
Anastrozole (Arimidex) Powder For Bodybuilding CAS: 120511-73-1
Arimidex belongs rau ib pawg thiab chav kawm ntawm cov tshuaj hu ua aromatase inhibitors (AIs).Aromatase inhibitors belongs rau ntau cov chav kawm dav dav ntawm cov tshuaj hu ua anti-estrogens.Lwm subcategory ntawm cov tshuaj nyob rau hauv pawg anti-estrogen yog hu ua xaiv estrogen receptor modulators. (SERMs), xws li Nolvadex thiab Clomid.
yog dab tsiArimidex?
Arimidex belongs rau qeb thiab chav kawm ntawm cov tshuaj hu ua aromatase inhibitors (AIs).
Aromatase inhibitors muaj nyob rau hauv cov chav kawm dav dav ntawm cov tshuaj hu ua anti-estrogens.
Lwm subcategory ntawm cov tshuaj nyob rau hauv anti-estrogen qeb yog hu ua xaiv estrogen receptor modulators (SERMs), xws li Nolvadex thiab Clomid.
Aromatase inhibitors thiab SERMs tsim cov chav kawm ntawm cov tshuaj tiv thaiv estrogens.
Aromatase inhibitors txawv qhov txawv ntawm SERMs nyob rau hauv lawv ua haujlwm li cas thiab lawv hais txog kev tswj cov tshuaj estrogen.
Nws yog ib qho tseem ceeb kom tshem tawm qhov kev xav tsis zoo uas SERMs zoo li Nolvadex thiab Clomid ua kom txo qis cov tshuaj estrogen.
Qhov no yog ib qho lus dab neeg uas nyuam qhuav pib tuag hauv cov zej zog siv tshuaj anabolic steroid, tab sis nws tseem nyob.
SERMs ua los thaiv cov tshuaj estrogen's receptor site qhov kev txiav txim los ntawm qhov chaw ntawm estrogen, tiv thaiv estrogen nws tus kheej los ntawm exerting nws cov teebmeem nyob rau hauv cov ntaub so ntswg ntawm lub mis los ntawm receptor site binding.
Conversely, SERMs kuj ua raws li estrogen ntawm qhov chaw receptor ntawm lwm lub hlwb nyob rau hauv lwm qhov chaw ntawm lub cev (xws li, lub siab nyob rau hauv cov ntaub ntawv ntawm Nolvadex).
SERMs tsis txo qis cov tshuaj estrogen hauv cov ntshav.
Aromatase inhibitors ua qhov no los ntawm kev tshem tawm cov tshuaj estrogen los ntawm kev khi rau thiab neutralizing aromatase enzyme, cov enzyme uas hloov (los yog aromatizes) androgens rau hauv estrogen.


Daim ntawv thov thiab qhov chaw ntawm Arimidex
Arimidex yog tsim los ua ib qho aromatase inhibitor tsim los ntawm Genentech Pharmaceuticals (tam sim no AstraZeneca) rau kev kho cov poj niam cov neeg mob uas mob qog noj ntshav siab.
Nws tau pom zoo rau kev siv los ntawm FDA thiab tau tshaj tawm rau Asmeskas cov khw muag tshuaj hauv xyoo 1995.
Arimidex yog suav tias yog ib qho ntawm cov tshuaj aromatase tshiab tshaj plaws, lub npe hu ua tus thib peb tiam aromatase inhibitor.
Yog vim li cas aromatase inhibitors thiab SERMs thaiv cov teebmeem ntawm cov tshuaj estrogen nyob rau hauv ntau txoj kev yog vim nws tau pom tias feem ntau cov qog nqaij hlav hauv lub mis tau txhawb nqa thiab txhawb nqa cov tshuaj estrogen.
Arimidex yog lub npe hu ua kev kho mob ntxiv thaum kho mob qog noj ntshav.
Qhov no feem ntau yog ib qho kev kho mob ntxiv uas siv thaum lwm yam kev kho mob tsis tau raws li qhov xav tau.
Ua ntej Arimidex tau tsim thiab tsim los ua kev kho mob cancer mis, cov tshuaj uas tau siv ntau xyoo los kho tus kab mob yog Nolvadex (tamoxifen).
