MK-2866 mimics cov metabolism hauv anabolic ntawm anabolic steroids los ntawm stimulating AR (androgen receptors), ua rau cov leeg pob txha thiab pob txha muaj zog.
MK-2866 kuj tseem txhim kho satellite cell voj voog ua haujlwm, ua rau fusion nrog cov leeg nqaij thiab nce hauv myocyte nuclei hauv cov leeg.
Vim nws cov ntaub so ntswg -cov khoom xaiv, MK-2866 tuaj yeem ua rau cov leeg nqaij ntshiv tsis ua rau androgenic phiv ntawm steroids, thiab yuav pab tiv thaiv benign prostatic hyperplasia (BPH).
Hauv kev tshawb fawb ntawm cov txiv neej thiab poj niam laus, cov neeg koom nrog uas tau noj MK-2866 ntawm koob tshuaj 3 mg / hnub rau 12 lub lis piam tau ntsib 3% nce hauv lub cev hnyav. Qhov no sib npaug rau 80 kg (176 lb) txiv neej nce 2.4 kg (5.3 lb) ntawm cov leeg.
Cov txiaj ntsig no tau txhawb nqa vim tias koob tshuaj siv (3 mg / hnub) tsuas yog ib feem me me ntawm kev txhim kho hauv lub cev muaj pes tsawg leeg pom hauv cov neeg nqa hnyav.
Cov txiv neej thiab cov poj niam laus no kuj tau muaj kev nce siab hauv cov leeg nqaij, nrog rau lawv lub rooj zaum xovxwm nce 22 phaus thaum kawg ntawm 12 lub lis piam.
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