov ntaub ntawv tsawg ntawm cov ntaub ntawv ntawm tib neeg.

Ntsiab lus:Vim tias qhov ntev ib nrab - lub neej,Thaum - kev noj txhua hnub txhua hnub yog txaustxhawm rau tswj cov ntshav ruaj khov. Noj nws ib zaug txhua hnub, zoo nyob rau tib lub sijhawm txhua hnub (piv txwv li, thaum sawv ntxov), yooj yim rau cov regimen. Splitting qhov tshuaj (piv txwv li, 5mg kuv / 5mg PM) tsis tsim nyog thiab tsis muaj chaw muag tshuaj kom zoo dua. Lub ntev ib nrab- lub neej kuj txhais tau tias cuam tshuam rau ib hnub lossis ob xyoos tom qab txuas.

PCT (post {{- kev voj voog kev kho) -} ib tug misnomer

● Tsis yog hormonal:GW501516 does not suppress the body's natural production of testosterone or other hormones via the hypothalamic-pituitary-gonadal (HPG) axis like anabolic steroids or SARMs do. Nws tsis ua rau "kaw" lossis xav tau hormonal rov pib dua.

● Yuav tsum muaj cov pct ib txwm muaj:MuajTsis xav tauRau cov tub ntxhais kawm (xaiv tshuaj estrogen receptor modulators) zoo li tamoxifen (Nolvadee (CLOMIPALEX) lossis clomid) lossis hCG tom qab ib tug cardarine -}}. Cov tshuaj no tsis muaj txiaj ntsig thiab cuam tshuam rau cov laus tsis muaj kev ntxhov siab.

● Xyuas txog kev soj ntsuam kev noj qab haus huv (qhov tseem ceeb (qhov tseem ceeb):Vim yog carcinogenic pheej hmoo, tustsuaslub luag haujlwm "tshaj tawm -} kev sib yuav" kev txiav txim siab yogkev soj ntsuam kev noj qab haus huv saib xyuas kev noj qab haus huv.Qhov no suav nrog:

○ Muaj ntshav tawm tsam ntshav ua haujlwm:Kev soj xyuas lipids, daim siab enzymes (alt, ast), ntshav ua haujlwm, ntshav suav, thiab cov cim qog nqaij hlav (tab sis cov no feem ntau yog cov ntsuas cov cim tau lig).

○ Kev Ntsuam Xyuas Lub Cev:Tsis tu ncua-}}} Uts nrog tus kws kho mob, kev mob siab, kev hloov pauv, lossis lwm cov cim ceeb toom.

○ Kev Ntsuas:Ua raws li kev ntsuas muaj kev pheej hmoo thiab ntev ntawm kev siv, kev ntsuas lub sijhawm (ultrasound, thiab lwm yam)tej zaumraug txiav txim siab, tab sis qhov no tsis yog kev coj ua thiab tsis hais txog kev pheej hmoo ntawm kev pheej hmoo.

○ Ntev- Term Vigilance:Txoj kev pheej hmoo mob cancer yuav mob siab ntev tom qab ua haujlwm vim yog muaj peev xwm pib ntawm cell. Qhov no tsis yog kev pheej hmoo uas xaus thaum lub sijhawm "kev voj voj voog" nres.

Cov ntaub ntawv kho mob

Hom

Tus hma

Kev Lag Luam Npe

GW501516, Cardarine,Endurobol, GSK-516

Cas

317318-70-0

Tus hniav loj

453.49

Mf

C21H18F3Tsis muaj3S2

Kev coj dawb huv

Saum toj no 98%

Kev tsim nyog

10mg * 100

 

 

Kev xav tau, thov hu rau peb

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Xaus: Cov khoom txhais los ntawm nws txoj kev pheej hmoo

GW501516 (Cardarine) yog lub zog pppen allonist ntawm kev ua kom zoo nkauj ua rau muaj kev sib cav sib ceg Lub 10mg koob tshuaj los ntawm kev txiav txim siab tib neeg metabolic kev sim.

Txawm li cas los xij, nws txhais cov yam ntxwv tsis sib xws: nws yog tus qauv carcinogen hauv cov qauv tsiaj ntawm cov tshuaj cuam tshuam rau tib neeg siv (suav nrog 10mg).Cov ntaub ntawv FDA qhia tau cov qog nqaij ceev ceev hauv ntau lub plab nyob thoob hom. Tsis muaj pov thawj lees paub los qhia kom tib neeg muaj kev tiv thaiv kab mob no; Lub tshuab ntawm carcinogenicity (pparΔ agonism) yog txuag.

While its long half-life (~16-24 hours) allows for convenient once-daily dosing and it requires no traditional PCT as it's non-hormonal, these factors are irrelevant in the face of its profound cancer risk. Cov kev sib tham ntawm nws "cov txiaj ntsig" rau kev ua haujlwm ntawm lub cev yog saib tsis taus thiab negated los ntawm qhov kev tsis tuaj yeem uas tsis tsim nyog. Kev nrhiav kev nrhiav lub cev kom zoo nkauj lossis kev ua tau zoo yeej tsis tsim nyog twv txiaj nrog mob qog noj ntshav.GW501516 belongs nruj me ntsis nyob rau hauv realm kev tshawb fawb, tsis yog nyob rau hauv lub hnab gym.Cov ntaub ntawv uas muaj lub luag haujlwm nthuav tawm yuav tsum ua ntej cov lus kev nyab xeeb zoo tshaj txhua yam.

Cim npe nrov: Stromusc GW501516 (Cardarine) 10Mg rau Cas: 317318-70-0, Suav Teb) 10M318-70-0 Cov Chaw Tsim Tshuaj, Chaw Tsim Tshuaj, Hoobkas

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