Nolvadex paub tias yuav siv los ua thawj kab thiab kev kho mob rau cov neeg mob qog noj ntshav mis.
Thaum kho mob qog noj ntshav mis, yog tias kev kho mob Nolvadex tsis ua raws li qhov kev cia siab rau ntau yam laj thawj, cov tshuaj thib ob xws li Arimidex tau siv.
Hauv ib txoj kev tshawb fawb ntawm Arimidex uas muaj ntau dua 9, 000 cov poj niam tom qab phais mob cancer mis, nws tau pom tias piv rau Nolvadex (ob leeg ib leeg thiab ua ke), Arimidex tau txais txiaj ntsig zoo dua li Nolvadex.
Txoj kev tshawb no, ua nyob rau xyoo 2002, xaus lus tias Arimidex tau ua haujlwm zoo dua hauv kev kho mob qog noj ntshav thiab tseem ua rau muaj sia nyob ntawm cov neeg mob qog noj ntshav tom qab kho.
Nrog rau qhov no thiab lwm yam kev tshawb fawb, nws tsuas yog ntuj rau lub zej zog anabolic steroid-siv kom ceeb toom ntawm Arimidex thiab pib tshawb nrhiav nws cov tshuaj estrogen muaj zog.
Cov kev tshawb fawb tom qab tau pom tias thaum siv Arimidex txo qhov kev pheej hmoo ntawm mob qog noj ntshav ntawm lub mis los ntawm 40%, cov neeg mob tau ntsib kev puas tsuaj ntxiv.
Qhov no yog vim cov tshuaj estrogen ua lub luag haujlwm tseem ceeb hauv kev saib xyuas cov pob txha thiab pob zeb hauv av kom zoo, uas yog txo qis los ntawm kev txo qis hauv cov tshuaj estrogen los ntawm kev tswj hwm Arimidex.
Arimidex yog qhov feem ntau siv aromatase inhibitor ntawm cov neeg siv tshuaj anabolic steroid rau lub hom phiaj ntawm kev tswj tshuaj estrogen, vim nws yog thawj aromatase inhibitor los rau ntau lub cev tsim.
Nws yog siv los tswj yuav luag txhua yam kev mob tshwm sim ntawm cov tshuaj estrogen ntawm cov neeg ncaws pob uas siv cov tshuaj anabolic steroids, uas yog gynecomastia, dej tuav thiab tsam plab, thiab nce ntshav siab (ib qho tshwm sim ntawm cov tshuaj estrogen-induced nce dej tuav).
Qhov no yog qhov sib piv rau SERMs zoo li Nolvadex, uas tsuas yog ua los thaiv gynecomastia.
Qhov tseeb, cov kev tshawb fawb tau pom tias kev siv Arimidex hauv cov txiv neej muaj txiaj ntsig txaus los txo cov ntshav estrogen los ntawm 50% nrog ib koob tshuaj txhua hnub ntawm 0.5 txog 1 mg.
Thaum qhov no yog qhov txo qis hauv cov txiv neej, thiab qhov sib txawv ntawm 80% txo qis hauv cov poj niam cov neeg mob qog noj ntshav, nws yog ib qho tseem ceeb kom nco ntsoov tias cov tshuaj estrogen thiab poj niam lub cev muaj zog txawv dua li cov txiv neej.
Ntxiv nrog rau nws siv hauv bodybuilders, Arimidex kuj tau siv tshuaj rau cov txiv neej.
Qee tus txiv neej muaj ntau yam tshuaj estrogen txawv txav rau ntau yam laj thawj, thiab Arimidex tau siv los kho cov mob no.
Tshwj xeeb, Arimidex tau siv los kho cov txiv neej hluas uas pom cov tshuaj estrogen ntau dhau thaum lub hnub nyoog laus, ua rau tsis xav pubertal gynecomastia.
Cov tshuaj estrogen ntau dhau ntawm cov txiv neej hluas thaum lub hnub nyoog laus tuaj yeem ua rau muaj kev loj hlob tsis zoo, vim tias tshuaj estrogen ua lub luag haujlwm tseem ceeb hauv kev sib xyaw cov pob txha loj hlob, tiv thaiv kev loj hlob ntxiv, thiab Arimidex kuj tau siv los kho tus mob no.
Chemical Properties ntawm Arimidex
Arimidex yog non-steroidal aromatase inhibitor.
Qhov no txhais tau hais tias nws tsis muaj tus yam ntxwv 4- koom nrog cycloalkane nplhaib carbon qauv uas muaj rau txhua hom steroids.
Cov yam ntxwv ntawm Arimidex
Qhov ua tau zoo ntawm Arimidex hauv kev tswj cov tshuaj estrogen hauv cov ntshav yog qhov tseem ceeb ntawm qhov koob tshuaj 1 mg txhua hnub.
Estrogen suppression ntawm koob tshuaj no tau pom nyob rau hauv ntau dua 80% ntawm cov neeg mob.
Vim tias Arimidex muaj txiaj ntsig zoo ntawm kev txo qis cov tshuaj estrogen los ntawm inhibiting aromatase enzyme, nws feem ntau tsuas yog muab rau cov poj niam tom qab yug menyuam lossis thaum lwm yam kev kho mob thawj zaug rau mob qog noj ntshav tau ua tsis tiav.
Ob leeg Arimidex thiab letrozole yog cais raws li non-steroidal thiab tsis-txhaj tshuaj aromatase inhibitors, uas sib tw nrog substrates rau khi rau lub enzyme active site.
Qhov no txawv heev ntawm aromasin (Exemestane), uas yog ib tug steroidal thiab suicidal aromatase inhibitor raws li ib tug mechanism uas mimics lub substrate thiab yog hloov los ntawm cov enzyme mus rau hauv ib tug reactive intermediate, uas ua rau inactivation ntawm aromatase enzyme.
Nyob rau hauv layman cov ntsiab lus, qhov no txhais tau hais tias aromasin cov tshuaj qauv zoo ib yam li cov tsoos 'cov hom phiaj' uas aromatase khi rau (xws li testosterone), thiab nws tseem ceeb 'tricks' lub aromatase enzyme rau hauv khi rau inhibit / inactivate nws.
Vim tias lub zog khi muaj zog heev, qhov inhibition ntawm aromatase enzyme uas aromasin khi rau yog ruaj khov.
Txij li thaum Arimidex thiab Letrozole yog cov tsis ua kom tuag taus aromatase inhibitors, lawv sib tw nrog cov tsoos 'lub hom phiaj' ntawm cov enzyme es tsis txhob muaj qhov chaw ruaj khov (ib qho zoo ntawm aromasin tshaj ob).
Cov kws tsim lub cev thiab cov neeg ncaws pob uas siv cov tshuaj anabolic steroids nyiam aromatase inhibitors zoo li Arimidex vim tias lawv muaj peev xwm tshem tawm aromatase, uas yog lub hauv paus ua rau nce qib estrogen.
Los ntawm neutralizing cov aromatase enzyme, supraphysiological theem ntawm aromatizable androgens xws li testosterone, dianabol, thiab boldenone tsis hloov mus rau estrogen, tshem tawm cov kev pheej hmoo ntawm cov tshuaj estrogen.
Cov teebmeem ntawm Arimidex
Arimidex (Anastrozole) yog ib qho kev sib xyaw uas feem ntau ua tau zoo los ntawm cov txiv neej cov neeg siv vim tias nws yog ib qho chaw nruab nrab uas lub hom phiaj tswj cov tshuaj estrogen hauv lub cev.
Txawm li cas los xij, muaj qee qhov kev mob tshwm sim Arimidex yuav tsum txhawj xeeb txog.
Cov no feem ntau tuaj nyob rau hauv daim ntawv ntawm kev txo qis hauv plasma qib ntawm cov tshuaj estrogen hauv lub cev thiab cov tshuaj estrogen mus ntev.
Arimidex cuam tshuam rau cov poj niam ntau dua thiab tseem ceeb dua li cov neeg siv txiv neej.
Thaum nws los txog rau kev txo cov tshuaj estrogen thiab kev tawm tsam, nws yog ib qho tseem ceeb kom nkag siab tias tsis zoo li SERMs (xaiv cov tshuaj estrogen receptor modulators) zoo li Nolvadex los yog Clomid (clomiphene citrate), Arimidex belongs rau tsev neeg aromatase inhibitor.
Qhov no txhais tau hais tias nws ua hauj lwm los ntawm neutralizing aromatase enzyme, uas yog lub luag hauj lwm rau lub aromatization los yog hloov dua siab tshiab ntawm testosterone rau hauv estrogen.
Hauv lwm lo lus, tsis zoo li SERMs, uas ua haujlwm los thaiv kev ua haujlwm ntawm cov tshuaj estrogen ntawm cov chaw receptor tshwj xeeb, Arimidex txo qis tag nrho cov tshuaj estrogen hauv cov hauv paus hauv paus.
Cov kev tshawb fawb tau pom tias kev siv Arimidex nce qhov tshwm sim thiab qhov tshwm sim ntawm pob txha.
Thaum qhov no yog ib qho kev mob tshwm sim ntawm poj niam tshwj xeeb ntawm kev siv Arimidex, estrogen kuj tseem ua lub luag haujlwm tseem ceeb hauv kev txhawb nqa thiab tswj cov pob txha ceev hauv cov txiv neej.
Cov kev tshawb fawb tau pom tias txawm tias siv sijhawm luv luv ntawm Arimidex tsis zoo cuam tshuam rau calcium turnover hauv cov pob txha.
Kev qaug zog thiab qaug zog feem ntau cuam tshuam nrog kev siv Arimidex.
Raws li nrog yuav luag tag nrho cov tshuaj estrogen txo cov tebchaw, qhov txo qis hauv cov tshuaj estrogen tuaj yeem ua rau qaug zog ntev vim qhov txo qis hauv lub luag haujlwm tseem ceeb estrogen plays hauv nruab nrab paj hlwb.
Qhov no feem ntau yog qhov tshwm sim ntawm cov tshuaj estrogen raug txo qis rau qib tsis zoo.
Ib qho kev mob tshwm sim tshwj xeeb ntawm kev siv Arimidex yog nws qhov cuam tshuam tsis zoo rau cov ntshav cholesterol.
Zoo li yuav luag txhua cov tshuaj estrogen-txo cov tebchaw, Arimidex txo HDL (zoo) cholesterol thiab nce LDL (phem) cholesterol.
Qhov no yog vim cov tshuaj estrogen yog lub luag haujlwm txhawb kev noj qab haus huv cov roj cholesterol hauv lub cev, thiab qhov kev ua no cuam tshuam thaum cov tshuaj estrogen hauv plasma tsis tswj.
Tau kawg, nws mus yam tsis tau hais tias qhov hnyav dua qhov txo qis hauv cov tshuaj estrogen, qhov cuam tshuam loj dua ntawm cov hlab plawv.
Ib qho ntawm cov kev mob tshwm sim tseem ceeb ntawm Arimidex yog qhov ua tau ntawm estrogen rebound.
Qhov no tshwj xeeb yog tam sim no nrog ob ntawm peb feem ntau siv aromatase inhibitors (Arimidex thiab Letrozole).
Qhov thib peb aromatase inhibitor, aromasin (Exemestane), tsis qhia tib yam khoom ntawm estrogen rebound peev xwm.
Qhov no yog vim hais tias, tsis zoo li aromasin, Arimidex yog ib tug uas tsis yog-tshem aromatase inhibitor.
Ntawd yog, Arimidex khi rau thiab neutralizes aromatase enzyme, tab sis tsis ua tas mus li.
Qee lub sij hawm, Arimidex yuav cuam tshuam los ntawm cov enzyme thiab cov enzyme yuav muaj kev ywj pheej los ua nws txoj haujlwm hauv lub cev dua.
Qhov no txhais tau li cas rau cov neeg siv kawg yog tias yog tias koj tsis siv Arimidex sai dhau los yog sai sai tom qab pib, koj khiav txoj kev pheej hmoo ntawm cov tshuaj estrogen rebounding (thiab yog li cov tshuaj estrogen-txog cov kev mob tshwm sim).
Kev noj tshuaj thiab kev tswj hwm ntawm Arimidex
Kev kho mob, Arimidex (anastrozole) yog siv los kho mob qog noj ntshav hauv cov poj niam postmenopausal qhov twg estrogen tau pom tias yog thawj qhov ua rau.
Hauv cov xwm txheej no, cov koob tshuaj thiab kev tswj hwm ntawm Arimidex yog 1 mg ib hnub ib zaug kom txog thaum mob qog noj ntshav tsis tuaj.
Arimidex ntawm lub voj voog rau gynecomastia thiab estrogen tswj
Rau kev tswj gynecomastia thiab kev tswj hwm ntawm lub voj voog estrogen, Arimidex feem ntau yuav tsum tau siv nyob rau hauv thaj tsam ntawm 0.5 mus rau 1 mg ib hnub twg, uas tuaj yeem hloov kho raws li tus neeg siv lub siab ntev thiab cov lus teb rau qhov sib xyaw.
Txhua tus neeg yuav tsum tau kho lawv cov tshuaj Arimidex raws li lawv tus kheej cov lus teb.
Nws tsis yog qhov tsis yooj yim rau 0.5mg ib hnub twg yuav ntau dhau lossis tsawg dhau rau qee tus neeg.
Koj yuav tsum nco ntsoov nco ntsoov tias lub hom phiaj ntawm no yog tswj cov tshuaj estrogen thaum lub voj voog, tsis yog kom tshem tawm cov tshuaj estrogen tag nrho.
Arimidex rau Post Cycle Therapy (PCT)
Arimidex tau pom nyob rau hauv cov kev tshawb fawb los txhawb endogenous natural testosterone ntau lawm nyob rau hauv cov txiv neej, yog li ib koob ntawm 0.5mg rau 1mg ntawm Arimidex ib hnub twg yog txaus thaum PCT.
Nws tseem ceeb heev kom nkag siab tias Arimidex muaj ib nrab-lub neej ntawm kwv yees li 48 teev, thiab qhov siab tshaj plaws plasma concentrations tuaj yeem ncav cuag tsuas yog tom qab ib lub lim tiam (7 hnub) ntawm kev noj tshuaj zoo ib yam.
Arimidex tuaj yeem noj txhua lub sijhawm ntawm hnub, nrog lossis tsis noj mov.
Cov ntaub ntawv kho mob
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Cov npe lag luam |
Arimidex, Aremed, Anastrazole; anastrozol; ICI-D1033; ZD-1033 |
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CAS |
120511-73-1 |
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Molar loj |
293.374 |
|
Formula |
C17H19N5 |
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Purity |
Tshaj 98% |
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Yam khoom |
Dawb crystalline hmoov |
Txhua yam kev xav tau, thov hu rau peb
Email: Jasonraws106@gmail.com
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Kev cai lij choj thiab muaj nyob ntawm Arimidex
Arimidex yog ib qho khoom siv tsis raug cai hauv ntau lub tebchaws thoob ntiaj teb.
Qhov tshwj xeeb tshaj plaws, hauv Canada thiab Tebchaws Meskas, nws yog cov khoom lag luam nkaus xwb, tab sis vim nws tsis yog cov tshuaj tswj hwm, nws tuaj yeem raug cai, yuav, thiab muaj, tab sis nws tsis muaj nyob hauv lub txee hauv tsev.
Hauv tebchaws United Kingdom, kev cai lij choj ntawm Arimidex yog tib yam.
Hauv ntau lub tebchaws nyob sab hnub tuaj Europe, Asia, thiab Middle East, Arimidex feem ntau muaj yam tsis muaj tshuaj.
Cim npe nrov: Anastrozole (Arimidex) Powder Rau Bodybuilding CAS: 120511-73-1, Tuam Tshoj Anastrozole (Arimidex) hmoov rau lub cev tsim CAS: 120511-73-1 tuam ntxhab, lwm tus muag khoom, Hoobkas
